PL3766884T3 - Postać krystaliczna i rodzaj soli związku triazolopirymidynowego oraz sposób jej wytwarzania - Google Patents

Postać krystaliczna i rodzaj soli związku triazolopirymidynowego oraz sposób jej wytwarzania

Info

Publication number
PL3766884T3
PL3766884T3 PL19793622.2T PL19793622T PL3766884T3 PL 3766884 T3 PL3766884 T3 PL 3766884T3 PL 19793622 T PL19793622 T PL 19793622T PL 3766884 T3 PL3766884 T3 PL 3766884T3
Authority
PL
Poland
Prior art keywords
preparation
crystal form
method therefor
salt type
triazolopyrimidine compound
Prior art date
Application number
PL19793622.2T
Other languages
English (en)
Inventor
Kevin X Chen
Yanxin YU
Xinde CHEN
Li Zhang
Zhaoguo CHEN
Cheng Xie
Original Assignee
Medshine Discovery Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Medshine Discovery Inc. filed Critical Medshine Discovery Inc.
Publication of PL3766884T3 publication Critical patent/PL3766884T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PL19793622.2T 2018-04-28 2019-04-28 Postać krystaliczna i rodzaj soli związku triazolopirymidynowego oraz sposób jej wytwarzania PL3766884T3 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CN201810399876 2018-04-28
PCT/CN2019/084822 WO2019206336A1 (zh) 2018-04-28 2019-04-28 一种三唑并嘧啶类化合物的晶型、盐型及其制备方法

Publications (1)

Publication Number Publication Date
PL3766884T3 true PL3766884T3 (pl) 2022-07-18

Family

ID=68294924

Family Applications (1)

Application Number Title Priority Date Filing Date
PL19793622.2T PL3766884T3 (pl) 2018-04-28 2019-04-28 Postać krystaliczna i rodzaj soli związku triazolopirymidynowego oraz sposób jej wytwarzania

Country Status (9)

Country Link
US (1) US11649239B2 (pl)
EP (1) EP3766884B1 (pl)
JP (1) JP7406691B2 (pl)
CN (1) CN112105617B (pl)
DK (1) DK3766884T3 (pl)
ES (1) ES2908424T3 (pl)
PL (1) PL3766884T3 (pl)
PT (1) PT3766884T (pl)
WO (1) WO2019206336A1 (pl)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL3766884T3 (pl) * 2018-04-28 2022-07-18 Medshine Discovery Inc. Postać krystaliczna i rodzaj soli związku triazolopirymidynowego oraz sposób jej wytwarzania
AR116315A1 (es) * 2018-09-12 2021-04-21 Dizal Jiangsu Pharmaceutical Co Ltd Compuestos de triazolo-pirimidina y usos de los mismos
US20220040184A1 (en) * 2018-11-20 2022-02-10 Merck Sharp Dohme Corp. Substituted amino triazolopyrimidine and amino triazolopyrazine adenosine receptor antagonists, pharmaceutical compositions and their use
CA3150766A1 (en) * 2019-08-26 2021-03-04 Incyte Corporation Triazolopyrimidines as a2a / a2b inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4195729B2 (ja) * 1997-03-24 2008-12-10 協和醗酵工業株式会社 [1,2,4]トリアゾロ[1,5−c]ピリミジン誘導体
AR038366A1 (es) * 2001-11-30 2005-01-12 Schering Corp Compuestos de 1,2,4-triazolo [1,5-c] pirimidinas sustituidas, antagonistas del receptor de adenosina a2a, composiciones farmaceuticas, el uso de dichos compuestos para la manufactura de un medicamento para el tratamiento de enfermedades del sistema nervioso central y un kit que comprende combinacion
US20060058320A1 (en) * 2002-09-24 2006-03-16 Kyowa Hakko Kogyo Co., Ltd. [1,2,4] Triazolo[1,5-c]pyrimidine derivatives
PT3611174T (pt) * 2017-04-07 2022-07-07 Medshine Discovery Inc Derivado de [1,2,4]triazolo[1,5-c]pirimidina como inibidor do recetor a2a
PL3766884T3 (pl) * 2018-04-28 2022-07-18 Medshine Discovery Inc. Postać krystaliczna i rodzaj soli związku triazolopirymidynowego oraz sposób jej wytwarzania

Also Published As

Publication number Publication date
EP3766884A1 (en) 2021-01-20
US20210094957A1 (en) 2021-04-01
EP3766884B1 (en) 2022-02-09
DK3766884T3 (da) 2022-03-28
CN112105617B (zh) 2022-04-05
PT3766884T (pt) 2022-03-31
ES2908424T3 (es) 2022-04-29
CN112105617A (zh) 2020-12-18
WO2019206336A1 (zh) 2019-10-31
EP3766884A4 (en) 2021-03-31
JP2021522335A (ja) 2021-08-30
JP7406691B2 (ja) 2023-12-28
US11649239B2 (en) 2023-05-16

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