JP2022000421A5 - - Google Patents

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Publication number
JP2022000421A5
JP2022000421A5 JP2021089538A JP2021089538A JP2022000421A5 JP 2022000421 A5 JP2022000421 A5 JP 2022000421A5 JP 2021089538 A JP2021089538 A JP 2021089538A JP 2021089538 A JP2021089538 A JP 2021089538A JP 2022000421 A5 JP2022000421 A5 JP 2022000421A5
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JP
Japan
Prior art keywords
compound
formula
hydrocarbyl
pharmaceutical composition
same
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021089538A
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English (en)
Japanese (ja)
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JP2022000421A (ja
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Publication date
Priority claimed from US13/940,016 external-priority patent/US10017736B2/en
Application filed filed Critical
Publication of JP2022000421A publication Critical patent/JP2022000421A/ja
Publication of JP2022000421A5 publication Critical patent/JP2022000421A5/ja
Priority to JP2022198455A priority Critical patent/JP7419486B2/ja
Pending legal-status Critical Current

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JP2021089538A 2012-07-13 2021-05-27 τリン酸化を阻害する方法 Pending JP2022000421A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2022198455A JP7419486B2 (ja) 2012-07-13 2022-12-13 τリン酸化を阻害する方法

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201261671235P 2012-07-13 2012-07-13
US61/671,235 2012-07-13
US201361789180P 2013-03-15 2013-03-15
US61/789,180 2013-03-15
US13/940,016 2013-07-11
US13/940,016 US10017736B2 (en) 2012-07-13 2013-07-11 Method of inhibiting tau phosphorylation
JP2018189789A JP2019031520A (ja) 2012-07-13 2018-10-05 τリン酸化を阻害する方法

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2018189789A Division JP2019031520A (ja) 2012-07-13 2018-10-05 τリン酸化を阻害する方法

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2022198455A Division JP7419486B2 (ja) 2012-07-13 2022-12-13 τリン酸化を阻害する方法

Publications (2)

Publication Number Publication Date
JP2022000421A JP2022000421A (ja) 2022-01-04
JP2022000421A5 true JP2022000421A5 (https=) 2022-02-03

Family

ID=49914489

Family Applications (5)

Application Number Title Priority Date Filing Date
JP2015521820A Active JP6417324B2 (ja) 2012-07-13 2013-07-11 τリン酸化を阻害する方法
JP2018000198A Active JP6630374B2 (ja) 2012-07-13 2018-01-04 τリン酸化を阻害する方法
JP2018189789A Pending JP2019031520A (ja) 2012-07-13 2018-10-05 τリン酸化を阻害する方法
JP2021089538A Pending JP2022000421A (ja) 2012-07-13 2021-05-27 τリン酸化を阻害する方法
JP2022198455A Active JP7419486B2 (ja) 2012-07-13 2022-12-13 τリン酸化を阻害する方法

Family Applications Before (3)

Application Number Title Priority Date Filing Date
JP2015521820A Active JP6417324B2 (ja) 2012-07-13 2013-07-11 τリン酸化を阻害する方法
JP2018000198A Active JP6630374B2 (ja) 2012-07-13 2018-01-04 τリン酸化を阻害する方法
JP2018189789A Pending JP2019031520A (ja) 2012-07-13 2018-10-05 τリン酸化を阻害する方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2022198455A Active JP7419486B2 (ja) 2012-07-13 2022-12-13 τリン酸化を阻害する方法

Country Status (6)

Country Link
US (7) US10017736B2 (https=)
EP (1) EP2882428B1 (https=)
JP (5) JP6417324B2 (https=)
DK (1) DK2882428T3 (https=)
ES (1) ES2716049T3 (https=)
WO (1) WO2014011917A2 (https=)

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GB201312499D0 (en) * 2013-07-12 2013-08-28 Isis Innovation Therapeutic compounds
US9433604B2 (en) 2013-10-08 2016-09-06 Pain Therapeutics Inc. Method for inhibiting growth of cancer cells
CN104030933A (zh) * 2014-05-16 2014-09-10 烟台恒迪克能源科技有限公司 一种β-异烷醇基氨基戊酸环己胺的合成方法
MA44037B1 (fr) 2016-06-06 2020-03-31 Arena Pharm Inc Modulateurs du récepteur adrénergique bêta 3 utile dans le traitement ou la prévention de troubles associés à ceux-ci
US11040935B2 (en) 2016-10-05 2021-06-22 University of Pittsburgh—of the Commonwealth System of Higher Education Small molecule AMPK activators
US12186307B2 (en) 2019-02-13 2025-01-07 Yale University Methods of treating epilepsy
CA3131146A1 (en) 2019-02-21 2020-08-27 Pain Therapeutics, Inc. Solid polymorphs of a flna-binding compound and its hydrochloride salts
EP4027987A4 (en) 2019-09-10 2023-11-29 University of Pittsburgh - Of the Commonwealth System of Higher Education Methods and materials for increasing level of phosphorylated ampk protein
JP7721130B2 (ja) * 2020-01-15 2025-08-12 国立大学法人東海国立大学機構 進行性核上性麻痺の治療
WO2022098700A1 (en) * 2020-11-03 2022-05-12 Cassava Sciences, Inc. Inhibiting an immune response mediated by one or more of tlr2, rage, ccr5, cxcr4 and cd4
CN114252324B (zh) * 2022-03-02 2022-05-13 中国人民解放军军事科学院军事医学研究院 一种方便使用的多孔脑片孵育装置
WO2024151661A2 (en) * 2023-01-10 2024-07-18 Washington University Methods of decreasing pathological neuroinflammation

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