JP2021536475A5 - - Google Patents
Info
- Publication number
- JP2021536475A5 JP2021536475A5 JP2021512696A JP2021512696A JP2021536475A5 JP 2021536475 A5 JP2021536475 A5 JP 2021536475A5 JP 2021512696 A JP2021512696 A JP 2021512696A JP 2021512696 A JP2021512696 A JP 2021512696A JP 2021536475 A5 JP2021536475 A5 JP 2021536475A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- group
- needed
- optionally substituted
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862728639P | 2018-09-07 | 2018-09-07 | |
| US62/728,639 | 2018-09-07 | ||
| PCT/US2019/050023 WO2020051503A1 (en) | 2018-09-07 | 2019-09-06 | Alternative processes for the preparation of tubulysins and intermediates thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021536475A JP2021536475A (ja) | 2021-12-27 |
| JP2021536475A5 true JP2021536475A5 (enExample) | 2022-09-14 |
| JP7511543B2 JP7511543B2 (ja) | 2024-07-05 |
Family
ID=68000124
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021512696A Active JP7511543B2 (ja) | 2018-09-07 | 2019-09-06 | チューブリシンおよびそれらの中間体の調製のための代替プロセス |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US20230002440A1 (enExample) |
| EP (1) | EP3847161A1 (enExample) |
| JP (1) | JP7511543B2 (enExample) |
| KR (1) | KR20210073525A (enExample) |
| CN (1) | CN112996778A (enExample) |
| AU (1) | AU2019336231A1 (enExample) |
| BR (1) | BR112021004317A2 (enExample) |
| CA (1) | CA3111149A1 (enExample) |
| EA (1) | EA202190699A1 (enExample) |
| IL (1) | IL281090A (enExample) |
| MA (1) | MA53550A (enExample) |
| MX (1) | MX2021002570A (enExample) |
| SA (1) | SA521421375B1 (enExample) |
| SG (1) | SG11202102126VA (enExample) |
| TW (1) | TWI825169B (enExample) |
| UA (1) | UA128730C2 (enExample) |
| WO (1) | WO2020051503A1 (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2020482800B2 (en) * | 2020-12-23 | 2025-08-21 | Genequantum Healthcare (Suzhou) Co., Ltd. | Novel isomeric compounds comprising a ring-opened thiosuccinimide group, an oligopeptide fragment and a chiral moiety |
| JP2024510435A (ja) | 2021-03-18 | 2024-03-07 | シージェン インコーポレイテッド | 生体活性化合物の内部移行複合体からの選択的薬物放出 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2148886B1 (en) * | 2007-05-10 | 2014-02-19 | R & D Biopharmaceuticals Gmbh | Tubulysine derivatives |
| IT1394860B1 (it) | 2009-07-22 | 2012-07-20 | Kemotech S R L | Composti farmaceutici |
| US11229708B2 (en) | 2015-12-04 | 2022-01-25 | Seagen Inc. | Conjugates of quaternized tubulysin compounds |
| MA50124A (fr) * | 2017-09-08 | 2020-07-15 | Seattle Genetics Inc | Procédé de préparation de tubulysines et d'intermédiaires de celles-ci |
-
2019
- 2019-09-06 KR KR1020217010157A patent/KR20210073525A/ko not_active Withdrawn
- 2019-09-06 JP JP2021512696A patent/JP7511543B2/ja active Active
- 2019-09-06 US US17/273,693 patent/US20230002440A1/en not_active Abandoned
- 2019-09-06 MA MA053550A patent/MA53550A/fr unknown
- 2019-09-06 SG SG11202102126VA patent/SG11202102126VA/en unknown
- 2019-09-06 CN CN201980071734.XA patent/CN112996778A/zh active Pending
- 2019-09-06 MX MX2021002570A patent/MX2021002570A/es unknown
- 2019-09-06 AU AU2019336231A patent/AU2019336231A1/en not_active Abandoned
- 2019-09-06 EA EA202190699A patent/EA202190699A1/ru unknown
- 2019-09-06 BR BR112021004317-9A patent/BR112021004317A2/pt unknown
- 2019-09-06 WO PCT/US2019/050023 patent/WO2020051503A1/en not_active Ceased
- 2019-09-06 TW TW108132162A patent/TWI825169B/zh active
- 2019-09-06 EP EP19773284.5A patent/EP3847161A1/en active Pending
- 2019-09-06 UA UAA202101737A patent/UA128730C2/uk unknown
- 2019-09-06 CA CA3111149A patent/CA3111149A1/en active Pending
-
2021
- 2021-02-24 IL IL281090A patent/IL281090A/en unknown
- 2021-03-03 SA SA521421375A patent/SA521421375B1/ar unknown
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