JP2021534084A5 - - Google Patents

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Publication number
JP2021534084A5
JP2021534084A5 JP2021505646A JP2021505646A JP2021534084A5 JP 2021534084 A5 JP2021534084 A5 JP 2021534084A5 JP 2021505646 A JP2021505646 A JP 2021505646A JP 2021505646 A JP2021505646 A JP 2021505646A JP 2021534084 A5 JP2021534084 A5 JP 2021534084A5
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JP
Japan
Prior art keywords
optionally substituted
optionally
substituted
alkyl
formula
Prior art date
Application number
JP2021505646A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021534084A (ja
JPWO2020033377A5 (https=
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Application filed filed Critical
Priority claimed from PCT/US2019/045259 external-priority patent/WO2020033377A1/en
Publication of JP2021534084A publication Critical patent/JP2021534084A/ja
Publication of JP2021534084A5 publication Critical patent/JP2021534084A5/ja
Publication of JPWO2020033377A5 publication Critical patent/JPWO2020033377A5/ja
Pending legal-status Critical Current

Links

JP2021505646A 2018-08-06 2019-08-06 ヒストンデメチラーゼ5阻害剤およびその使用 Pending JP2021534084A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201862715122P 2018-08-06 2018-08-06
US62/715,122 2018-08-06
US201862715687P 2018-08-07 2018-08-07
US62/715,687 2018-08-07
US201962803332P 2019-02-08 2019-02-08
US62/803,332 2019-02-08
PCT/US2019/045259 WO2020033377A1 (en) 2018-08-06 2019-08-06 Histone demethylase 5 inhibitors and uses thereof

Publications (3)

Publication Number Publication Date
JP2021534084A JP2021534084A (ja) 2021-12-09
JP2021534084A5 true JP2021534084A5 (https=) 2022-08-15
JPWO2020033377A5 JPWO2020033377A5 (https=) 2022-08-15

Family

ID=69414411

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021505646A Pending JP2021534084A (ja) 2018-08-06 2019-08-06 ヒストンデメチラーゼ5阻害剤およびその使用

Country Status (6)

Country Link
US (1) US20230382865A1 (https=)
EP (1) EP3833347A4 (https=)
JP (1) JP2021534084A (https=)
AU (1) AU2019318046B2 (https=)
CA (1) CA3106548A1 (https=)
WO (1) WO2020033377A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11232861B1 (en) 2021-06-18 2022-01-25 Argos Health Inc. Systems and methods for displaying predetermined information for clinical use
WO2024233765A1 (en) * 2023-05-09 2024-11-14 Ohio State Innovation Foundation Therapeutic approach to block terminal exhaustion of t cells and synergize the efficacy of t cell immunotherapies

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9408577D0 (en) * 1994-04-29 1994-06-22 Fujisawa Pharmaceutical Co New compound
BRPI0415179A (pt) * 2003-10-07 2006-11-28 Renovis Inc derivados de amida como ligandos de canal de ìon e composições farmacêuticas e métodos de empregar as mesmas
WO2012162291A1 (en) * 2011-05-24 2012-11-29 The Wistar Institute Compositions and methods for modulating the activity of epstein-barr nuclear antigen 1
RS55764B1 (sr) * 2012-10-02 2017-07-31 Gilead Sciences Inhibitori histonskih demetilaza
CA2901022C (en) * 2013-02-27 2021-05-04 Epitherapeutics Aps Substituted pyridine compounds as inhibitors of histone demethylases
EP3102193B1 (en) * 2014-02-06 2023-01-11 Rutgers, The State University of New Jersey Antibacterial agents: n(alpha)-aroyl-n-aryl-phenylalaninamides
EP3126345A1 (en) * 2014-03-31 2017-02-08 Gilead Sciences, Inc. Inhibitors of histone demethylases
SG11201701182VA (en) * 2014-08-27 2017-03-30 Gilead Sciences Inc Compounds and methods for inhibiting histone demethylases
CN105837575B (zh) * 2015-01-13 2019-01-15 四川大学 3-乙炔基吡唑并嘧啶衍生物及其制备方法和用途

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