JP2021532148A5 - - Google Patents

Info

Publication number
JP2021532148A5
JP2021532148A5 JP2021504360A JP2021504360A JP2021532148A5 JP 2021532148 A5 JP2021532148 A5 JP 2021532148A5 JP 2021504360 A JP2021504360 A JP 2021504360A JP 2021504360 A JP2021504360 A JP 2021504360A JP 2021532148 A5 JP2021532148 A5 JP 2021532148A5
Authority
JP
Japan
Prior art keywords
cancer
compound
disease
derivative
approximately
Prior art date
Application number
JP2021504360A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021532148A (ja
JPWO2020023391A5 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/042827 external-priority patent/WO2020023391A1/en
Publication of JP2021532148A publication Critical patent/JP2021532148A/ja
Publication of JP2021532148A5 publication Critical patent/JP2021532148A5/ja
Publication of JPWO2020023391A5 publication Critical patent/JPWO2020023391A5/ja
Priority to JP2024087006A priority Critical patent/JP2024119868A/ja
Pending legal-status Critical Current

Links

JP2021504360A 2018-07-21 2019-07-22 病態および状態の処置に使用するための、エナンチオマー的に精製されたgperアゴニスト Pending JP2021532148A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024087006A JP2024119868A (ja) 2018-07-21 2024-05-29 病態および状態の処置に使用するための、エナンチオマー的に精製されたgperアゴニスト

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862701726P 2018-07-21 2018-07-21
US62/701,726 2018-07-21
PCT/US2019/042827 WO2020023391A1 (en) 2018-07-21 2019-07-22 Enantiomerically purified gper agonist for use in treating disease states and conditions

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024087006A Division JP2024119868A (ja) 2018-07-21 2024-05-29 病態および状態の処置に使用するための、エナンチオマー的に精製されたgperアゴニスト

Publications (3)

Publication Number Publication Date
JP2021532148A JP2021532148A (ja) 2021-11-25
JP2021532148A5 true JP2021532148A5 (https=) 2022-07-29
JPWO2020023391A5 JPWO2020023391A5 (https=) 2022-07-29

Family

ID=69160978

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021504360A Pending JP2021532148A (ja) 2018-07-21 2019-07-22 病態および状態の処置に使用するための、エナンチオマー的に精製されたgperアゴニスト
JP2024087006A Pending JP2024119868A (ja) 2018-07-21 2024-05-29 病態および状態の処置に使用するための、エナンチオマー的に精製されたgperアゴニスト

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024087006A Pending JP2024119868A (ja) 2018-07-21 2024-05-29 病態および状態の処置に使用するための、エナンチオマー的に精製されたgperアゴニスト

Country Status (23)

Country Link
US (6) US20200024262A1 (https=)
EP (2) EP3823617B1 (https=)
JP (2) JP2021532148A (https=)
KR (1) KR20210049778A (https=)
CN (1) CN112469409B (https=)
AU (1) AU2019310029B2 (https=)
BR (1) BR112021001031A2 (https=)
CA (1) CA3107109A1 (https=)
DK (1) DK3823617T3 (https=)
ES (1) ES2980434T3 (https=)
FI (1) FI3823617T3 (https=)
HR (1) HRP20240661T1 (https=)
HU (1) HUE067185T2 (https=)
IL (2) IL312938A (https=)
LT (1) LT3823617T (https=)
MX (2) MX2021000809A (https=)
NZ (1) NZ771952A (https=)
PL (1) PL3823617T3 (https=)
PT (1) PT3823617T (https=)
RS (1) RS65599B1 (https=)
SI (1) SI3823617T1 (https=)
SM (1) SMT202400205T1 (https=)
WO (1) WO2020023391A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022091029A1 (en) * 2020-10-30 2022-05-05 Resverlogix Corp. Methods for lowering hba1c level with a combination of a bet bromodomain inhibitor and a sodium dependent glucose transport 2 inhibitor
US20240376547A1 (en) * 2021-04-08 2024-11-14 Linnaeus Therapeutics, Inc. Oncologic variations associated with cancer and methods of treatment
WO2022245899A2 (en) * 2021-05-19 2022-11-24 Linaeus Therapeutics, Inc. Diagnostic methods and compositions for treatment of cancer

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US251870A (en) * 1882-01-03 Automatic gate
US6809104B2 (en) * 2001-05-04 2004-10-26 Tularik Inc. Fused heterocyclic compounds
US7875721B2 (en) * 2005-08-04 2011-01-25 Stc.Unm Compounds for binding to ERα/β and GPR30, methods of treating disease states and conditions mediated through these receptors and identification thereof
WO2008153945A2 (en) * 2007-06-06 2008-12-18 University Of South Florida Nutraceutical co-crystal compositions
MX382354B (es) * 2010-11-01 2025-03-13 Celgene Car Llc Compuestos heterocíclicos y usos de los mismos.
US10251870B2 (en) * 2015-03-06 2019-04-09 Stc.Unm Method for treating obesity, diabetes, cardiovascular and kidney diseases by regulating GPR30/GPER activity
AU2016246688B2 (en) * 2015-04-06 2020-11-12 The Trustees Of The University Of Pennsylvania Compositions and methods for decreasing, or preventing or reversing gain of, skin pigmentation in a mammalian subject
US11369618B2 (en) 2016-06-17 2022-06-28 The Trustees Of The University Of Pennsylvania Compounds, compositions and methods for prevention and/or treatment of cancer

Similar Documents

Publication Publication Date Title
KR102744039B1 (ko) 인간 히스톤 메틸트랜스퍼라제 ezh2 억제제의 염 형태
CN104981458B (zh) 组蛋白去甲基化酶抑制剂
CN113354653B (zh) 二芳基大环多晶型物及其制备方法
JP2021532148A5 (https=)
CN103339139A (zh) 组蛋白甲基转移酶的7-氮杂嘌呤调节剂及其使用方法
CN117659051A (zh) Kras g12d蛋白抑制剂和其用途
JP6836693B2 (ja) A2a受容体アンタゴニストとしての縮合環誘導体
HRP20240661T1 (hr) Enantiomerno pročišćeni agonist gper za upotrebu u liječenju bolesti stanja i bolesnih stanja
TW202416964A (zh) 製備激酶抑制劑之方法
KR102588109B1 (ko) 암 치료에 유용한 1-(사이클로) 알킬 피리딘-2-온의 트리사이클릭 융합 유도체
JP2023544173A (ja) 転写活性化タンパク質のイミダゾピペラジン阻害剤
EP3397641A1 (en) 2h-chromeno[2,3-d]pyrimidine-2,4(3h)-diones as nf-kb inhibitors
CA2914282A1 (en) Ethynyl derivatives as metabotropic glutamate receptor antagonists
JPWO2020023391A5 (https=)
AU2021232072A1 (en) STAT inhibitory compounds and compositions
JP2023544732A (ja) 転写活性化タンパク質のイミダゾピペラジン阻害剤
WO2006018955A1 (ja) イソインドール誘導体の製造方法
CN116655497B (zh) 脒类衍生化合物及其制备方法和用途
TW201938154A (zh) 具有抗疼痛活性之鄰苯氧基及鄰苄氧基丙胺基衍生物
CN116589464B (zh) 嘧啶并环类化合物、其制备方法和应用
TW202120095A (zh) 7,8-二氫-4H-吡唑并[4,3-c]氮呯-6-酮化合物
WO2021178841A1 (en) Heterocycle containing stat inhibitors and compositions
WO2021178857A1 (en) Alpha substituted stat inhibitors and compositions thereof
CN117285455A (zh) 2-苯甲酰基吲哚类化合物及其应用
WO2018007957A1 (en) Novel thiazolo[5,4-d]pyrimidine derivatives as inverse agonists of a2a adenosine receptors