JP2021531338A5 - - Google Patents

Info

Publication number
JP2021531338A5
JP2021531338A5 JP2021523581A JP2021523581A JP2021531338A5 JP 2021531338 A5 JP2021531338 A5 JP 2021531338A5 JP 2021523581 A JP2021523581 A JP 2021523581A JP 2021523581 A JP2021523581 A JP 2021523581A JP 2021531338 A5 JP2021531338 A5 JP 2021531338A5
Authority
JP
Japan
Prior art keywords
methyl
amino
dihydropyridine
pyrazole
oxo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021523581A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021531338A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/041699 external-priority patent/WO2020014669A1/en
Publication of JP2021531338A publication Critical patent/JP2021531338A/ja
Publication of JP2021531338A5 publication Critical patent/JP2021531338A5/ja
Priority to JP2025031155A priority Critical patent/JP2025098029A/ja
Pending legal-status Critical Current

Links

JP2021523581A 2018-07-13 2019-07-12 トロンビン阻害薬、製剤、及びそれらの使用 Pending JP2021531338A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025031155A JP2025098029A (ja) 2018-07-13 2025-02-28 トロンビン阻害薬、製剤、及びそれらの使用

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862697817P 2018-07-13 2018-07-13
US62/697,817 2018-07-13
PCT/US2019/041699 WO2020014669A1 (en) 2018-07-13 2019-07-12 Thrombin inhibitors, formulations, and uses thereof

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025031155A Division JP2025098029A (ja) 2018-07-13 2025-02-28 トロンビン阻害薬、製剤、及びそれらの使用

Publications (2)

Publication Number Publication Date
JP2021531338A JP2021531338A (ja) 2021-11-18
JP2021531338A5 true JP2021531338A5 (enExample) 2022-07-20

Family

ID=67470750

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021523581A Pending JP2021531338A (ja) 2018-07-13 2019-07-12 トロンビン阻害薬、製剤、及びそれらの使用
JP2025031155A Pending JP2025098029A (ja) 2018-07-13 2025-02-28 トロンビン阻害薬、製剤、及びそれらの使用

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025031155A Pending JP2025098029A (ja) 2018-07-13 2025-02-28 トロンビン阻害薬、製剤、及びそれらの使用

Country Status (13)

Country Link
US (1) US11865110B2 (enExample)
EP (1) EP3820564A1 (enExample)
JP (2) JP2021531338A (enExample)
KR (1) KR20210080347A (enExample)
CN (1) CN113164765B (enExample)
AU (1) AU2019300161B2 (enExample)
BR (1) BR112021000515A2 (enExample)
CA (1) CA3106359A1 (enExample)
IL (1) IL280078B2 (enExample)
MX (1) MX2021000472A (enExample)
SG (1) SG11202100247WA (enExample)
WO (1) WO2020014669A1 (enExample)
ZA (1) ZA202100955B (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116735514B (zh) * 2023-08-11 2023-11-03 昆明理工大学 纳米酶结合液液微萃取快速检测天麻硫熏标志物的方法
WO2025184627A1 (en) * 2024-03-01 2025-09-04 Cadrenal Therapeutics, Inc. Method for preventing coagulation in patients with implanted cardiac devices

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5579843A (en) 1994-08-16 1996-12-03 Loitherstein; Joel S. Resilient spider for well installation
SE9900070D0 (sv) 1999-01-13 1999-01-13 Astra Ab New use
SI21097A (sl) 2001-12-04 2003-06-30 Univerza V Ljubljani Inhibitorji trombina
SE0200198D0 (sv) 2002-01-23 2002-01-23 Astrazeneca Ab New use
AR061996A1 (es) 2006-07-17 2008-08-10 Boehringer Ingelheim Int Indicaciones para los inhibidores directos de la trombina en el campo cardiovascular
EA201100358A1 (ru) 2008-08-19 2011-10-31 Бёрингер Ингельхайм Интернациональ Гмбх Дабигатран для чрескожной хирургической катетеризации сердца
US20110190352A1 (en) 2008-08-19 2011-08-04 Boehringer Ingelheim International Gmbh Use of dabigatranetexilate for treating patients with pulmonary hypertension
WO2010020601A1 (en) 2008-08-19 2010-02-25 Boehringer Ingelheim International Gmbh Dabigatran in tumour therapy
WO2014145986A1 (en) * 2013-03-15 2014-09-18 Verseon, Inc. Multisubstituted aromatic compounds as serine protease inhibitors
KR20170048410A (ko) * 2014-09-17 2017-05-08 베르선 코포레이션 세린 프로테아제 저해제로서의 피라졸릴-치환된 피리돈 화합물

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