JP2021530559A5 - - Google Patents

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Publication number
JP2021530559A5
JP2021530559A5 JP2021520287A JP2021520287A JP2021530559A5 JP 2021530559 A5 JP2021530559 A5 JP 2021530559A5 JP 2021520287 A JP2021520287 A JP 2021520287A JP 2021520287 A JP2021520287 A JP 2021520287A JP 2021530559 A5 JP2021530559 A5 JP 2021530559A5
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JP
Japan
Prior art keywords
compound according
hydrogen
compound
halogen
pharmaceutically acceptable
Prior art date
Application number
JP2021520287A
Other languages
English (en)
Japanese (ja)
Other versions
JP7373170B2 (ja
JPWO2019246603A5 (https=
JP2021530559A (ja
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Priority claimed from PCT/US2019/038622 external-priority patent/WO2019246603A1/en
Publication of JP2021530559A publication Critical patent/JP2021530559A/ja
Publication of JP2021530559A5 publication Critical patent/JP2021530559A5/ja
Publication of JPWO2019246603A5 publication Critical patent/JPWO2019246603A5/ja
Application granted granted Critical
Publication of JP7373170B2 publication Critical patent/JP7373170B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2021520287A 2018-06-22 2019-06-22 ジヒドロオロト酸デヒドロゲナーゼ阻害のための方法及び組成物 Active JP7373170B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862688612P 2018-06-22 2018-06-22
US62/688,612 2018-06-22
PCT/US2019/038622 WO2019246603A1 (en) 2018-06-22 2019-06-22 Methods and compositions for inhibition of dihydroorotate dehydrogenase

Publications (4)

Publication Number Publication Date
JP2021530559A JP2021530559A (ja) 2021-11-11
JP2021530559A5 true JP2021530559A5 (https=) 2022-06-30
JPWO2019246603A5 JPWO2019246603A5 (https=) 2022-06-30
JP7373170B2 JP7373170B2 (ja) 2023-11-02

Family

ID=68984309

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021520287A Active JP7373170B2 (ja) 2018-06-22 2019-06-22 ジヒドロオロト酸デヒドロゲナーゼ阻害のための方法及び組成物

Country Status (14)

Country Link
US (3) US11312686B2 (https=)
EP (2) EP4438042A3 (https=)
JP (1) JP7373170B2 (https=)
KR (1) KR102821649B1 (https=)
CN (1) CN112672744B (https=)
AU (2) AU2019288813B2 (https=)
BR (1) BR112020026308A2 (https=)
CA (1) CA3103557A1 (https=)
ES (1) ES2994093T3 (https=)
IL (1) IL279586B (https=)
MX (1) MX2021000143A (https=)
SG (1) SG11202012029PA (https=)
WO (1) WO2019246603A1 (https=)
ZA (1) ZA202007620B (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3773579A4 (en) 2018-03-26 2022-03-09 Clear Creek Bio, Inc. COMPOSITIONS AND METHODS FOR INHIBITING DIHYDROOROTATE DEHYDROGENASE
WO2021134045A1 (en) * 2019-12-26 2021-07-01 Ohio State Innovation Foundation Methods and compositions for inhibition of dihydroorotate dehydrogenase in combination with an anti-cd38 therapeutic agent
AU2020411507A1 (en) * 2019-12-26 2022-07-14 Hendrix College Methods and compositions for inhibition of dihydroorotate dehydrogenase
EP4121050A4 (en) * 2020-03-20 2024-04-17 Clear Creek Bio, Inc. STABLE POLYMORPHOUS COMPOSITIONS OF BREQUINA SODIUM, METHODS OF USE AND PRODUCTION THEREOF
US20210300873A1 (en) 2020-03-20 2021-09-30 Clear Creek Bio, Inc. Stable polymorphic compositions of brequinar sodium and methods of use and manufacture thereof
CN113943312A (zh) * 2020-07-17 2022-01-18 轶诺(浙江)药业有限公司 一类肠道裂解型共药及其制备和用途
WO2023278778A1 (en) * 2021-06-30 2023-01-05 Ohio State Innovation Foundation Methods and compositions for inhibition of dihydroorotate dehydrogenase in combination with an anti-cd47-sirpα therapeutic agent
CN115896025B (zh) * 2021-08-20 2025-08-26 合肥中科普瑞昇生物医药科技有限公司 人原代急性髓系白血病细胞的培养基及培养方法
US20250009740A1 (en) * 2021-11-22 2025-01-09 Ohio State Innovation Foundation Methods and compositions for targeting alternative metabolism along with flt3 inhibitor-mediated antileukemic actions
CN115532290B (zh) * 2022-10-13 2024-04-30 浙江昌海制药有限公司 一种特定晶面选择性氢化催化剂及其制备方法和应用
WO2025227007A1 (en) * 2024-04-26 2025-10-30 Ohio State Innovation Foundation Methods and compositions for inhibition of dihydroorotate dehydrogenase

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2888346A (en) * 1955-08-22 1959-05-26 Gen Aniline & Film Corp Ultra-violet absorbing compounds
AU2896097A (en) * 1996-05-10 1997-12-05 Novartis Ag Use of brequinar and derivatives in chronic rejection of allografts and xenotransplantation
JP2003510352A (ja) * 1999-10-01 2003-03-18 インスティチュート オブ モレキュラー アンド セル バイオロジー ウイルス媒介性疾病の治療用化合物
US6841561B1 (en) 1999-10-01 2005-01-11 Institute Of Molecular And Cell Biology Dihydroorotate dehydrogenase inhibitors for the treatment of viral-mediated diseases
HRPK20041072B3 (hr) * 2002-05-17 2007-07-31 Aventis Pharma S.A. Primjena docetaxela/doxorubicina/ciklofosfamida uadjuvantnoj terapiji karcinoma dojke i jajnika
EP2948450A4 (en) 2013-01-28 2016-11-09 Viamet Pharmaceuticals Inc METALLOENZYMINHIBITORVERBINDUNGEN
HRP20181908T1 (hr) 2013-02-25 2019-01-11 Aurigene Discovery Technologies Limited Derivati trosupstituiranog benzotriazola kao inhibitori dihidroorotat oksigenaze
US20190192501A1 (en) * 2016-08-23 2019-06-27 Icahn School Of Medicine At Mount Sinai Methods for treating pten-mutant tumors

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