JP2021525270A5 - - Google Patents
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- JP2021525270A5 JP2021525270A5 JP2020565928A JP2020565928A JP2021525270A5 JP 2021525270 A5 JP2021525270 A5 JP 2021525270A5 JP 2020565928 A JP2020565928 A JP 2020565928A JP 2020565928 A JP2020565928 A JP 2020565928A JP 2021525270 A5 JP2021525270 A5 JP 2021525270A5
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Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2023174642A JP2023168629A (ja) | 2018-05-30 | 2023-10-06 | Ａｘｌ／ｍｅｒ ｒｔｋおよびｃｓｆ１ｒの阻害剤としてのキノリン誘導体 |
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| Application Number | Priority Date | Filing Date | Title |
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| US201862677902P | 2018-05-30 | 2018-05-30 | |
| US62/677,902 | 2018-05-30 | ||
| PCT/EP2019/064214 WO2019229251A1 (en) | 2018-05-30 | 2019-05-31 | Quinoline derivatives as inhibitors of axl/mer rtk and csf1r |
Related Child Applications (1)
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| JP2023174642A Division JP2023168629A (ja) | 2018-05-30 | 2023-10-06 | Ａｘｌ／ｍｅｒ ｒｔｋおよびｃｓｆ１ｒの阻害剤としてのキノリン誘導体 |
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| Publication Number | Publication Date |
|---|---|
| JP2021525270A JP2021525270A (ja) | 2021-09-24 |
| JP2021525270A5 true JP2021525270A5 (enExample) | 2021-12-09 |
| JP7390313B2 JP7390313B2 (ja) | 2023-12-01 |
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| Application Number | Title | Priority Date | Filing Date |
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| JP2020565928A Active JP7390313B2 (ja) | 2018-05-30 | 2019-05-31 | Ａｘｌ／ｍｅｒ ｒｔｋおよびｃｓｆ１ｒの阻害剤としてのキノリン誘導体 |
| JP2023174642A Withdrawn JP2023168629A (ja) | 2018-05-30 | 2023-10-06 | Ａｘｌ／ｍｅｒ ｒｔｋおよびｃｓｆ１ｒの阻害剤としてのキノリン誘導体 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023174642A Withdrawn JP2023168629A (ja) | 2018-05-30 | 2023-10-06 | Ａｘｌ／ｍｅｒ ｒｔｋおよびｃｓｆ１ｒの阻害剤としてのキノリン誘導体 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US12162858B2 (enExample) |
| EP (1) | EP3774776A1 (enExample) |
| JP (2) | JP7390313B2 (enExample) |
| CN (1) | CN112313216B (enExample) |
| AU (1) | AU2019276359B2 (enExample) |
| BR (1) | BR112020021370A2 (enExample) |
| CA (1) | CA3097694A1 (enExample) |
| IL (1) | IL278960B2 (enExample) |
| MX (1) | MX2020011636A (enExample) |
| PH (1) | PH12020551806A1 (enExample) |
| SG (1) | SG11202009971QA (enExample) |
| WO (1) | WO2019229251A1 (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB201905721D0 (en) | 2019-04-24 | 2019-06-05 | Univ Dundee | Compounds |
| IL315474A (en) * | 2022-03-30 | 2024-11-01 | Qurient Co Ltd | New forms of n-(5-((6,7-dimethoxyquinolin-4-yl)oxy)pyridin-2-yl)-1-propyl-4-(2,2,2-trifluoroethoxy)-1h-pyrazole-3 -carboxamide hydrochloride |
| CN117637185B (zh) * | 2024-01-25 | 2024-04-23 | 首都医科大学宣武医院 | 一种基于影像的颅咽管瘤治疗辅助决策方法、系统及设备 |
| CN118593494B (zh) * | 2024-08-08 | 2024-11-01 | 四川大学华西医院 | Nampt抑制剂在制备预防和/或治疗色素沉着绒毛结节性滑膜炎的药物中的用途 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6143764A (en) | 1995-11-07 | 2000-11-07 | Kirin Beer Kabushiki Kaisha | Quinoline and quinazoline derivatives inhibiting platelet-derived growth factor receptor autophosphorylation and pharmaceutical compositions containing the same |
| EP2311809A1 (en) | 2009-10-16 | 2011-04-20 | Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. | Quinolinyloxyphenylsulfonamides |
| EP2423208A1 (en) | 2010-08-28 | 2012-02-29 | Lead Discovery Center GmbH | Pharmaceutically active compounds as Axl inhibitors |
| ES2590778T3 (es) | 2011-02-28 | 2016-11-23 | Calitor Sciences, Llc | Compuestos de quinolina sustituida |
| ES2749726T3 (es) | 2014-12-25 | 2020-03-23 | Ono Pharmaceutical Co | Derivado de quinolina |
| EP3286177B1 (en) * | 2015-04-14 | 2020-05-06 | Qurient Co. Ltd. | Quinoline derivatives as tam rtk inhibitors |
| WO2019231942A1 (en) | 2018-06-01 | 2019-12-05 | Rigel Pharmaceuticals, Inc. | Quinoline derivatives useful as tyrosine kinase inhibitors |
-
2019
- 2019-05-31 AU AU2019276359A patent/AU2019276359B2/en active Active
- 2019-05-31 IL IL278960A patent/IL278960B2/en unknown
- 2019-05-31 US US17/047,961 patent/US12162858B2/en active Active
- 2019-05-31 SG SG11202009971QA patent/SG11202009971QA/en unknown
- 2019-05-31 JP JP2020565928A patent/JP7390313B2/ja active Active
- 2019-05-31 BR BR112020021370-5A patent/BR112020021370A2/pt unknown
- 2019-05-31 WO PCT/EP2019/064214 patent/WO2019229251A1/en not_active Ceased
- 2019-05-31 CN CN201980036560.3A patent/CN112313216B/zh active Active
- 2019-05-31 MX MX2020011636A patent/MX2020011636A/es unknown
- 2019-05-31 CA CA3097694A patent/CA3097694A1/en active Pending
- 2019-05-31 EP EP19728645.3A patent/EP3774776A1/en active Pending
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2020
- 2020-10-29 PH PH12020551806A patent/PH12020551806A1/en unknown
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2023
- 2023-10-06 JP JP2023174642A patent/JP2023168629A/ja not_active Withdrawn
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