JP2021522335A5 - - Google Patents
Info
- Publication number
- JP2021522335A5 JP2021522335A5 JP2021508055A JP2021508055A JP2021522335A5 JP 2021522335 A5 JP2021522335 A5 JP 2021522335A5 JP 2021508055 A JP2021508055 A JP 2021508055A JP 2021508055 A JP2021508055 A JP 2021508055A JP 2021522335 A5 JP2021522335 A5 JP 2021522335A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- crystalline form
- crystal
- pattern shown
- angles
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN201810399876 | 2018-04-28 | ||
| CN201810399876.6 | 2018-04-28 | ||
| PCT/CN2019/084822 WO2019206336A1 (zh) | 2018-04-28 | 2019-04-28 | 一种三唑并嘧啶类化合物的晶型、盐型及其制备方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021522335A JP2021522335A (ja) | 2021-08-30 |
| JP2021522335A5 true JP2021522335A5 (https=) | 2022-05-06 |
| JP7406691B2 JP7406691B2 (ja) | 2023-12-28 |
Family
ID=68294924
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021508055A Active JP7406691B2 (ja) | 2018-04-28 | 2019-04-28 | トリアゾロピリミジン系化合物の結晶形、塩のタイプおよびその調製方法 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US11649239B2 (https=) |
| EP (1) | EP3766884B1 (https=) |
| JP (1) | JP7406691B2 (https=) |
| CN (1) | CN112105617B (https=) |
| DK (1) | DK3766884T3 (https=) |
| ES (1) | ES2908424T3 (https=) |
| PL (1) | PL3766884T3 (https=) |
| PT (1) | PT3766884T (https=) |
| WO (1) | WO2019206336A1 (https=) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL3766884T3 (pl) * | 2018-04-28 | 2022-07-18 | Medshine Discovery Inc. | Postać krystaliczna i rodzaj soli związku triazolopirymidynowego oraz sposób jej wytwarzania |
| AR116315A1 (es) * | 2018-09-12 | 2021-04-21 | Dizal Jiangsu Pharmaceutical Co Ltd | Compuestos de triazolo-pirimidina y usos de los mismos |
| US12414952B2 (en) | 2018-11-20 | 2025-09-16 | Merck Sharp & Dohme Llc | Substituted amino triazolopyrimidine and amino triazolopyrazine adenosine receptor antagonists, pharmaceutical compositions and their use |
| PE20230372A1 (es) * | 2019-08-26 | 2023-03-06 | Incyte Corp | Triazolopirimidinas como inhibidores de a2a/a2b |
| CN120022278A (zh) * | 2023-11-22 | 2025-05-23 | 英诺湖医药(杭州)有限公司 | 用于治疗癌症的化合物 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE69820866T2 (de) | 1997-03-24 | 2004-12-30 | Kyowa Hakko Kogyo Co., Ltd. | [1,2,4]TRIAZOLO[1,5-c]PYRIMIDIN-DERIVATE |
| AR038366A1 (es) | 2001-11-30 | 2005-01-12 | Schering Corp | Compuestos de 1,2,4-triazolo [1,5-c] pirimidinas sustituidas, antagonistas del receptor de adenosina a2a, composiciones farmaceuticas, el uso de dichos compuestos para la manufactura de un medicamento para el tratamiento de enfermedades del sistema nervioso central y un kit que comprende combinacion |
| WO2004029056A1 (ja) | 2002-09-24 | 2004-04-08 | Kyowa Hakko Kogyo Co., Ltd. | [1,2,4]トリアゾロ[1,5−c]ピリミジン誘導体 |
| PL3611174T3 (pl) * | 2017-04-07 | 2022-08-08 | Medshine Discovery Inc. | Pochodne [1,2,4]triazolo[1,5-c]pirymidyny jako inhibitor receptora a2a |
| PL3766884T3 (pl) * | 2018-04-28 | 2022-07-18 | Medshine Discovery Inc. | Postać krystaliczna i rodzaj soli związku triazolopirymidynowego oraz sposób jej wytwarzania |
-
2019
- 2019-04-28 PL PL19793622.2T patent/PL3766884T3/pl unknown
- 2019-04-28 DK DK19793622.2T patent/DK3766884T3/da active
- 2019-04-28 PT PT197936222T patent/PT3766884T/pt unknown
- 2019-04-28 CN CN201980023228.3A patent/CN112105617B/zh active Active
- 2019-04-28 WO PCT/CN2019/084822 patent/WO2019206336A1/zh not_active Ceased
- 2019-04-28 EP EP19793622.2A patent/EP3766884B1/en active Active
- 2019-04-28 JP JP2021508055A patent/JP7406691B2/ja active Active
- 2019-04-28 ES ES19793622T patent/ES2908424T3/es active Active
- 2019-04-28 US US17/044,127 patent/US11649239B2/en active Active
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