JP2020527175A5 - - Google Patents

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JP2020527175A5
JP2020527175A5 JP2020524667A JP2020524667A JP2020527175A5 JP 2020527175 A5 JP2020527175 A5 JP 2020527175A5 JP 2020524667 A JP2020524667 A JP 2020524667A JP 2020524667 A JP2020524667 A JP 2020524667A JP 2020527175 A5 JP2020527175 A5 JP 2020527175A5
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JP2020524667A
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JP2020527175A (ja
JP7067725B2 (ja
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Priority claimed from PCT/CN2018/095973 external-priority patent/WO2019015583A1/en
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JP2020524667A 2017-07-17 2018-07-17 Ａｃｃ阻害剤としての新規な化合物およびそれらの使用 Expired - Fee Related JP7067725B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CNPCT/CN2017/093106 2017-07-17
CNPCT/CN2017/093106 2017-07-17
PCT/CN2018/095973 WO2019015583A1 (en) 2017-07-17 2018-07-17 NOVEL COMPOUNDS AND THEIR USES AS ACC INHIBITORS

Publications (3)

Publication Number Publication Date
JP2020527175A JP2020527175A (ja) 2020-09-03
JP2020527175A5 true JP2020527175A5 (https=) 2021-07-26
JP7067725B2 JP7067725B2 (ja) 2022-05-16

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JP2020524667A Expired - Fee Related JP7067725B2 (ja) 2017-07-17 2018-07-17 Ａｃｃ阻害剤としての新規な化合物およびそれらの使用

Country Status (5)

Country Link
US (1) US10995099B2 (https=)
EP (1) EP3655409B1 (https=)
JP (1) JP7067725B2 (https=)
CN (1) CN111201234A (https=)
WO (2) WO2019015583A1 (https=)

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Publication number Priority date Publication date Assignee Title
TW201910338A (zh) * 2017-07-26 2019-03-16 大陸商南京聖和藥業股份有限公司 作為acc抑制劑的化合物及其應用
EP3995498A4 (en) 2019-07-02 2023-03-01 Sunshine Lake Pharma Co., Ltd. THIENOPYRIMIDI DERIVATIVES WITH STEREO CONFIGURATION AND THEIR USE IN MEDICINE
AR119594A1 (es) * 2019-08-09 2021-12-29 Gilead Sciences Inc Derivados de tienopirimidina como inhibidores acc y usos de los mismos
JP7612682B2 (ja) 2019-10-15 2025-01-14 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規なテトラゾール
CN112778325A (zh) 2019-11-07 2021-05-11 南京瑞捷医药科技有限公司 一种acc抑制剂及其用途
CN116348471B (zh) * 2020-10-14 2025-10-31 勃林格殷格翰国际有限公司 作为trpa1抑制剂的四唑衍生物
AU2021363101A1 (en) * 2020-10-14 2023-03-23 Boehringer Ingelheim International Gmbh Tetrazole derivatives as TRPA1 inhibitors
WO2022166761A1 (zh) * 2021-02-07 2022-08-11 正大天晴药业集团股份有限公司 噻吩并嘧啶衍生物
AU2022257269A1 (en) 2021-04-14 2023-08-17 Boehringer Ingelheim International Gmbh 3H,4H-THIENO[2,3-d]PYRIMIDIN-4-ONE DERIVATIVES AS TRPA1 INHIBITORS
CN114409664B (zh) * 2021-12-24 2023-07-18 河北威远生物化工有限公司 一种螺杂环四氢吡喃化合物及其制备方法和应用
CN114815020B (zh) * 2022-04-21 2023-09-22 岭南师范学院 一种高品质因数折射率传感器的设计方法及折射率传感器
CN116747321B (zh) * 2023-06-14 2025-09-05 厦门君德医药科技有限公司 一种接枝改性的介孔二氧化硅及其制备方法和应用

Family Cites Families (15)

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RS57157B1 (sr) * 2011-11-11 2018-07-31 Gilead Apollo Llc Acc inhibitori i njihove primene
AU2013269662B2 (en) * 2012-05-30 2016-12-15 Bayer Cropscience Ag Compositions comprising a biological control agent and an insecticide
AU2014262547A1 (en) 2013-05-10 2015-11-26 Gilead Apollo, Llc ACC inhibitors and uses thereof
WO2015003879A1 (en) * 2013-07-08 2015-01-15 Syngenta Participations Ag Microbiocidal heterobicylic derivatives
CN106008516A (zh) * 2014-01-29 2016-10-12 苏州晶云药物科技有限公司 依鲁替尼的新晶型及其制备方法
GB201419102D0 (en) * 2014-10-27 2014-12-10 Imp Innovations Ltd Novel compounds
EA201791258A1 (ru) 2015-01-09 2017-12-29 Джилид Аполло, Ллс Комбинированная терапия с применением ингибитора ацетил-коа-карбоксилазы (acc) для лечения неалкогольной жировой болезни печени
CN205115664U (zh) * 2015-10-15 2016-03-30 阳光能源（青海）有限公司 一种用于单晶炉的二次填料装置
CN106137971A (zh) * 2015-11-17 2016-11-23 南京瑞捷医药科技有限公司 一种他克莫司分散体及其缓释组合物及制备方法
PL3380479T3 (pl) * 2015-11-25 2023-05-08 Gilead Apollo, Llc Triazolowe inhibitory acc i ich zastosowania
AU2016361412A1 (en) 2015-11-25 2018-05-24 Gilead Apollo, Llc Pyrazole ACC inhibitors and uses thereof
SG11201807077RA (en) 2016-03-02 2018-09-27 Gilead Apollo Llc Solid forms of a thienopyrimidinedione acc inhibitor and methods for production thereof
CN110382503B (zh) * 2017-03-03 2022-07-19 吉利德科学公司 制备acc抑制剂及其固体形式的方法
CN110709402B (zh) * 2017-06-15 2022-05-10 浙江海正药业股份有限公司 杂芳基并嘧啶酮类衍生物、其制备方法及其在医药上用途
TW201910338A (zh) * 2017-07-26 2019-03-16 大陸商南京聖和藥業股份有限公司 作為acc抑制劑的化合物及其應用

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