JP2020527175A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2020527175A5 JP2020527175A5 JP2020524667A JP2020524667A JP2020527175A5 JP 2020527175 A5 JP2020527175 A5 JP 2020527175A5 JP 2020524667 A JP2020524667 A JP 2020524667A JP 2020524667 A JP2020524667 A JP 2020524667A JP 2020527175 A5 JP2020527175 A5 JP 2020527175A5
- Authority
- JP
- Japan
- Prior art keywords
- compound according
- alkyl
- haloalkyl
- halo
- independently
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CNPCT/CN2017/093106 | 2017-07-17 | ||
| CNPCT/CN2017/093106 | 2017-07-17 | ||
| PCT/CN2018/095973 WO2019015583A1 (en) | 2017-07-17 | 2018-07-17 | NOVEL COMPOUNDS AND THEIR USES AS ACC INHIBITORS |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2020527175A JP2020527175A (ja) | 2020-09-03 |
| JP2020527175A5 true JP2020527175A5 (https=) | 2021-07-26 |
| JP7067725B2 JP7067725B2 (ja) | 2022-05-16 |
Family
ID=65014996
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020524667A Expired - Fee Related JP7067725B2 (ja) | 2017-07-17 | 2018-07-17 | Ａｃｃ阻害剤としての新規な化合物およびそれらの使用 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US10995099B2 (https=) |
| EP (1) | EP3655409B1 (https=) |
| JP (1) | JP7067725B2 (https=) |
| CN (1) | CN111201234A (https=) |
| WO (2) | WO2019015583A1 (https=) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2019020041A1 (zh) * | 2017-07-26 | 2019-01-31 | 南京圣和药业股份有限公司 | 作为acc抑制剂的化合物及其应用 |
| EP3995498A4 (en) | 2019-07-02 | 2023-03-01 | Sunshine Lake Pharma Co., Ltd. | THIENOPYRIMIDI DERIVATIVES WITH STEREO CONFIGURATION AND THEIR USE IN MEDICINE |
| AR119594A1 (es) | 2019-08-09 | 2021-12-29 | Gilead Sciences Inc | Derivados de tienopirimidina como inhibidores acc y usos de los mismos |
| JP7612682B2 (ja) | 2019-10-15 | 2025-01-14 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 新規なテトラゾール |
| CN112778325A (zh) * | 2019-11-07 | 2021-05-11 | 南京瑞捷医药科技有限公司 | 一种acc抑制剂及其用途 |
| JP7565439B2 (ja) * | 2020-10-14 | 2024-10-10 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Ｔｒｐａ１阻害剤としてのテトラゾール誘導体 |
| WO2022079091A1 (en) * | 2020-10-14 | 2022-04-21 | Boehringer Ingelheim International Gmbh | Tetrazole derivatives as trpa1 inhibitors |
| TW202233632A (zh) * | 2021-02-07 | 2022-09-01 | 大陸商正大天晴藥業集團股份有限公司 | 噻吩并嘧啶衍生物 |
| CA3210965A1 (en) | 2021-04-14 | 2022-10-20 | Boehringer Ingelheim International Gmbh | 3h,4h-thieno[2,3-d]pyrimidin-4-one derivatives as trpa1 inhibitors |
| CN114409664B (zh) * | 2021-12-24 | 2023-07-18 | 河北威远生物化工有限公司 | 一种螺杂环四氢吡喃化合物及其制备方法和应用 |
| CN114815020B (zh) * | 2022-04-21 | 2023-09-22 | 岭南师范学院 | 一种高品质因数折射率传感器的设计方法及折射率传感器 |
| CN116747321B (zh) * | 2023-06-14 | 2025-09-05 | 厦门君德医药科技有限公司 | 一种接枝改性的介孔二氧化硅及其制备方法和应用 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| LT2776038T (lt) | 2011-11-11 | 2018-04-25 | Gilead Apollo, Llc | Acc inhibitoriai ir jų panaudojimas |
| NZ701495A (en) * | 2012-05-30 | 2016-11-25 | Bayer Cropscience Ag | Compositions comprising a biological control agent and an insecticide |
| AU2014262547A1 (en) * | 2013-05-10 | 2015-11-26 | Gilead Apollo, Llc | ACC inhibitors and uses thereof |
| WO2015003879A1 (en) * | 2013-07-08 | 2015-01-15 | Syngenta Participations Ag | Microbiocidal heterobicylic derivatives |
| CN103923084B (zh) * | 2014-01-29 | 2016-08-17 | 苏州晶云药物科技有限公司 | 几种晶型及其制备方法 |
| GB201419102D0 (en) * | 2014-10-27 | 2014-12-10 | Imp Innovations Ltd | Novel compounds |
| JP2018501276A (ja) | 2015-01-09 | 2018-01-18 | ギリアド アポロ， エルエルシー | 非アルコール性脂肪肝疾患の処置のためのａｃｃ阻害剤併用療法 |
| CN205115664U (zh) * | 2015-10-15 | 2016-03-30 | 阳光能源（青海）有限公司 | 一种用于单晶炉的二次填料装置 |
| CN106137971A (zh) * | 2015-11-17 | 2016-11-23 | 南京瑞捷医药科技有限公司 | 一种他克莫司分散体及其缓释组合物及制备方法 |
| EP3380479B1 (en) | 2015-11-25 | 2022-12-07 | Gilead Apollo, LLC | Triazole acc inhibitors and uses thereof |
| CA3004796C (en) | 2015-11-25 | 2023-11-14 | Gilead Apollo, Llc | Pyrazole acc inhibitors and uses thereof |
| CN119977993A (zh) | 2016-03-02 | 2025-05-13 | 吉利德阿波罗公司 | 噻吩并嘧啶二酮acc抑制剂的固体形式及其制备方法 |
| EP4273132A3 (en) * | 2017-03-03 | 2024-01-10 | Gilead Sciences, Inc. | Processes for preparing acc inhibitors and solid forms thereof |
| WO2018228369A1 (zh) * | 2017-06-15 | 2018-12-20 | 浙江海正药业股份有限公司 | 杂芳基并嘧啶酮类衍生物、其制备方法及其在医药上用途 |
| WO2019020041A1 (zh) * | 2017-07-26 | 2019-01-31 | 南京圣和药业股份有限公司 | 作为acc抑制剂的化合物及其应用 |
-
2018
- 2018-07-17 WO PCT/CN2018/095973 patent/WO2019015583A1/en not_active Ceased
- 2018-07-17 US US16/631,800 patent/US10995099B2/en active Active
- 2018-07-17 EP EP18835671.1A patent/EP3655409B1/en active Active
- 2018-07-17 JP JP2020524667A patent/JP7067725B2/ja not_active Expired - Fee Related
- 2018-07-17 CN CN201880053983.1A patent/CN111201234A/zh active Pending
-
2019
- 2019-01-14 WO PCT/CN2019/071630 patent/WO2020015343A1/en not_active Ceased