JP2020518621A - 呼吸器疾患の治療のための化合物 - Google Patents

呼吸器疾患の治療のための化合物 Download PDF

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Publication number
JP2020518621A
JP2020518621A JP2019560254A JP2019560254A JP2020518621A JP 2020518621 A JP2020518621 A JP 2020518621A JP 2019560254 A JP2019560254 A JP 2019560254A JP 2019560254 A JP2019560254 A JP 2019560254A JP 2020518621 A JP2020518621 A JP 2020518621A
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compound according
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group
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Japanese (ja)
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JP2020518621A5 (enExample
JPWO2018201192A5 (enExample
Inventor
ウィリアムズ、スペンサー
シャー、サヤリ
ハッキ、ザリヘ
スチュワート、アラステア
Original Assignee
ザ ユニヴァーシティー オブ メルボルン
ザ ユニヴァーシティー オブ メルボルン
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Priority claimed from AU2017901611A external-priority patent/AU2017901611A0/en
Application filed by ザ ユニヴァーシティー オブ メルボルン, ザ ユニヴァーシティー オブ メルボルン filed Critical ザ ユニヴァーシティー オブ メルボルン
Publication of JP2020518621A publication Critical patent/JP2020518621A/ja
Publication of JP2020518621A5 publication Critical patent/JP2020518621A5/ja
Priority to JP2023101906A priority Critical patent/JP2023134493A/ja
Publication of JPWO2018201192A5 publication Critical patent/JPWO2018201192A5/ja
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2019560254A 2017-05-03 2018-05-03 呼吸器疾患の治療のための化合物 Pending JP2020518621A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023101906A JP2023134493A (ja) 2017-05-03 2023-06-21 呼吸器疾患の治療のための化合物

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
AU2017901611 2017-05-03
AU2017901611A AU2017901611A0 (en) 2017-05-03 Compounds for the treatment of respiratory diseases
AU2017901647A AU2017901647A0 (en) 2017-05-05 Compounds for the treatment of respiratory diseases
AU2017901647 2017-05-05
PCT/AU2018/050404 WO2018201192A1 (en) 2017-05-03 2018-05-03 Compounds for the treatment of respiratory diseases

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023101906A Division JP2023134493A (ja) 2017-05-03 2023-06-21 呼吸器疾患の治療のための化合物

Publications (3)

Publication Number Publication Date
JP2020518621A true JP2020518621A (ja) 2020-06-25
JP2020518621A5 JP2020518621A5 (enExample) 2021-05-27
JPWO2018201192A5 JPWO2018201192A5 (enExample) 2025-04-14

Family

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Family Applications (2)

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JP2019560254A Pending JP2020518621A (ja) 2017-05-03 2018-05-03 呼吸器疾患の治療のための化合物
JP2023101906A Pending JP2023134493A (ja) 2017-05-03 2023-06-21 呼吸器疾患の治療のための化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2023101906A Pending JP2023134493A (ja) 2017-05-03 2023-06-21 呼吸器疾患の治療のための化合物

Country Status (8)

Country Link
US (2) US20200079757A1 (enExample)
EP (1) EP3619204B1 (enExample)
JP (2) JP2020518621A (enExample)
CN (1) CN110753688A (enExample)
AU (3) AU2018262108A1 (enExample)
FI (1) FI3619204T3 (enExample)
PT (1) PT3619204T (enExample)
WO (1) WO2018201192A1 (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2022507118A (ja) * 2018-11-07 2022-01-18 ザ ユニヴァーシティー オブ メルボルン 呼吸器疾患の処置のための化合物及び組成物

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10722513B2 (en) 2015-03-23 2020-07-28 The University Of Melbourne Treatment of respiratory diseases
CN110452880B (zh) * 2019-09-09 2021-09-21 温州医科大学附属第一医院 急性肺损伤细胞模型的制备方法及其应用

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH09500137A (ja) * 1993-07-16 1997-01-07 スミスクライン・ビーチャム・コーポレイション 複数の治療特性を有するトリ置換イミダゾール
JPH11513017A (ja) * 1995-06-07 1999-11-09 スミスクライン・ビーチャム・コーポレイション イミダゾール化合物
WO2016149756A1 (en) * 2015-03-23 2016-09-29 The University Of Melbourne Treatment of respiratory diseases

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5593991A (en) * 1993-07-16 1997-01-14 Adams; Jerry L. Imidazole compounds, use and process of making
US5593992A (en) * 1993-07-16 1997-01-14 Smithkline Beecham Corporation Compounds
AU1924699A (en) * 1997-12-19 1999-07-12 Smithkline Beecham Corporation Compounds of heteroaryl substituted imidazole, their pharmaceutical compositionsand uses
JP5784620B2 (ja) * 2009-10-28 2015-09-24 ファイザー・インク カゼインキナーゼ阻害剤としてのイミダゾール誘導体
CZ2012538A3 (cs) * 2012-08-08 2014-02-19 Masarykova Univerzita Inhibitory pro léčbu B-buněčné chronické lymfocytární leukémie

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH09500137A (ja) * 1993-07-16 1997-01-07 スミスクライン・ビーチャム・コーポレイション 複数の治療特性を有するトリ置換イミダゾール
JPH11513017A (ja) * 1995-06-07 1999-11-09 スミスクライン・ビーチャム・コーポレイション イミダゾール化合物
WO2016149756A1 (en) * 2015-03-23 2016-09-29 The University Of Melbourne Treatment of respiratory diseases

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
KIM, DAE-KEE ET AL.: "Synthesis and biological evaluation of trisubstituted imidazole derivatives as inhibitors of p38α m", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 18, JPN6022013598, 2008, pages 4006 - 4010, XP022852885, ISSN: 0004995149, DOI: 10.1016/j.bmcl.2008.06.007 *

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2022507118A (ja) * 2018-11-07 2022-01-18 ザ ユニヴァーシティー オブ メルボルン 呼吸器疾患の処置のための化合物及び組成物
JP2022507117A (ja) * 2018-11-07 2022-01-18 ザ ユニヴァーシティー オブ メルボルン 呼吸器疾患の処理のための新規な化合物
JP7575099B2 (ja) 2018-11-07 2024-10-29 ティアンリ バイオテック プロプライエタリ リミテッド 呼吸器疾患の処理のための新規な化合物
JP7614646B2 (ja) 2018-11-07 2025-01-16 ティアンリ バイオテック プロプライエタリ リミテッド 呼吸器疾患の処置のための化合物及び組成物

Also Published As

Publication number Publication date
AU2024200521B2 (en) 2025-10-02
FI3619204T3 (fi) 2025-11-06
US20200079757A1 (en) 2020-03-12
WO2018201192A1 (en) 2018-11-08
EP3619204B1 (en) 2025-10-01
US20220380343A1 (en) 2022-12-01
EP3619204A1 (en) 2020-03-11
AU2018262108A1 (en) 2019-11-21
JP2023134493A (ja) 2023-09-27
AU2024200521A1 (en) 2024-02-15
AU2022202774A1 (en) 2022-05-19
CN110753688A (zh) 2020-02-04
EP3619204A4 (en) 2021-03-24
PT3619204T (pt) 2025-10-29

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