JP2020510016A - クローン病及び潰瘍性大腸炎を処置する方法 - Google Patents

クローン病及び潰瘍性大腸炎を処置する方法 Download PDF

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Publication number
JP2020510016A
JP2020510016A JP2019548450A JP2019548450A JP2020510016A JP 2020510016 A JP2020510016 A JP 2020510016A JP 2019548450 A JP2019548450 A JP 2019548450A JP 2019548450 A JP2019548450 A JP 2019548450A JP 2020510016 A JP2020510016 A JP 2020510016A
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patient
weeks
pharmaceutically acceptable
upadacitinib
acceptable salt
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Japanese (ja)
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JP2020510016A5 (OSRAM
Inventor
タッカー，ルーパール・ビー
ジュンガーワース，スティーブン
マチャド・デ・ラセルダ，アナ・ポーラ
ロビンソン，アン・エム
エネホサ，ホセ・ジェフリー・ブイ
パンガン，アイリーン・エル
モハメッド，モハメッド−エスラーム
オスマン，アハメド
クリュンダー，ベン
アライアン，アイマン・ディー
ボーチャート，トーマス・ビー
ノルドストローム，フレドリック・ラース
シャイフ，アフマド・ワイ
マルハーン，マシュー・エム
ジャヤンス，ジャヤンシー
マローム，パトリック・ジェイ
メイヤー，ピーター・ティー
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AbbVie Inc
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AbbVie Inc
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Publication of JP2020510016A publication Critical patent/JP2020510016A/ja
Publication of JP2020510016A5 publication Critical patent/JP2020510016A5/ja
Priority to JP2023177288A priority Critical patent/JP2024009963A/ja
Priority to JP2025207808A priority patent/JP2026041823A/ja
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
JP2019548450A 2017-03-09 2018-03-09 クローン病及び潰瘍性大腸炎を処置する方法 Pending JP2020510016A (ja)

Priority Applications (2)

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JP2023177288A JP2024009963A (ja) 2017-03-09 2023-10-13 クローン病及び潰瘍性大腸炎を処置する方法
JP2025207808A JP2026041823A (ja) 2017-03-09 2025-11-28 クローン病及び潰瘍性大腸炎を処置する方法

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US201762469337P 2017-03-09 2017-03-09
US62/469,337 2017-03-09
US201762470565P 2017-03-13 2017-03-13
US62/470,565 2017-03-13
US201762483289P 2017-04-07 2017-04-07
US62/483,289 2017-04-07
US201762593629P 2017-12-01 2017-12-01
US62/593,629 2017-12-01
PCT/US2018/021800 WO2018165581A1 (en) 2017-03-09 2018-03-09 Methods of treating crohn's disease and ulcerative colitis

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JP2023177288A Division JP2024009963A (ja) 2017-03-09 2023-10-13 クローン病及び潰瘍性大腸炎を処置する方法

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JP2020510016A true JP2020510016A (ja) 2020-04-02
JP2020510016A5 JP2020510016A5 (OSRAM) 2021-04-22

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JP2019548450A Pending JP2020510016A (ja) 2017-03-09 2018-03-09 クローン病及び潰瘍性大腸炎を処置する方法
JP2023177288A Pending JP2024009963A (ja) 2017-03-09 2023-10-13 クローン病及び潰瘍性大腸炎を処置する方法
JP2025207808A Pending JP2026041823A (ja) 2017-03-09 2025-11-28 クローン病及び潰瘍性大腸炎を処置する方法

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JP2023177288A Pending JP2024009963A (ja) 2017-03-09 2023-10-13 クローン病及び潰瘍性大腸炎を処置する方法
JP2025207808A Pending JP2026041823A (ja) 2017-03-09 2025-11-28 クローン病及び潰瘍性大腸炎を処置する方法

Country Status (9)

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US (3) US20190046527A1 (OSRAM)
EP (2) EP3592353A1 (OSRAM)
JP (3) JP2020510016A (OSRAM)
CN (2) CN110392572A (OSRAM)
AU (2) AU2018230500B2 (OSRAM)
BR (1) BR112019018576A2 (OSRAM)
MX (2) MX2019010733A (OSRAM)
TW (2) TWI851536B (OSRAM)
WO (2) WO2018165581A1 (OSRAM)

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WO2022178492A1 (en) 2022-08-25
JP2024009963A (ja) 2024-01-23
EP3592353A1 (en) 2020-01-15
EP4487908A2 (en) 2025-01-08
TW201840318A (zh) 2018-11-16
US20210361647A1 (en) 2021-11-25
EP4487908A3 (en) 2025-01-15
TWI851536B (zh) 2024-08-11
CA3052873A1 (en) 2018-09-13
MX2019010733A (es) 2019-11-01
AU2024203642A1 (en) 2024-06-20
MX2022015499A (es) 2023-01-24
CN120661512A (zh) 2025-09-19
WO2018165581A1 (en) 2018-09-13
AU2018230500A1 (en) 2019-09-19
CN110392572A (zh) 2019-10-29
BR112019018576A2 (pt) 2020-04-14
US11607411B2 (en) 2023-03-21
JP2026041823A (ja) 2026-03-10
TW202517269A (zh) 2025-05-01
US20220233527A1 (en) 2022-07-28
AU2024203642B2 (en) 2025-08-21
AU2018230500B2 (en) 2024-03-07
US20190046527A1 (en) 2019-02-14

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