JP2020037517A - ミノキシジルを含有する外用組成物、および、ミノキシジルの析出防止方法 - Google Patents
ミノキシジルを含有する外用組成物、および、ミノキシジルの析出防止方法 Download PDFInfo
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- JP2020037517A JP2020037517A JP2018164395A JP2018164395A JP2020037517A JP 2020037517 A JP2020037517 A JP 2020037517A JP 2018164395 A JP2018164395 A JP 2018164395A JP 2018164395 A JP2018164395 A JP 2018164395A JP 2020037517 A JP2020037517 A JP 2020037517A
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- Prior art keywords
- minoxidil
- composition
- external
- ethyl ether
- external use
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 239000000203 mixture Substances 0.000 title claims abstract description 66
- ZFMITUMMTDLWHR-UHFFFAOYSA-N Minoxidil Chemical compound NC1=[N+]([O-])C(N)=CC(N2CCCCC2)=N1 ZFMITUMMTDLWHR-UHFFFAOYSA-N 0.000 title claims abstract description 54
- 229960003632 minoxidil Drugs 0.000 title claims abstract description 54
- 238000000034 method Methods 0.000 title claims description 8
- 230000003405 preventing effect Effects 0.000 title claims description 5
- 230000008021 deposition Effects 0.000 title abstract 2
- MRAMPOPITCOOIN-VIFPVBQESA-N (2r)-n-(3-ethoxypropyl)-2,4-dihydroxy-3,3-dimethylbutanamide Chemical compound CCOCCCNC(=O)[C@H](O)C(C)(C)CO MRAMPOPITCOOIN-VIFPVBQESA-N 0.000 claims abstract description 20
- 235000010354 butylated hydroxytoluene Nutrition 0.000 claims abstract description 19
- SPSPIUSUWPLVKD-UHFFFAOYSA-N 2,3-dibutyl-6-methylphenol Chemical compound CCCCC1=CC=C(C)C(O)=C1CCCC SPSPIUSUWPLVKD-UHFFFAOYSA-N 0.000 claims abstract description 13
- 238000001556 precipitation Methods 0.000 claims description 19
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- 229920005989 resin Polymers 0.000 claims description 7
- 239000011347 resin Substances 0.000 claims description 7
- ZAKOWWREFLAJOT-CEFNRUSXSA-N D-alpha-tocopherylacetate Chemical compound CC(=O)OC1=C(C)C(C)=C2O[C@@](CCC[C@H](C)CCC[C@H](C)CCCC(C)C)(C)CCC2=C1C ZAKOWWREFLAJOT-CEFNRUSXSA-N 0.000 claims description 5
- ZUFQODAHGAHPFQ-UHFFFAOYSA-N pyridoxine hydrochloride Chemical compound Cl.CC1=NC=C(CO)C(CO)=C1O ZUFQODAHGAHPFQ-UHFFFAOYSA-N 0.000 claims description 5
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- NOOLISFMXDJSKH-UTLUCORTSA-N (+)-Neomenthol Chemical compound CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1O NOOLISFMXDJSKH-UTLUCORTSA-N 0.000 claims 1
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- 239000000725 suspension Substances 0.000 description 2
- BJEPYKJPYRNKOW-REOHCLBHSA-N (S)-malic acid Chemical compound OC(=O)[C@@H](O)CC(O)=O BJEPYKJPYRNKOW-REOHCLBHSA-N 0.000 description 1
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- ZIMGGGWCDYVHOY-UHFFFAOYSA-N 3-hydroxy-2-imino-6-(1-piperidinyl)-4-pyrimidinamine Chemical compound N=C1N(O)C(N)=CC(N2CCCCC2)=N1 ZIMGGGWCDYVHOY-UHFFFAOYSA-N 0.000 description 1
- CYDQOEWLBCCFJZ-UHFFFAOYSA-N 4-(4-fluorophenyl)oxane-4-carboxylic acid Chemical compound C=1C=C(F)C=CC=1C1(C(=O)O)CCOCC1 CYDQOEWLBCCFJZ-UHFFFAOYSA-N 0.000 description 1
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- VEXZGXHMUGYJMC-UHFFFAOYSA-N Hydrochloric acid Chemical compound Cl VEXZGXHMUGYJMC-UHFFFAOYSA-N 0.000 description 1
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Landscapes
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medical Preparation Storing Or Oral Administration Devices (AREA)
- Cosmetics (AREA)
Priority Applications (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2023023902A JP7577774B2 (ja) | 2017-09-04 | 2023-02-20 | ミノキシジルを含有する外用組成物、および、ミノキシジルの析出防止方法 |
| JP2023149731A JP2023169290A (ja) | 2017-09-04 | 2023-09-15 | ミノキシジルを含有する外用組成物、および、ミノキシジルの析出防止方法 |
| JP2024024745A JP7577881B2 (ja) | 2017-09-04 | 2024-02-21 | ミノキシジルを含有する外用組成物、および、ミノキシジルの析出防止方法 |
| JP2024166540A JP2024169680A (ja) | 2017-09-04 | 2024-09-25 | ミノキシジルを含有する外用組成物、および、ミノキシジルの析出防止方法 |
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2017169628 | 2017-09-04 | ||
| JP2017169628 | 2017-09-04 | ||
| JP2018162803 | 2018-08-31 | ||
| JP2018162803 | 2018-08-31 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023023902A Division JP7577774B2 (ja) | 2017-09-04 | 2023-02-20 | ミノキシジルを含有する外用組成物、および、ミノキシジルの析出防止方法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JP2020037517A true JP2020037517A (ja) | 2020-03-12 |
Family
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| JP2023149731A Withdrawn JP2023169290A (ja) | 2017-09-04 | 2023-09-15 | ミノキシジルを含有する外用組成物、および、ミノキシジルの析出防止方法 |
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| JP2023149731A Withdrawn JP2023169290A (ja) | 2017-09-04 | 2023-09-15 | ミノキシジルを含有する外用組成物、および、ミノキシジルの析出防止方法 |
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Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2019131474A (ja) * | 2018-01-29 | 2019-08-08 | 富士化学工業株式会社 | ミノキシジル含有外用組成物 |
| JP2021134164A (ja) * | 2020-02-26 | 2021-09-13 | 東亜薬品株式会社 | ミノキシジル及びパントテニールエチルエーテルを含有する育毛外用剤、並びにそのパントテニールエチルエーテルの安定化及びミノキシジル等の結晶化抑制方法 |
| JP2023161047A (ja) * | 2020-03-27 | 2023-11-02 | ロート製薬株式会社 | 育毛促進用組成物 |
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| JP2020037517A (ja) * | 2017-09-04 | 2020-03-12 | ロート製薬株式会社 | ミノキシジルを含有する外用組成物、および、ミノキシジルの析出防止方法 |
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| JP2002308740A (ja) * | 2001-04-05 | 2002-10-23 | Taisho Pharmaceut Co Ltd | ミノキシジル含有製剤 |
| JP2002326913A (ja) * | 2001-02-27 | 2002-11-15 | Taisho Pharmaceut Co Ltd | 育毛組成物 |
| JP2006022092A (ja) * | 2004-06-09 | 2006-01-26 | Dai Ichi Seiyaku Co Ltd | 新規育毛用組成物 |
| JP2010018555A (ja) * | 2008-07-10 | 2010-01-28 | Taisho Pharmaceutical Co Ltd | ミノキシジル含有液剤 |
| JP2012025770A (ja) * | 2000-04-07 | 2012-02-09 | Taisho Pharmaceutical Co Ltd | 育毛組成物 |
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| JP2017119688A (ja) * | 2015-12-29 | 2017-07-06 | 大正製薬株式会社 | 外用組成物 |
| JP2019073505A (ja) * | 2017-10-12 | 2019-05-16 | ロート製薬株式会社 | 外用組成物 |
| JP2020023467A (ja) * | 2018-01-19 | 2020-02-13 | ロート製薬株式会社 | 外用製剤、液切れ性を改善する方法、および、液切れ性改善剤 |
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| JP2020037517A (ja) | 2017-09-04 | 2020-03-12 | ロート製薬株式会社 | ミノキシジルを含有する外用組成物、および、ミノキシジルの析出防止方法 |
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2023
- 2023-02-20 JP JP2023023902A patent/JP7577774B2/ja active Active
- 2023-09-15 JP JP2023149731A patent/JP2023169290A/ja not_active Withdrawn
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2024
- 2024-02-21 JP JP2024024745A patent/JP7577881B2/ja active Active
- 2024-09-25 JP JP2024166540A patent/JP2024169680A/ja active Pending
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| JP2012025770A (ja) * | 2000-04-07 | 2012-02-09 | Taisho Pharmaceutical Co Ltd | 育毛組成物 |
| JP2002326913A (ja) * | 2001-02-27 | 2002-11-15 | Taisho Pharmaceut Co Ltd | 育毛組成物 |
| JP2002308740A (ja) * | 2001-04-05 | 2002-10-23 | Taisho Pharmaceut Co Ltd | ミノキシジル含有製剤 |
| JP2006022092A (ja) * | 2004-06-09 | 2006-01-26 | Dai Ichi Seiyaku Co Ltd | 新規育毛用組成物 |
| JP2010018555A (ja) * | 2008-07-10 | 2010-01-28 | Taisho Pharmaceutical Co Ltd | ミノキシジル含有液剤 |
| JP2012144536A (ja) * | 2012-02-27 | 2012-08-02 | Taisho Pharmaceutical Co Ltd | ミノキシジル配合育毛剤の着色防止方法 |
| JP2013177471A (ja) * | 2013-06-27 | 2013-09-09 | Taisho Pharmaceutical Co Ltd | ミノキシジル含有製剤 |
| JP2016145179A (ja) * | 2015-02-06 | 2016-08-12 | ダイヤ製薬株式会社 | ミノキシジル含有外用液剤および外用液剤の製造方法 |
| JP2017119688A (ja) * | 2015-12-29 | 2017-07-06 | 大正製薬株式会社 | 外用組成物 |
| JP2019073505A (ja) * | 2017-10-12 | 2019-05-16 | ロート製薬株式会社 | 外用組成物 |
| JP2020023467A (ja) * | 2018-01-19 | 2020-02-13 | ロート製薬株式会社 | 外用製剤、液切れ性を改善する方法、および、液切れ性改善剤 |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2019131474A (ja) * | 2018-01-29 | 2019-08-08 | 富士化学工業株式会社 | ミノキシジル含有外用組成物 |
| JP2021134164A (ja) * | 2020-02-26 | 2021-09-13 | 東亜薬品株式会社 | ミノキシジル及びパントテニールエチルエーテルを含有する育毛外用剤、並びにそのパントテニールエチルエーテルの安定化及びミノキシジル等の結晶化抑制方法 |
| JP2023161047A (ja) * | 2020-03-27 | 2023-11-02 | ロート製薬株式会社 | 育毛促進用組成物 |
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| JP7577774B2 (ja) | 2024-11-05 |
| JP2024169680A (ja) | 2024-12-05 |
| JP2023062102A (ja) | 2023-05-02 |
| JP2023169290A (ja) | 2023-11-29 |
| JP7577881B2 (ja) | 2024-11-05 |
| JP2024050998A (ja) | 2024-04-10 |
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