JP2019516708A5 - - Google Patents
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- JP2019516708A5 JP2019516708A5 JP2018560490A JP2018560490A JP2019516708A5 JP 2019516708 A5 JP2019516708 A5 JP 2019516708A5 JP 2018560490 A JP2018560490 A JP 2018560490A JP 2018560490 A JP2018560490 A JP 2018560490A JP 2019516708 A5 JP2019516708 A5 JP 2019516708A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- catalyst
- halogen
- alkoxy
- aryl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2022118930A JP2022141912A (ja) | 2016-05-19 | 2022-07-26 | 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成 |
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662338562P | 2016-05-19 | 2016-05-19 | |
| US62/338,562 | 2016-05-19 | ||
| US201662416811P | 2016-11-03 | 2016-11-03 | |
| US62/416,811 | 2016-11-03 | ||
| PCT/US2017/033489 WO2017201377A1 (en) | 2016-05-19 | 2017-05-19 | Synthesis of 6-aryl-4-aminopicolinates and 2-aryl-6-aminopyrimidine-4-carboxylates by direct suzuki coupling |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022118930A Division JP2022141912A (ja) | 2016-05-19 | 2022-07-26 | 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2019516708A JP2019516708A (ja) | 2019-06-20 |
| JP2019516708A5 true JP2019516708A5 (https=) | 2020-07-02 |
| JP7113762B2 JP7113762B2 (ja) | 2022-08-05 |
Family
ID=60326419
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018560490A Active JP7113762B2 (ja) | 2016-05-19 | 2017-05-19 | 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成 |
| JP2022118930A Ceased JP2022141912A (ja) | 2016-05-19 | 2022-07-26 | 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022118930A Ceased JP2022141912A (ja) | 2016-05-19 | 2022-07-26 | 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成 |
Country Status (12)
| Country | Link |
|---|---|
| US (3) | US10087164B2 (https=) |
| EP (1) | EP3458442B1 (https=) |
| JP (2) | JP7113762B2 (https=) |
| KR (1) | KR20190007048A (https=) |
| CN (1) | CN109415319A (https=) |
| AU (2) | AU2017268424B2 (https=) |
| BR (1) | BR112018073348B8 (https=) |
| CA (1) | CA3023935A1 (https=) |
| IL (1) | IL263075A (https=) |
| MX (1) | MX2018014174A (https=) |
| RU (1) | RU2018144344A (https=) |
| WO (1) | WO2017201377A1 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2018144344A (ru) * | 2016-05-19 | 2020-06-19 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | Синтез 6-арил-4-аминопиколинатов и 2-арил-6-аминопиримидин-4-карбоксилатов прямым сочетанием сузуки |
| CN113015721B (zh) | 2018-09-19 | 2025-07-25 | 科迪华农业科技有限责任公司 | 毒莠定卤素类似物的制备 |
| WO2020133403A1 (zh) * | 2018-12-29 | 2020-07-02 | 青岛清原化合物有限公司 | 取代的嘧啶芳酯衍生物及其制备方法、除草组合物和应用 |
| BR112022018508A2 (pt) | 2020-03-18 | 2022-10-25 | Corteva Agriscience Llc | Síntese melhorada de 4-amino-6-(heterocíclico)picolinatos |
| US20230174490A1 (en) * | 2020-03-18 | 2023-06-08 | Corteva Agriscience Llc | Improved synthesis of 6-aryl-4-aminopicolinates |
| WO2021231196A1 (en) * | 2020-05-11 | 2021-11-18 | Corteva Agriscience Llc | Preparation of compounds having pesticidal activity |
| WO2023248174A1 (en) * | 2022-06-22 | 2023-12-28 | Hetero Labs Limited | An improved process for preparation of voxelotor |
| CN115819334B (zh) * | 2022-06-28 | 2025-03-18 | 安徽众邦生物工程有限公司 | 一种氯氟吡啶酯的制备方法 |
Family Cites Families (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR037228A1 (es) | 2001-07-30 | 2004-11-03 | Dow Agrosciences Llc | Compuestos del acido 6-(aril o heteroaril)-4-aminopicolinico, composicion herbicida que los comprende y metodo para controlar vegetacion no deseada |
| DE602007008052D1 (de) * | 2006-01-13 | 2010-09-09 | Dow Agrosciences Llc | 2-(polysubstituiertes aryl)-6-amino-5-halogen-4-pyrimidincarbonsäuren und deren verwendung als herbizide |
| WO2009023438A1 (en) * | 2007-08-13 | 2009-02-19 | Dow Agrosciences Llc | 2-(2-fluoro-substituted phenyl)-6-amino-5-chloro-4-pyrimidinecarboxylates and their use as herbicides |
| BRPI0816075A2 (pt) * | 2007-08-30 | 2015-02-24 | Dow Agrosciences Llc | 2-(fenil substituído)-6-amino-5-alcóxi, tioalcóxi e aminoalquil-4-pirimidinacarboxilatos e seus usos como herbicidas |
| HUE030847T2 (hu) | 2007-10-02 | 2017-06-28 | Dow Agrosciences Llc | 2-szubsztituált-6-amino-5-alkil-, alkenil- vagy alkinil-4-pirimidin-karbonsavak és 6-szubsztituált-4-amino-3-alkil-, alkenil- vagy alkinil-pikolinsavak és alkalmazásuk herbicidként |
| BRPI0911207B8 (pt) * | 2008-04-18 | 2022-10-11 | Dow Agrosciences Llc | 2-(fenil substituído)-6-hidróxi ou alcóxi-5-substituído-4-pirimidinacarboxilatos, composição herbicida, e método para controle de vegetação indesejável". |
| GB0808664D0 (en) * | 2008-05-13 | 2008-06-18 | Syngenta Ltd | Chemical compounds |
| GB0902474D0 (en) * | 2009-02-13 | 2009-04-01 | Syngenta Ltd | Chemical compounds |
| GB0907625D0 (en) * | 2009-05-01 | 2009-06-10 | Syngenta Ltd | Method of controlling undesired vegetation |
| HK1201122A1 (en) * | 2011-01-25 | 2015-08-28 | 陶氏益农公司 | 6-amino-2-substituted-5-vinylsilylpyrimidine-4-carboxylic acids and esters and 4-amino-6-substituted-3-vinylsilylpyridine-2-carboxylic acids and esters as herbicides |
| TWI520943B (zh) * | 2011-01-25 | 2016-02-11 | 陶氏農業科學公司 | 用於製備４－胺基－３－氯－５－氟－６－（經取代的）吡啶甲酸酯的方法（二） |
| TWI592401B (zh) * | 2011-01-25 | 2017-07-21 | 陶氏農業科學公司 | 用於製備４－胺基－３－氯－５－氟－６－（經取代的）吡啶甲酸酯的方法（一） |
| TWI529163B (zh) * | 2011-01-25 | 2016-04-11 | 陶氏農業科學公司 | 用於製備４－胺基－５－氟－３－鹵素－６－（經取代之）吡啶甲酸酯的方法 |
| MX370455B (es) * | 2011-07-27 | 2019-12-13 | Bayer Ip Gmbh | Ácidos picolínicos y piridimin-4-carboxílicos sustituidos, procedimiento para su preparación y su uso como herbicidas y reguladores del crecimiento de plantas. |
| US9045502B2 (en) | 2011-12-30 | 2015-06-02 | Dow Agrosciences Llc | Methods of isolating (4-chloro-2-fluoro-3-substituted-phenyl)boronates and methods of using the same |
| EP2797890B1 (en) | 2011-12-30 | 2016-10-05 | Dow AgroSciences LLC | Methods of producing methyl 4-amino-3-chloro-6-(4-chloro-2-fluoro-3-methoxyphenyl)pyridine-2-carboxylate |
| AR091856A1 (es) | 2012-07-24 | 2015-03-04 | Dow Agrosciences Llc | Proceso para la preparacion de 4-amino-5-fluor-3-halo-6-(substituido) picolinatos |
| CN102875456B (zh) * | 2012-10-23 | 2013-12-11 | 西华大学 | 3,6-二氯-2-氨基吡啶的化学合成方法 |
| US20140170058A1 (en) * | 2012-12-13 | 2014-06-19 | Dow Agrosciences Llc | Process for the removal of palladium from 4-amino-3-halo-5-fluoro-6-(aryl) pyridine-2-carboxylates and 4-amino-3-halo-6-(aryl)pyridine-2-carboxylates |
| PL2967057T3 (pl) * | 2013-03-15 | 2019-05-31 | Dow Agrosciences Llc | Nowe karboksylany 4-aminopirydyny i 6-aminopirymidyny jako herbicydy |
| PT2970185T (pt) * | 2013-03-15 | 2023-10-06 | Corteva Agriscience Llc | 4-amino-6-(heterocíclico)picolinatos e 6-amino-2-(heterocíclico)pirimidino-4-carboxilatos e seu uso como herbicidas |
| JP6513073B2 (ja) | 2013-03-15 | 2019-05-15 | ダウ アグロサイエンシィズ エルエルシー | ４−アミノ−６−（複素環式）ピコリネートおよび６−アミノ−２−（複素環式）ピリミジン−４−カルボキシレートならびに除草剤としてのそれらの使用 |
| US9113629B2 (en) | 2013-03-15 | 2015-08-25 | Dow Agrosciences Llc | 4-amino-6-(4-substituted-phenyl)-picolinates and 6-amino-2-(4-substituted-phenyl)-pyrimidine-4-carboxylates and their use as herbicides |
| US9637505B2 (en) | 2013-03-15 | 2017-05-02 | Dow Agrosciences Llc | 4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic)pyrimidine-4-carboxylates and their use as herbicides |
| RU2018144344A (ru) * | 2016-05-19 | 2020-06-19 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | Синтез 6-арил-4-аминопиколинатов и 2-арил-6-аминопиримидин-4-карбоксилатов прямым сочетанием сузуки |
-
2017
- 2017-05-19 RU RU2018144344A patent/RU2018144344A/ru unknown
- 2017-05-19 WO PCT/US2017/033489 patent/WO2017201377A1/en not_active Ceased
- 2017-05-19 MX MX2018014174A patent/MX2018014174A/es unknown
- 2017-05-19 KR KR1020187036364A patent/KR20190007048A/ko not_active Abandoned
- 2017-05-19 BR BR112018073348A patent/BR112018073348B8/pt active IP Right Grant
- 2017-05-19 EP EP17800225.9A patent/EP3458442B1/en active Active
- 2017-05-19 CN CN201780042463.6A patent/CN109415319A/zh active Pending
- 2017-05-19 JP JP2018560490A patent/JP7113762B2/ja active Active
- 2017-05-19 CA CA3023935A patent/CA3023935A1/en active Pending
- 2017-05-19 AU AU2017268424A patent/AU2017268424B2/en not_active Ceased
- 2017-05-19 US US15/599,716 patent/US10087164B2/en active Active
-
2018
- 2018-07-26 US US16/045,901 patent/US10570114B2/en active Active
- 2018-07-26 US US16/045,896 patent/US10544121B2/en active Active
- 2018-11-18 IL IL263075A patent/IL263075A/en unknown
-
2021
- 2021-05-20 AU AU2021203233A patent/AU2021203233A1/en not_active Abandoned
-
2022
- 2022-07-26 JP JP2022118930A patent/JP2022141912A/ja not_active Ceased
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