JP2018530566A5 - - Google Patents

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Publication number
JP2018530566A5
JP2018530566A5 JP2018517867A JP2018517867A JP2018530566A5 JP 2018530566 A5 JP2018530566 A5 JP 2018530566A5 JP 2018517867 A JP2018517867 A JP 2018517867A JP 2018517867 A JP2018517867 A JP 2018517867A JP 2018530566 A5 JP2018530566 A5 JP 2018530566A5
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JP
Japan
Prior art keywords
pharmaceutical composition
composition according
linagliptin
tablets
polymorphic form
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2018517867A
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English (en)
Japanese (ja)
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JP6839708B2 (ja
JP2018530566A (ja
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Publication date
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Priority claimed from PCT/EP2016/073952 external-priority patent/WO2017060398A1/en
Publication of JP2018530566A publication Critical patent/JP2018530566A/ja
Publication of JP2018530566A5 publication Critical patent/JP2018530566A5/ja
Application granted granted Critical
Publication of JP6839708B2 publication Critical patent/JP6839708B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2018517867A 2015-10-09 2016-10-07 8−[(3r)−3−アミノ−1−ピペリジニル]−7−(2−ブチン−1−イル)−3,7−ジヒドロ−3−メチル−1−[4−メチル−2−キナゾリニル)メチル]−1h−プリン−2,6−ジオンまたは薬学上許容できるその塩を含有する医薬組成物 Expired - Fee Related JP6839708B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP15189208 2015-10-09
EP15189208.0 2015-10-09
PCT/EP2016/073952 WO2017060398A1 (en) 2015-10-09 2016-10-07 Pharmaceutical composition containing 8-[(3r)-3-amino-1-piperidinyl]-7-(2-butyn-1-yl)-3,7-dihydro-3-methyl-1-[4-methyl-2-quinazolinyl)methyl]-1h-purine-2,6-dione or a pharmaceutically acceptable salt thereof

Publications (3)

Publication Number Publication Date
JP2018530566A JP2018530566A (ja) 2018-10-18
JP2018530566A5 true JP2018530566A5 (https=) 2019-11-07
JP6839708B2 JP6839708B2 (ja) 2021-03-10

Family

ID=54293102

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2018517867A Expired - Fee Related JP6839708B2 (ja) 2015-10-09 2016-10-07 8−[(3r)−3−アミノ−1−ピペリジニル]−7−(2−ブチン−1−イル)−3,7−ジヒドロ−3−メチル−1−[4−メチル−2−キナゾリニル)メチル]−1h−プリン−2,6−ジオンまたは薬学上許容できるその塩を含有する医薬組成物

Country Status (8)

Country Link
US (1) US10668073B2 (https=)
EP (1) EP3359136A1 (https=)
JP (1) JP6839708B2 (https=)
CN (1) CN108174596A (https=)
AU (1) AU2016335082A1 (https=)
CA (1) CA2998982A1 (https=)
EA (1) EA037498B1 (https=)
WO (1) WO2017060398A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2020009675A2 (en) 2018-06-01 2020-01-09 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Solid oral pharmaceutical compositions of linagliptin
CN110496129B (zh) * 2018-11-23 2021-06-04 北京中医药大学 利拉利汀的抗肿瘤活性及其新用途
JP7245694B2 (ja) * 2019-03-26 2023-03-24 エルメッド株式会社 リナグリプチン含有医薬組成物及びその製造方法、並びにリナグリプチン含有医薬組成物の品質の向上方法
JPWO2022102457A1 (https=) * 2020-11-10 2022-05-19

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1532149B9 (de) 2002-08-21 2011-04-20 Boehringer Ingelheim Pharma GmbH & Co. KG 8-[3-amino-piperidin-1-yl] -xanthine, deren herstellung und deren verwendung als arzneimittel
EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
KR101452915B1 (ko) 2006-05-04 2014-10-21 베링거 인겔하임 인터내셔날 게엠베하 다형태
JP2012512848A (ja) 2008-12-23 2012-06-07 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 有機化合物の塩の形態
US20120258170A1 (en) * 2009-05-20 2012-10-11 Nutracryst Therapeutics Private Limited Pharmaceutical co-crystals of quercetin
CA2835332C (en) 2011-05-10 2019-03-26 Sandoz Ag Polymorph of linagliptin benzoate
CN103006663A (zh) * 2011-09-23 2013-04-03 重庆药友制药有限责任公司 一种瑞舒伐他汀钙的药物组合物
CN102631331A (zh) * 2012-04-26 2012-08-15 北京哈三联科技股份有限公司 奥氮平口腔崩解片制剂及其制备方法
IN2015DN00280A (https=) * 2012-08-13 2015-06-12 Sandoz Ag
WO2014193528A1 (en) * 2013-04-29 2014-12-04 Anovel Pharmaceuticals, Llc Amorphous dosage forms and methods
US20160106679A1 (en) * 2013-05-16 2016-04-21 Sandoz Ag Tablet with increased drug load of odanacatib
EP2848242A1 (en) * 2013-09-12 2015-03-18 Sanovel Ilac Sanayi ve Ticaret A.S. Orally disintegrating formulations of Linagliptin

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