JP2018524337A5 - - Google Patents
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- JP2018524337A5 JP2018524337A5 JP2017567379A JP2017567379A JP2018524337A5 JP 2018524337 A5 JP2018524337 A5 JP 2018524337A5 JP 2017567379 A JP2017567379 A JP 2017567379A JP 2017567379 A JP2017567379 A JP 2017567379A JP 2018524337 A5 JP2018524337 A5 JP 2018524337A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- cycloalkyl
- cyano
- formula
- halogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 125000004093 cyano group Chemical group *C#N 0.000 claims description 36
- 125000000217 alkyl group Chemical group 0.000 claims description 35
- 229910052736 halogen Inorganic materials 0.000 claims description 34
- 150000002367 halogens Chemical class 0.000 claims description 34
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 30
- 150000001875 compounds Chemical class 0.000 claims description 30
- 125000001424 substituent group Chemical group 0.000 claims description 23
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 16
- -1 C 2 -C 6 haloalkynyl Chemical group 0.000 claims description 16
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims description 14
- 125000004770 (C1-C4) haloalkylsulfanyl group Chemical group 0.000 claims description 14
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims description 12
- 229910052717 sulfur Inorganic materials 0.000 claims description 12
- 125000003545 alkoxy group Chemical group 0.000 claims description 10
- 229910052739 hydrogen Inorganic materials 0.000 claims description 10
- 239000001257 hydrogen Substances 0.000 claims description 10
- 125000004435 hydrogen atom Chemical class [H]* 0.000 claims description 10
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims description 8
- 229910052760 oxygen Inorganic materials 0.000 claims description 8
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 7
- 241000607479 Yersinia pestis Species 0.000 claims description 7
- 238000000034 method Methods 0.000 claims description 7
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims description 6
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 6
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims description 6
- 125000001188 haloalkyl group Chemical group 0.000 claims description 6
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims description 6
- 125000000753 cycloalkyl group Chemical group 0.000 claims description 5
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims description 4
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 claims description 4
- 125000001559 cyclopropyl group Chemical group [H]C1([H])C([H])([H])C1([H])* 0.000 claims description 4
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims description 4
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 4
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims description 4
- 150000003839 salts Chemical class 0.000 claims description 4
- 125000004749 (C1-C6) haloalkylsulfinyl group Chemical group 0.000 claims description 3
- 125000004738 (C1-C6) alkyl sulfinyl group Chemical group 0.000 claims description 2
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims description 2
- 125000004740 (C1-C6) haloalkylsulfanyl group Chemical group 0.000 claims description 2
- 125000004741 (C1-C6) haloalkylsulfonyl group Chemical group 0.000 claims description 2
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 claims description 2
- 150000001204 N-oxides Chemical class 0.000 claims description 2
- 239000004480 active ingredient Substances 0.000 claims description 2
- 125000004644 alkyl sulfinyl group Chemical group 0.000 claims description 2
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims description 2
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims description 2
- 239000012752 auxiliary agent Substances 0.000 claims 1
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 description 7
- 125000004414 alkyl thio group Chemical group 0.000 description 3
- 241001465754 Metazoa Species 0.000 description 2
- 125000000232 haloalkynyl group Chemical group 0.000 description 2
- 0 *C(CC1)=CC(*2)=C1N=C2C(*1)=C(CI)C([P+])=C1N=P Chemical compound *C(CC1)=CC(*2)=C1N=C2C(*1)=C(CI)C([P+])=C1N=P 0.000 description 1
- 241000256118 Aedes aegypti Species 0.000 description 1
- 125000004448 alkyl carbonyl group Chemical group 0.000 description 1
- 238000002405 diagnostic procedure Methods 0.000 description 1
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 description 1
- 125000004440 haloalkylsulfinyl group Chemical group 0.000 description 1
- 238000003359 percent control normalization Methods 0.000 description 1
- 230000000361 pesticidal effect Effects 0.000 description 1
- 238000001356 surgical procedure Methods 0.000 description 1
- 238000002560 therapeutic procedure Methods 0.000 description 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP15174759.9 | 2015-07-01 | ||
| EP15174759 | 2015-07-01 | ||
| EP15184066 | 2015-09-07 | ||
| EP15184066.7 | 2015-09-07 | ||
| PCT/EP2016/064778 WO2017001311A1 (en) | 2015-07-01 | 2016-06-27 | Pesticidally active tetracyclic derivatives with sulfur containing substituents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2018524337A JP2018524337A (ja) | 2018-08-30 |
| JP2018524337A5 true JP2018524337A5 (cg-RX-API-DMAC10.html) | 2019-08-08 |
Family
ID=56203411
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017567379A Pending JP2018524337A (ja) | 2015-07-01 | 2016-06-27 | 硫黄含有置換基を有する有害生物防除に活性な四環式誘導体 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US10202380B2 (cg-RX-API-DMAC10.html) |
| EP (1) | EP3317275B1 (cg-RX-API-DMAC10.html) |
| JP (1) | JP2018524337A (cg-RX-API-DMAC10.html) |
| CN (1) | CN107810186B (cg-RX-API-DMAC10.html) |
| BR (1) | BR112018000052A2 (cg-RX-API-DMAC10.html) |
| ES (1) | ES2762958T3 (cg-RX-API-DMAC10.html) |
| WO (1) | WO2017001311A1 (cg-RX-API-DMAC10.html) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2017144341A1 (de) * | 2016-02-23 | 2017-08-31 | Bayer Cropscience Aktiengesellschaft | Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel |
| MX2018010872A (es) | 2016-03-10 | 2019-02-07 | Nissan Chemical Corp | Compuestos heterociclicos condensados y pesticidas. |
| MX2019012728A (es) * | 2017-04-24 | 2020-01-23 | Bayer Ag | Derivados de heterociclos biciclicos fusionados como plaguicidas. |
| KR102600330B1 (ko) | 2017-08-22 | 2023-11-10 | 바이엘 악티엔게젤샤프트 | 해충 방제제로서의 헤테로시클렌 유도체 |
| CN111741958A (zh) | 2018-02-21 | 2020-10-02 | 拜耳公司 | 作为害虫防治剂的稠合双环杂环衍生物 |
| EP3765466B1 (de) * | 2018-03-12 | 2022-05-25 | Bayer Aktiengesellschaft | Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel |
| WO2019219689A1 (en) | 2018-05-18 | 2019-11-21 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfoximine containing substituents |
| MX2021002949A (es) | 2018-09-13 | 2021-05-12 | Bayer Ag | Derivados heterociclicos como plaguicidas. |
| ES2974634T3 (es) | 2018-12-21 | 2024-06-28 | Celgene Corp | Inhibidores de tienopiridinas de RIPK2 |
| AR119140A1 (es) | 2019-06-13 | 2021-11-24 | Pi Industries Ltd | Compuestos heterocíclicos fusionados y su uso como agentes de control de plagas |
| AR120982A1 (es) | 2020-01-06 | 2022-04-06 | Syngenta Crop Protection Ag | Derivados heterocíclicos activos como plaguicidas con sustituyentes que contienen azufre |
| CN120882309A (zh) | 2023-03-14 | 2025-10-31 | 先正达农作物保护股份公司 | 对杀昆虫剂具有抗性的有害生物的控制 |
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| CA1340685C (en) | 1988-07-29 | 1999-07-27 | Frederick Meins | Dna sequences encoding polypeptides having beta-1,3-glucanase activity |
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| EP0392225B1 (en) | 1989-03-24 | 2003-05-28 | Syngenta Participations AG | Disease-resistant transgenic plants |
| GB8910624D0 (en) | 1989-05-09 | 1989-06-21 | Ici Plc | Bacterial strains |
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| US5639949A (en) | 1990-08-20 | 1997-06-17 | Ciba-Geigy Corporation | Genes for the synthesis of antipathogenic substances |
| UA48104C2 (uk) | 1991-10-04 | 2002-08-15 | Новартіс Аг | Фрагмент днк, який містить послідовність,що кодує інсектицидний протеїн, оптимізовану для кукурудзи,фрагмент днк, який забезпечує направлену бажану для серцевини стебла експресію зв'язаного з нею структурного гена в рослині, фрагмент днк, який забезпечує специфічну для пилку експресію зв`язаного з нею структурного гена в рослині, рекомбінантна молекула днк, спосіб одержання оптимізованої для кукурудзи кодуючої послідовності інсектицидного протеїну, спосіб захисту рослин кукурудзи щонайменше від однієї комахи-шкідника |
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| WO2000015615A1 (en) | 1998-09-15 | 2000-03-23 | Syngenta Participations Ag | Pyridine ketones useful as herbicides |
| WO2002015701A2 (en) | 2000-08-25 | 2002-02-28 | Syngenta Participations Ag | Bacillus thuringiensis crystal protein hybrids |
| JP3789749B2 (ja) | 2000-12-19 | 2006-06-28 | エア・ウォーター・ケミカル株式会社 | チオサリチル酸の製造方法 |
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| TWI528899B (zh) | 2010-12-29 | 2016-04-11 | 杜邦股份有限公司 | 中離子性殺蟲劑 |
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| WO2013191113A1 (ja) | 2012-06-18 | 2013-12-27 | 住友化学株式会社 | 縮合複素環化合物 |
| JP6677637B2 (ja) * | 2013-07-02 | 2020-04-08 | シンジェンタ パーティシペーションズ アーゲー | 有害生物防除的に活性な、硫黄含有置換基を有する二環式または三環式複素環 |
| CN107428743A (zh) * | 2015-03-12 | 2017-12-01 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性四环衍生物 |
| US10323031B2 (en) * | 2015-03-12 | 2019-06-18 | Syngenta Participations Ag | Pesticidally active tetracyclic derivatives with sulfur containing substituents |
| WO2016169882A1 (en) * | 2015-04-24 | 2016-10-27 | Syngenta Participations Ag | Pesticidally active polycyclic derivatives with sulfur substituted five membered ring heterocyles |
-
2016
- 2016-06-27 ES ES16731935T patent/ES2762958T3/es active Active
- 2016-06-27 EP EP16731935.9A patent/EP3317275B1/en active Active
- 2016-06-27 CN CN201680038616.5A patent/CN107810186B/zh not_active Expired - Fee Related
- 2016-06-27 WO PCT/EP2016/064778 patent/WO2017001311A1/en not_active Ceased
- 2016-06-27 BR BR112018000052-3A patent/BR112018000052A2/pt not_active Application Discontinuation
- 2016-06-27 JP JP2017567379A patent/JP2018524337A/ja active Pending
- 2016-06-27 US US15/732,804 patent/US10202380B2/en not_active Expired - Fee Related