JP2018514568A - テトラヒドロナフチリジニルプロピオン酸誘導体およびその使用法 - Google Patents
テトラヒドロナフチリジニルプロピオン酸誘導体およびその使用法 Download PDFInfo
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- Biomedical Technology (AREA)
- Physical Education & Sports Medicine (AREA)
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| US201562154894P | 2015-04-30 | 2015-04-30 | |
| US62/154,894 | 2015-04-30 | ||
| PCT/US2016/029962 WO2016176532A1 (en) | 2015-04-30 | 2016-04-29 | Tetrahydronaphthyridinyl propionic acid derivatives and uses thereof |
Publications (2)
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| JP2018514568A true JP2018514568A (ja) | 2018-06-07 |
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| EP (1) | EP3288555A1 (enExample) |
| JP (1) | JP2018514568A (enExample) |
| KR (1) | KR20170141757A (enExample) |
| CN (1) | CN108040467A (enExample) |
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2021529755A (ja) * | 2018-06-27 | 2021-11-04 | プライアント・セラピューティクス・インコーポレイテッドＰｌｉａｎｔ Ｔｈｅｒａｐｅｕｔｉｃｓ， Ｉｎｃ． | 非分岐リンカーを伴うアミノ酸化合物およびその使用方法 |
| JP2022053156A (ja) * | 2020-09-24 | 2022-04-05 | 株式会社ファンケル | セラミド含有ニオソームを含む化粧料 |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
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| US8901144B2 (en) * | 2013-02-07 | 2014-12-02 | Scifluor Life Sciences, Llc | Fluorinated 3-(2-oxo-3-(3-arylpropyl)imidazolidin-1-yl)-3-arylpropanoic acid derivatives |
| WO2014124302A1 (en) | 2013-02-07 | 2014-08-14 | Scifluor Life Sciences, Llc | Fluorinated integrin antagonists |
| JP2018510139A (ja) | 2015-02-19 | 2018-04-12 | サイフルーア ライフ サイエンシズ インコーポレイテッド | フッ化テトラヒドロナフチリジニルノナン酸誘導体およびその使用法 |
| WO2017189828A1 (en) | 2016-04-27 | 2017-11-02 | Scifluor Life Sciences, Inc. | Nonanoic and decanoic acid derivatives and uses thereof |
| MX394210B (es) | 2017-02-28 | 2025-03-04 | Morphic Therapeutic Inc | INHIBIDORES DE INTEGRINA AVß6. |
| CA3054792A1 (en) | 2017-02-28 | 2018-09-07 | Morphic Therapeutic, Inc. | Inhibitors of .alpha.v.beta.6 integrin |
| ES2983950T3 (es) * | 2018-04-27 | 2024-10-28 | Arrowhead Pharmaceuticals Inc | Ligandos dirigidos a integrinas y usos de los mismos |
| JP7540998B2 (ja) | 2018-08-29 | 2024-08-27 | モーフィック セラピューティック，インコーポレイテッド | αｖβ６インテグリンの阻害 |
| WO2021225912A1 (en) * | 2020-05-07 | 2021-11-11 | Pliant Therapeutics, Inc. | Treatment of respiratory diseases with amino acid compounds |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1318254C (en) | 1988-01-06 | 1993-05-25 | Munehiro Tomikawa | Inhibitory agent of hepatic fibrosis containing pantethine |
| JPH06506471A (ja) | 1991-04-01 | 1994-07-21 | デューク ユニバーシティー | 繊維症阻害法 |
| JP3818322B2 (ja) | 1994-04-28 | 2006-09-06 | 敏一 中村 | コラーゲン分解促進剤 |
| US5645839A (en) | 1995-06-07 | 1997-07-08 | Trustees Of Boston University | Combined use of angiotensin inhibitors and nitric oxide stimulators to treat fibrosis |
| US6664227B1 (en) | 1996-03-01 | 2003-12-16 | Genetics Institute, Llc | Treatment of fibrosis by antagonism of IL-13 and IL-13 receptor chains |
| AU3215597A (en) | 1996-08-30 | 1998-03-19 | Biomeasure Incorporated | Method of inhibiting fibrosis with a somatostatin agonist |
| CN1284955A (zh) * | 1997-12-17 | 2001-02-21 | 麦克公司 | 整联蛋白受体拮抗剂 |
| US6017926A (en) | 1997-12-17 | 2000-01-25 | Merck & Co., Inc. | Integrin receptor antagonists |
| US6117445A (en) | 1998-01-28 | 2000-09-12 | Link Technology Inc. | Methods for the prevention and treatment of fibrosis and sclerosis |
| KR20010108519A (ko) | 2000-02-22 | 2001-12-07 | 도리이 신이치로 | 키마제 억제제를 유효성분으로 하는 선유증의 예방 또는치료약 |
| WO2002022615A1 (en) | 2000-09-14 | 2002-03-21 | Merck & Co., Inc. | Alpha v integrin receptor antagonists |
| US6509347B2 (en) * | 2001-06-11 | 2003-01-21 | Merck & Co., Inc. | Crystalline forms of an integrin receptor antagonist |
| WO2014124302A1 (en) | 2013-02-07 | 2014-08-14 | Scifluor Life Sciences, Llc | Fluorinated integrin antagonists |
| US8901144B2 (en) | 2013-02-07 | 2014-12-02 | Scifluor Life Sciences, Llc | Fluorinated 3-(2-oxo-3-(3-arylpropyl)imidazolidin-1-yl)-3-arylpropanoic acid derivatives |
| JP2018510139A (ja) * | 2015-02-19 | 2018-04-12 | サイフルーア ライフ サイエンシズ インコーポレイテッド | フッ化テトラヒドロナフチリジニルノナン酸誘導体およびその使用法 |
| WO2016154369A1 (en) * | 2015-03-26 | 2016-09-29 | Merck Sharp & Dohme Corp. | Composition and methods for treating chronic kidney disease |
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2016
- 2016-04-29 US US15/142,023 patent/US9572801B2/en not_active Expired - Fee Related
- 2016-04-29 EP EP16724172.8A patent/EP3288555A1/en not_active Withdrawn
- 2016-04-29 JP JP2017556988A patent/JP2018514568A/ja not_active Withdrawn
- 2016-04-29 RU RU2017141561A patent/RU2017141561A/ru not_active Application Discontinuation
- 2016-04-29 KR KR1020177034091A patent/KR20170141757A/ko not_active Withdrawn
- 2016-04-29 AU AU2016255494A patent/AU2016255494A1/en not_active Abandoned
- 2016-04-29 WO PCT/US2016/029962 patent/WO2016176532A1/en not_active Ceased
- 2016-04-29 MX MX2017013880A patent/MX2017013880A/es unknown
- 2016-04-29 CN CN201680036759.2A patent/CN108040467A/zh active Pending
- 2016-04-29 CA CA2983312A patent/CA2983312A1/en not_active Abandoned
- 2016-04-29 BR BR112017023432A patent/BR112017023432A2/pt not_active Application Discontinuation
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2017
- 2017-10-16 IL IL255054A patent/IL255054A0/en unknown
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2021529755A (ja) * | 2018-06-27 | 2021-11-04 | プライアント・セラピューティクス・インコーポレイテッドＰｌｉａｎｔ Ｔｈｅｒａｐｅｕｔｉｃｓ， Ｉｎｃ． | 非分岐リンカーを伴うアミノ酸化合物およびその使用方法 |
| JP7425757B2 (ja) | 2018-06-27 | 2024-01-31 | プライアント・セラピューティクス・インコーポレイテッド | 非分岐リンカーを伴うアミノ酸化合物およびその使用方法 |
| JP2022053156A (ja) * | 2020-09-24 | 2022-04-05 | 株式会社ファンケル | セラミド含有ニオソームを含む化粧料 |
| JP7585564B2 (ja) | 2020-09-24 | 2024-11-19 | 株式会社ファンケル | セラミド含有ニオソームを含む化粧料 |
Also Published As
| Publication number | Publication date |
|---|---|
| BR112017023432A2 (pt) | 2018-07-24 |
| RU2017141561A (ru) | 2019-05-31 |
| IL255054A0 (en) | 2017-12-31 |
| US9572801B2 (en) | 2017-02-21 |
| KR20170141757A (ko) | 2017-12-26 |
| EP3288555A1 (en) | 2018-03-07 |
| MX2017013880A (es) | 2018-08-01 |
| CA2983312A1 (en) | 2016-11-03 |
| US20160317527A1 (en) | 2016-11-03 |
| CN108040467A (zh) | 2018-05-15 |
| AU2016255494A1 (en) | 2017-11-02 |
| RU2017141561A3 (enExample) | 2019-09-25 |
| WO2016176532A1 (en) | 2016-11-03 |
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