JP2018513123A - Rorガンマ阻害剤を用いてがんを治療するための方法 - Google Patents

Rorガンマ阻害剤を用いてがんを治療するための方法 Download PDF

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JP2018513123A
JP2018513123A JP2017547968A JP2017547968A JP2018513123A JP 2018513123 A JP2018513123 A JP 2018513123A JP 2017547968 A JP2017547968 A JP 2017547968A JP 2017547968 A JP2017547968 A JP 2017547968A JP 2018513123 A JP2018513123 A JP 2018513123A
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cancer
rorγ
cells
agent
inhibitor
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JP2018513123A5 (https=
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ホンウ チェン
ホンウ チェン
ジューン エックス. ゾウ
ジューン エックス. ゾウ
チュンチエン ワン
チュンチエン ワン
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University of California
University of California Los Angeles UCLA
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University of California San Diego UCSD
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JP2017547968A 2015-03-12 2016-03-11 Rorガンマ阻害剤を用いてがんを治療するための方法 Pending JP2018513123A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201562132465P 2015-03-12 2015-03-12
US62/132,465 2015-03-12
US201662280081P 2016-01-18 2016-01-18
US62/280,081 2016-01-18
PCT/US2016/021983 WO2016145298A1 (en) 2015-03-12 2016-03-11 METHODS FOR TREATING CANCER WITH RORgamma INHIBITORS

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JP2018513123A true JP2018513123A (ja) 2018-05-24
JP2018513123A5 JP2018513123A5 (https=) 2019-04-18

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US (1) US10959984B2 (https=)
EP (1) EP3268087A4 (https=)
JP (1) JP2018513123A (https=)
CN (1) CN107614062A (https=)
HK (1) HK1249469A1 (https=)
WO (1) WO2016145298A1 (https=)

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JP2022520859A (ja) * 2019-02-20 2022-04-01 ザ リージェンツ オブ ザ ユニバーシティ オブ カリフォルニア レチノイン酸受容体関連オーファン受容体γ(RORγ)依存性がんのための治療

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EP3532062B1 (en) * 2016-10-27 2022-07-20 Escalier Biosciences, BV Ror-gamma modulators
WO2019023651A2 (en) 2017-07-28 2019-01-31 Massachusetts Institute Of Technology MODULATORS OF THE SMALL MOLECULE ANDROGEN RECEPTOR
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WO2020065682A1 (en) * 2018-09-29 2020-04-02 Translational Health Science And Technology Institute Ror antagonists, their use and method of treatment comprising the said modulators
RU2679625C1 (ru) * 2018-11-08 2019-02-12 Ильясов Шамиль Сионович ПРИМЕНЕНИЕ 3-О-СУЛЬФАМОИЛОКСИ-6-ОКСА-7β-МЕТИЛ-D-ГОМО-8α-ЭСТРА-1,3,5(10)-ТРИЕН-17а-ОНА ДЛЯ ЛЕЧЕНИЯ РАКА МОЛОЧНОЙ ЖЕЛЕЗЫ, ВКЛЮЧАЯ ТРИЖДЫ-НЕГАТИВНУЮ ФОРМУ, И СПОСОБ ЕГО ПОЛУЧЕНИЯ
CN109879784B (zh) * 2019-03-18 2021-06-29 中国科学院广州生物医药与健康研究院 一种联苯胺类化合物及其应用
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WO2021011493A1 (en) * 2019-07-12 2021-01-21 Duke University 3' utr crispr-dcas 13 engineering system and methods of using same
CN113912563B (zh) * 2020-07-10 2025-05-27 中国科学院广州生物医药与健康研究院 一种苯并五元氮杂环化合物及其应用
WO2022067185A1 (en) * 2020-09-27 2022-03-31 Veru Inc. Methods of treating prostate cancer with minimal side effects
WO2022122740A1 (en) * 2020-12-07 2022-06-16 Diaccurate Ror-gamma inhibitors for the treatment of ror-gamma-dependent cancer
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WO2023155846A1 (zh) * 2022-02-18 2023-08-24 上海醇健医药技术有限公司 17-吡啶基-10α-甲基-甾体衍生物及中间体化合物、其制备方法、其用途、以及其药物组合物

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