JP2018501251A - 新規イソチアゾールアミド、それらの調製方法および殺真菌剤としてのそれらの使用 - Google Patents

新規イソチアゾールアミド、それらの調製方法および殺真菌剤としてのそれらの使用 Download PDF

Info

Publication number
JP2018501251A
JP2018501251A JP2017533376A JP2017533376A JP2018501251A JP 2018501251 A JP2018501251 A JP 2018501251A JP 2017533376 A JP2017533376 A JP 2017533376A JP 2017533376 A JP2017533376 A JP 2017533376A JP 2018501251 A JP2018501251 A JP 2018501251A
Authority
JP
Japan
Prior art keywords
alkyl
alkoxy
cycloalkyl
residues
alkylsulfonyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2017533376A
Other languages
English (en)
Japanese (ja)
Other versions
JP2018501251A5 (enExample
Inventor
ベルニエ，ダヴィド
クリスト，ピエール
知己 土屋
知己 土屋
リノルフィ，フィリップ
ドロゲ，トマス
メイヒリング，シモン
シュミット，ジャン・ピーター
テルザー，ヨアヒム
ドラー，ウーヴェ
モズラン，マルク
レイ，ユリアン
ティーべ，ヨルグ
ヴァッヒェンドルフ−ノイマン，ウルリーケ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer CropScience AG
Original Assignee
Bayer CropScience AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer CropScience AG filed Critical Bayer CropScience AG
Publication of JP2018501251A publication Critical patent/JP2018501251A/ja
Publication of JP2018501251A5 publication Critical patent/JP2018501251A5/ja
Pending legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/18—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof containing a —O—CO—N< group, or a thio analogue thereof, directly attached to a heterocyclic or cycloaliphatic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
    • C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2017533376A 2014-12-22 2015-12-21 新規イソチアゾールアミド、それらの調製方法および殺真菌剤としてのそれらの使用 Pending JP2018501251A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14199548 2014-12-22
EP14199548.0 2014-12-22
PCT/EP2015/080739 WO2016102435A2 (en) 2014-12-22 2015-12-21 Novel isothiazolamides, processes for their preparation and their use as fungicides

Publications (2)

Publication Number Publication Date
JP2018501251A true JP2018501251A (ja) 2018-01-18
JP2018501251A5 JP2018501251A5 (enExample) 2019-02-07

Family

ID=52130123

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2017533376A Pending JP2018501251A (ja) 2014-12-22 2015-12-21 新規イソチアゾールアミド、それらの調製方法および殺真菌剤としてのそれらの使用

Country Status (7)

Country Link
US (1) US20190110476A1 (enExample)
EP (1) EP3236752A2 (enExample)
JP (1) JP2018501251A (enExample)
CN (1) CN107205394A (enExample)
BR (1) BR112017013610A2 (enExample)
TW (1) TW201632507A (enExample)
WO (1) WO2016102435A2 (enExample)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2018501252A (ja) * 2014-12-22 2018-01-18 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 新規イソチアゾールアミド、それらの調製方法ならびに除草剤および／または植物成長調節剤としてのそれらの使用
WO2020054531A1 (ja) * 2018-09-14 2020-03-19 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 植物病害防除剤
JPWO2020090603A1 (ja) * 2018-10-31 2021-09-30 クミアイ化学工業株式会社 ムギ類の病害防除方法、ムギ類の種子及びムギ類の倒伏被害抑制方法

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2017207395A1 (en) 2016-06-02 2017-12-07 Bayer Cropscience Aktiengesellschaft Isothiazolopyridones, processes for their preparation and their use as fungicides
CN109195974A (zh) 2016-06-02 2019-01-11 拜耳作物科学股份公司 异噻唑并吡啶酮、其制备方法及其用作除草剂和/或植物生长调节剂的用途
EP3648605A1 (en) 2017-07-03 2020-05-13 Bayer CropScience Aktiengesellschaft Novel isothiazolo-based bicycles, processes for their preparation and their use as herbicides and/or plant growth regulators
EP3648606A1 (en) 2017-07-03 2020-05-13 Bayer CropScience Aktiengesellschaft Novel substituted isothiazolopyridones, processes for their preparation and their use as herbicides and/or plant growth regulators
CN111433214A (zh) * 2017-11-29 2020-07-17 拜耳公司 新的异噻唑-氮杂*酮双环、其制备方法及其作为除草剂和/或植物生长调节剂的用途
US20210032205A1 (en) * 2018-02-27 2021-02-04 Nippon Soda Co., Ltd. Heteroaryl sulfonamide compound and formulation for controlling harmful organisms
EP3760627A4 (en) * 2018-02-28 2022-03-02 Hokko Chemical Industry Co., Ltd. IMIDE DERIVATIVE AND BACTERICIDE WITH THIS AS AN ACTIVE SUBSTANCE
WO2020161209A1 (en) 2019-02-06 2020-08-13 Syngenta Crop Protection Ag Herbicidal fused pyridazine compounds
WO2020161208A1 (en) 2019-02-06 2020-08-13 Syngenta Crop Protection Ag Herbicidal fused pyridazine compounds
JP2023527379A (ja) * 2020-05-27 2023-06-28 コンステレーション・ファーマシューティカルズ・インコーポレイテッド Ｔｒｅｘ１のモジュレーターとしての置換ベンズアミド
KR20240136380A (ko) 2022-01-14 2024-09-13 엔코 켐 인코포레이티드 프로토포르피리노겐 산화효소 억제제
WO2024059559A1 (en) * 2022-09-12 2024-03-21 Hotspot Therapeutics, Inc. Isothiazolylcarboxamide compounds and their use in therapy

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010018714A1 (ja) * 2008-08-13 2010-02-18 三井化学アグロ株式会社 アミド誘導体、該アミド誘導体を含有する有害生物防除剤およびその使用方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US896623A (en) * 1908-03-02 1908-08-18 Jesse Childs Pit-car.
DE1795344B2 (de) * 1968-09-17 1976-05-06 Bayer Ag, 5090 Leverkusen Verfahren zur herstellung von 3-aminoisothiazolen
GB1548397A (en) * 1976-06-01 1979-07-11 Lilly Industries Ltd Acylated amino-isoxazoles and aminoisothiazoles
US4267341A (en) * 1977-11-23 1981-05-12 Merck & Co., Inc. Process for preparing 2,3-substituted-1,2,-isothiazolium salt antimicrobials
US4292430A (en) * 1977-11-23 1981-09-29 Merck & Co., Inc. 2,3-Substituted-1,2-isothiazolium salt antimicrobials
JPH07500116A (ja) * 1992-03-26 1995-01-05 ダウエランコ 殺菌剤としてのｎ−複素環式ニトロアニリン
ATE243204T1 (de) * 1995-08-24 2003-07-15 Basf Ag Isoxazole- und isothiazole-5-carboxamid derivate, deren herstellung und deren verwendung als herbizide
WO2003010143A1 (en) * 2001-07-26 2003-02-06 Samsung Electronics Co., Ltd. Dialkylhydroxybenzoic acid derivatives containing metal chelating groups and their therapeutic uses
WO2004092123A2 (en) * 2003-04-10 2004-10-28 Microbia, Inc. Inhibitors of fungal invasion
TW200738701A (en) * 2005-07-26 2007-10-16 Du Pont Fungicidal carboxamides
US8686044B2 (en) * 2008-08-13 2014-04-01 Mitsui Chemicals Agro, Inc. Amide derivative, pest control agent containing the amide derivative, and use of the amide derivative

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010018714A1 (ja) * 2008-08-13 2010-02-18 三井化学アグロ株式会社 アミド誘導体、該アミド誘導体を含有する有害生物防除剤およびその使用方法

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
REGISTRY（STN）[ONLINE], JPN7019003100, ISSN: 0004121157 *

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2018501252A (ja) * 2014-12-22 2018-01-18 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 新規イソチアゾールアミド、それらの調製方法ならびに除草剤および／または植物成長調節剤としてのそれらの使用
WO2020054531A1 (ja) * 2018-09-14 2020-03-19 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 植物病害防除剤
JPWO2020090603A1 (ja) * 2018-10-31 2021-09-30 クミアイ化学工業株式会社 ムギ類の病害防除方法、ムギ類の種子及びムギ類の倒伏被害抑制方法
JP7524067B2 (ja) 2018-10-31 2024-07-29 クミアイ化学工業株式会社 ムギ類の病害防除方法、ムギ類の種子及びムギ類の倒伏被害抑制方法

Also Published As

Publication number Publication date
WO2016102435A2 (en) 2016-06-30
BR112017013610A2 (pt) 2018-03-06
WO2016102435A3 (en) 2016-09-09
EP3236752A2 (en) 2017-11-01
CN107205394A (zh) 2017-09-26
US20190110476A1 (en) 2019-04-18
TW201632507A (zh) 2016-09-16

Similar Documents

Publication Publication Date Title
JP2018501251A (ja) 新規イソチアゾールアミド、それらの調製方法および殺真菌剤としてのそれらの使用
WO2016156282A1 (en) Novel triazole compounds for controlling phytopathogenic harmful fungi
CN107635968A (zh) 新的5‑取代的咪唑衍生物
CN109983010A (zh) 作为用于作物保护的杀真菌剂的1-[2-(1-氯环丙基)-2-羟基-3-(3-苯基-1,2-噁唑-5-基)丙基]-1h-咪唑-5-甲腈衍生物及相关化合物
US10246420B2 (en) Pyrazole derivatives
TW201641493A (zh) 新穎三唑衍生物
CN109983000A (zh) 新的5-取代的咪唑基甲基衍生物
AU2017333333A1 (en) 5-substituted imidazolylmethyldioxolane derivatives as fungiciides
EP3519392A1 (en) Novel 5-substituted imidazole derivatives
CN107428706A (zh) 作为农药和植物生长调节剂的三唑衍生物
US20170303540A1 (en) Novel triazole derivatives
EP3277674B1 (en) Triazol derivatives as fungicides
JP2019530688A (ja) 新規５−置換イミダゾリルメチル誘導体
US20190223437A1 (en) Active compound combinations comprising a 5-substituted imidazole derivative
CN110267952A (zh) 三唑硫酮衍生物
CN109996796A (zh) 作为杀真菌剂的5-取代的咪唑基甲基环氧乙烷衍生物
US20190218187A1 (en) Novel 5-substituted imidazolylmethyl derivatives
WO2017207395A1 (en) Isothiazolopyridones, processes for their preparation and their use as fungicides

Legal Events

Date Code Title Description
A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20181218

A621 Written request for application examination

Free format text: JAPANESE INTERMEDIATE CODE: A621

Effective date: 20181218

A977 Report on retrieval

Free format text: JAPANESE INTERMEDIATE CODE: A971007

Effective date: 20190912

A131 Notification of reasons for refusal

Free format text: JAPANESE INTERMEDIATE CODE: A131

Effective date: 20191001

A02 Decision of refusal

Free format text: JAPANESE INTERMEDIATE CODE: A02

Effective date: 20200512