JP2018501251A - 新規イソチアゾールアミド、それらの調製方法および殺真菌剤としてのそれらの使用 - Google Patents

新規イソチアゾールアミド、それらの調製方法および殺真菌剤としてのそれらの使用 Download PDF

Info

Publication number
JP2018501251A
JP2018501251A JP2017533376A JP2017533376A JP2018501251A JP 2018501251 A JP2018501251 A JP 2018501251A JP 2017533376 A JP2017533376 A JP 2017533376A JP 2017533376 A JP2017533376 A JP 2017533376A JP 2018501251 A JP2018501251 A JP 2018501251A
Authority
JP
Japan
Prior art keywords
alkyl
alkoxy
cycloalkyl
residues
alkylsulfonyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2017533376A
Other languages
English (en)
Japanese (ja)
Other versions
JP2018501251A5 (enExample
Inventor
ベルニエ，ダヴィド
クリスト，ピエール
知己 土屋
知己 土屋
リノルフィ，フィリップ
ドロゲ，トマス
メイヒリング，シモン
シュミット，ジャン・ピーター
テルザー，ヨアヒム
ドラー，ウーヴェ
モズラン，マルク
レイ，ユリアン
ティーべ，ヨルグ
ヴァッヒェンドルフ−ノイマン，ウルリーケ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer CropScience AG
Original Assignee
Bayer CropScience AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer CropScience AG filed Critical Bayer CropScience AG
Publication of JP2018501251A publication Critical patent/JP2018501251A/ja
Publication of JP2018501251A5 publication Critical patent/JP2018501251A5/ja
Pending legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/18—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof containing a —O—CO—N< group, or a thio analogue thereof, directly attached to a heterocyclic or cycloaliphatic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
    • C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2017533376A 2014-12-22 2015-12-21 新規イソチアゾールアミド、それらの調製方法および殺真菌剤としてのそれらの使用 Pending JP2018501251A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14199548.0 2014-12-22
EP14199548 2014-12-22
PCT/EP2015/080739 WO2016102435A2 (en) 2014-12-22 2015-12-21 Novel isothiazolamides, processes for their preparation and their use as fungicides

Publications (2)

Publication Number Publication Date
JP2018501251A true JP2018501251A (ja) 2018-01-18
JP2018501251A5 JP2018501251A5 (enExample) 2019-02-07

Family

ID=52130123

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2017533376A Pending JP2018501251A (ja) 2014-12-22 2015-12-21 新規イソチアゾールアミド、それらの調製方法および殺真菌剤としてのそれらの使用

Country Status (7)

Country Link
US (1) US20190110476A1 (enExample)
EP (1) EP3236752A2 (enExample)
JP (1) JP2018501251A (enExample)
CN (1) CN107205394A (enExample)
BR (1) BR112017013610A2 (enExample)
TW (1) TW201632507A (enExample)
WO (1) WO2016102435A2 (enExample)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2018501252A (ja) * 2014-12-22 2018-01-18 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 新規イソチアゾールアミド、それらの調製方法ならびに除草剤および／または植物成長調節剤としてのそれらの使用
WO2020054531A1 (ja) * 2018-09-14 2020-03-19 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 植物病害防除剤
JPWO2020090603A1 (ja) * 2018-10-31 2021-09-30 クミアイ化学工業株式会社 ムギ類の病害防除方法、ムギ類の種子及びムギ類の倒伏被害抑制方法

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112018074920A2 (pt) 2016-06-02 2019-03-12 Bayer Cropscience Ag isotiazolopiridonas, processos para sua preparação e seu uso como herbicidas e/ou reguladores de crescimento de planta
WO2017207395A1 (en) 2016-06-02 2017-12-07 Bayer Cropscience Aktiengesellschaft Isothiazolopyridones, processes for their preparation and their use as fungicides
US20200123175A1 (en) * 2017-07-03 2020-04-23 Bayer Cropscience Aktiengesellschaft Novel isothiazolo-based bicycles, processes for their preparation and their use as herbicides and/or plant growth regulators
BR112020000083A2 (pt) * 2017-07-03 2020-07-07 Bayer Cropscience Aktiengesellschaft novas isotiazolopiridonas substituídas, processos para sua preparação e seu uso como herbicidas e/ou reguladores de crescimento da planta
BR112020010583A2 (pt) 2017-11-29 2020-11-10 Bayer Aktiengesellschaft novos biciclos de isotiazol-azepinona, processos para sua preparação e seu uso como herbicidas e/ou reguladores de crescimento de plantas
JPWO2019167863A1 (ja) * 2018-02-27 2021-03-04 日本曹達株式会社 ヘテロアリールスルホンアミド化合物および有害生物防除剤
EP3760627A4 (en) * 2018-02-28 2022-03-02 Hokko Chemical Industry Co., Ltd. IMIDE DERIVATIVE AND BACTERICIDE WITH THIS AS AN ACTIVE SUBSTANCE
WO2020161208A1 (en) 2019-02-06 2020-08-13 Syngenta Crop Protection Ag Herbicidal fused pyridazine compounds
WO2020161209A1 (en) 2019-02-06 2020-08-13 Syngenta Crop Protection Ag Herbicidal fused pyridazine compounds
CA3179627A1 (en) * 2020-05-27 2021-12-02 Aaron Coffin Substituted benzamides as modulators of trex1
JP2025503677A (ja) 2022-01-14 2025-02-04 エンコ ケム，インコーポレイテッド プロトポルフィリノーゲンオキシダーゼ阻害剤
WO2024059559A1 (en) * 2022-09-12 2024-03-21 Hotspot Therapeutics, Inc. Isothiazolylcarboxamide compounds and their use in therapy

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010018714A1 (ja) * 2008-08-13 2010-02-18 三井化学アグロ株式会社 アミド誘導体、該アミド誘導体を含有する有害生物防除剤およびその使用方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US896623A (en) * 1908-03-02 1908-08-18 Jesse Childs Pit-car.
DE1795344B2 (de) * 1968-09-17 1976-05-06 Bayer Ag, 5090 Leverkusen Verfahren zur herstellung von 3-aminoisothiazolen
GB1548397A (en) * 1976-06-01 1979-07-11 Lilly Industries Ltd Acylated amino-isoxazoles and aminoisothiazoles
US4267341A (en) * 1977-11-23 1981-05-12 Merck & Co., Inc. Process for preparing 2,3-substituted-1,2,-isothiazolium salt antimicrobials
US4292430A (en) * 1977-11-23 1981-09-29 Merck & Co., Inc. 2,3-Substituted-1,2-isothiazolium salt antimicrobials
WO1993019054A1 (en) * 1992-03-26 1993-09-30 Dowelanco N-heterocyclic nitro anilines as fungicides
DE69628705T2 (de) * 1995-08-24 2004-05-13 Basf Ag Isoxazole- und Isothiazole-5-carboxamid Derivate, deren Herstellung und deren Verwendung als Herbizide
WO2003010143A1 (en) * 2001-07-26 2003-02-06 Samsung Electronics Co., Ltd. Dialkylhydroxybenzoic acid derivatives containing metal chelating groups and their therapeutic uses
WO2004092123A2 (en) * 2003-04-10 2004-10-28 Microbia, Inc. Inhibitors of fungal invasion
TW200738701A (en) * 2005-07-26 2007-10-16 Du Pont Fungicidal carboxamides
US8686044B2 (en) * 2008-08-13 2014-04-01 Mitsui Chemicals Agro, Inc. Amide derivative, pest control agent containing the amide derivative, and use of the amide derivative

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010018714A1 (ja) * 2008-08-13 2010-02-18 三井化学アグロ株式会社 アミド誘導体、該アミド誘導体を含有する有害生物防除剤およびその使用方法

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
REGISTRY（STN）[ONLINE], JPN7019003100, ISSN: 0004121157 *

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2018501252A (ja) * 2014-12-22 2018-01-18 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 新規イソチアゾールアミド、それらの調製方法ならびに除草剤および／または植物成長調節剤としてのそれらの使用
WO2020054531A1 (ja) * 2018-09-14 2020-03-19 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 植物病害防除剤
JPWO2020090603A1 (ja) * 2018-10-31 2021-09-30 クミアイ化学工業株式会社 ムギ類の病害防除方法、ムギ類の種子及びムギ類の倒伏被害抑制方法
JP7524067B2 (ja) 2018-10-31 2024-07-29 クミアイ化学工業株式会社 ムギ類の病害防除方法、ムギ類の種子及びムギ類の倒伏被害抑制方法

Also Published As

Publication number Publication date
CN107205394A (zh) 2017-09-26
BR112017013610A2 (pt) 2018-03-06
WO2016102435A3 (en) 2016-09-09
TW201632507A (zh) 2016-09-16
EP3236752A2 (en) 2017-11-01
WO2016102435A2 (en) 2016-06-30
US20190110476A1 (en) 2019-04-18

Similar Documents

Publication Publication Date Title
CN107205394A (zh) 新的异噻唑酰胺、其制备方法及其作为杀真菌剂的用途
WO2016156282A1 (en) Novel triazole compounds for controlling phytopathogenic harmful fungi
CN107635968A (zh) 新的5‑取代的咪唑衍生物
CN109983010A (zh) 作为用于作物保护的杀真菌剂的1-[2-(1-氯环丙基)-2-羟基-3-(3-苯基-1,2-噁唑-5-基)丙基]-1h-咪唑-5-甲腈衍生物及相关化合物
CN107249329A (zh) 新的异噻唑酰胺、其制备方法及其作为除草剂和/或植物生长调节剂的用途
US10246420B2 (en) Pyrazole derivatives
TW201641493A (zh) 新穎三唑衍生物
CN109983000A (zh) 新的5-取代的咪唑基甲基衍生物
US20190223437A1 (en) Active compound combinations comprising a 5-substituted imidazole derivative
AU2017333333A1 (en) 5-substituted imidazolylmethyldioxolane derivatives as fungiciides
EP3519392A1 (en) Novel 5-substituted imidazole derivatives
CN107428706A (zh) 作为农药和植物生长调节剂的三唑衍生物
US20170303540A1 (en) Novel triazole derivatives
CN109982999A (zh) 新的5-取代的咪唑基甲基衍生物
CN110267952A (zh) 三唑硫酮衍生物
CN109996796A (zh) 作为杀真菌剂的5-取代的咪唑基甲基环氧乙烷衍生物
US20190218187A1 (en) Novel 5-substituted imidazolylmethyl derivatives
EP3277674A1 (en) Triazol derivatives as fungicides
WO2017207395A1 (en) Isothiazolopyridones, processes for their preparation and their use as fungicides

Legal Events

Date Code Title Description
A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20181218

A621 Written request for application examination

Free format text: JAPANESE INTERMEDIATE CODE: A621

Effective date: 20181218

A977 Report on retrieval

Free format text: JAPANESE INTERMEDIATE CODE: A971007

Effective date: 20190912

A131 Notification of reasons for refusal

Free format text: JAPANESE INTERMEDIATE CODE: A131

Effective date: 20191001

A02 Decision of refusal

Free format text: JAPANESE INTERMEDIATE CODE: A02

Effective date: 20200512