JP2018501251A - 新規イソチアゾールアミド、それらの調製方法および殺真菌剤としてのそれらの使用 - Google Patents

新規イソチアゾールアミド、それらの調製方法および殺真菌剤としてのそれらの使用 Download PDF

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Publication number
JP2018501251A
JP2018501251A JP2017533376A JP2017533376A JP2018501251A JP 2018501251 A JP2018501251 A JP 2018501251A JP 2017533376 A JP2017533376 A JP 2017533376A JP 2017533376 A JP2017533376 A JP 2017533376A JP 2018501251 A JP2018501251 A JP 2018501251A
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JP
Japan
Prior art keywords
alkyl
alkoxy
cycloalkyl
residues
alkylsulfonyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2017533376A
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English (en)
Japanese (ja)
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JP2018501251A5 (cg-RX-API-DMAC7.html
Inventor
ベルニエ，ダヴィド
クリスト，ピエール
知己 土屋
知己 土屋
リノルフィ，フィリップ
ドロゲ，トマス
メイヒリング，シモン
シュミット，ジャン・ピーター
テルザー，ヨアヒム
ドラー，ウーヴェ
モズラン，マルク
レイ，ユリアン
ティーべ，ヨルグ
ヴァッヒェンドルフ−ノイマン，ウルリーケ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer CropScience AG
Original Assignee
Bayer CropScience AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer CropScience AG filed Critical Bayer CropScience AG
Publication of JP2018501251A publication Critical patent/JP2018501251A/ja
Publication of JP2018501251A5 publication Critical patent/JP2018501251A5/ja
Pending legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/18—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof containing a —O—CO—N< group, or a thio analogue thereof, directly attached to a heterocyclic or cycloaliphatic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
    • C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2017533376A 2014-12-22 2015-12-21 新規イソチアゾールアミド、それらの調製方法および殺真菌剤としてのそれらの使用 Pending JP2018501251A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14199548.0 2014-12-22
EP14199548 2014-12-22
PCT/EP2015/080739 WO2016102435A2 (en) 2014-12-22 2015-12-21 Novel isothiazolamides, processes for their preparation and their use as fungicides

Publications (2)

Publication Number Publication Date
JP2018501251A true JP2018501251A (ja) 2018-01-18
JP2018501251A5 JP2018501251A5 (cg-RX-API-DMAC7.html) 2019-02-07

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
JP2017533376A Pending JP2018501251A (ja) 2014-12-22 2015-12-21 新規イソチアゾールアミド、それらの調製方法および殺真菌剤としてのそれらの使用

Country Status (7)

Country Link
US (1) US20190110476A1 (cg-RX-API-DMAC7.html)
EP (1) EP3236752A2 (cg-RX-API-DMAC7.html)
JP (1) JP2018501251A (cg-RX-API-DMAC7.html)
CN (1) CN107205394A (cg-RX-API-DMAC7.html)
BR (1) BR112017013610A2 (cg-RX-API-DMAC7.html)
TW (1) TW201632507A (cg-RX-API-DMAC7.html)
WO (1) WO2016102435A2 (cg-RX-API-DMAC7.html)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2018501252A (ja) * 2014-12-22 2018-01-18 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 新規イソチアゾールアミド、それらの調製方法ならびに除草剤および／または植物成長調節剤としてのそれらの使用
WO2020054531A1 (ja) * 2018-09-14 2020-03-19 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 植物病害防除剤
JPWO2020090603A1 (ja) * 2018-10-31 2021-09-30 クミアイ化学工業株式会社 ムギ類の病害防除方法、ムギ類の種子及びムギ類の倒伏被害抑制方法

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3464296B1 (en) 2016-06-02 2020-10-14 Bayer CropScience Aktiengesellschaft Isothiazolopyridones, processes for their preparation and their use as herbicides and/or plant growth regulators
WO2017207395A1 (en) 2016-06-02 2017-12-07 Bayer Cropscience Aktiengesellschaft Isothiazolopyridones, processes for their preparation and their use as fungicides
US10842152B2 (en) 2017-07-03 2020-11-24 Bayer Cropscience Aktiengesellschaft Isothiazolo-based bicycles, processes for their preparation and their use as herbicides and/or plant growth regulators
WO2019007793A1 (en) 2017-07-03 2019-01-10 Bayer Cropscience Aktiengesellschaft NOVEL ISOTHIAZOLO-BASED BICYCLES, PROCESSES FOR PREPARING THEM AND USE THEREOF AS HERBICIDES AND / OR PLANT GROWTH REGULATORS
US20210002301A1 (en) * 2017-11-29 2021-01-07 Bayer Aktiengesellschaft Novel isothiazolo-azepinone bicycles, processes for their preparation and their use as herbicides and/or plant growth regulators
EP3760615A4 (en) * 2018-02-27 2021-07-14 Nippon Soda Co., Ltd. HETEROARYL SULFONAMIDE COMPOUND AND PEST CONTROL AGENT
CN111788200A (zh) * 2018-02-28 2020-10-16 北兴化学工业株式会社 酰亚胺衍生物和包含所述衍生物作为活性成分的杀菌剂
WO2020161208A1 (en) 2019-02-06 2020-08-13 Syngenta Crop Protection Ag Herbicidal fused pyridazine compounds
WO2020161209A1 (en) 2019-02-06 2020-08-13 Syngenta Crop Protection Ag Herbicidal fused pyridazine compounds
WO2021243001A1 (en) * 2020-05-27 2021-12-02 Constellation Pharmaceuticals, Inc. Substituted benzamides as modulators of trex1
CN118525002A (zh) 2022-01-14 2024-08-20 恩科化学公司 原卟啉原氧化酶抑制剂
WO2024059559A1 (en) * 2022-09-12 2024-03-21 Hotspot Therapeutics, Inc. Isothiazolylcarboxamide compounds and their use in therapy

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DE1795344B2 (de) * 1968-09-17 1976-05-06 Bayer Ag, 5090 Leverkusen Verfahren zur herstellung von 3-aminoisothiazolen
GB1548397A (en) * 1976-06-01 1979-07-11 Lilly Industries Ltd Acylated amino-isoxazoles and aminoisothiazoles
US4292430A (en) * 1977-11-23 1981-09-29 Merck & Co., Inc. 2,3-Substituted-1,2-isothiazolium salt antimicrobials
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WO1993019054A1 (en) * 1992-03-26 1993-09-30 Dowelanco N-heterocyclic nitro anilines as fungicides
EP0761654B1 (en) * 1995-08-24 2003-06-18 Basf Aktiengesellschaft Isoxazole- and isothiazole-5-carboxamide derivatives, their preparation and their use as herbicides
WO2003010143A1 (en) * 2001-07-26 2003-02-06 Samsung Electronics Co., Ltd. Dialkylhydroxybenzoic acid derivatives containing metal chelating groups and their therapeutic uses
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US8686044B2 (en) * 2008-08-13 2014-04-01 Mitsui Chemicals Agro, Inc. Amide derivative, pest control agent containing the amide derivative, and use of the amide derivative

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Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2018501252A (ja) * 2014-12-22 2018-01-18 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 新規イソチアゾールアミド、それらの調製方法ならびに除草剤および／または植物成長調節剤としてのそれらの使用
WO2020054531A1 (ja) * 2018-09-14 2020-03-19 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 植物病害防除剤
JPWO2020090603A1 (ja) * 2018-10-31 2021-09-30 クミアイ化学工業株式会社 ムギ類の病害防除方法、ムギ類の種子及びムギ類の倒伏被害抑制方法
JP7524067B2 (ja) 2018-10-31 2024-07-29 クミアイ化学工業株式会社 ムギ類の病害防除方法、ムギ類の種子及びムギ類の倒伏被害抑制方法

Also Published As

Publication number Publication date
US20190110476A1 (en) 2019-04-18
TW201632507A (zh) 2016-09-16
CN107205394A (zh) 2017-09-26
EP3236752A2 (en) 2017-11-01
WO2016102435A3 (en) 2016-09-09
BR112017013610A2 (pt) 2018-03-06
WO2016102435A2 (en) 2016-06-30

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