JP2017534675A5 - - Google Patents

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Publication number
JP2017534675A5
JP2017534675A5 JP2017536216A JP2017536216A JP2017534675A5 JP 2017534675 A5 JP2017534675 A5 JP 2017534675A5 JP 2017536216 A JP2017536216 A JP 2017536216A JP 2017536216 A JP2017536216 A JP 2017536216A JP 2017534675 A5 JP2017534675 A5 JP 2017534675A5
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JP
Japan
Prior art keywords
alkyl
group
glycine
acid
prodrug according
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JP2017536216A
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English (en)
Japanese (ja)
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JP2017534675A (ja
JP6701208B2 (ja
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Priority claimed from PCT/US2015/051705 external-priority patent/WO2016049174A1/en
Publication of JP2017534675A publication Critical patent/JP2017534675A/ja
Publication of JP2017534675A5 publication Critical patent/JP2017534675A5/ja
Application granted granted Critical
Publication of JP6701208B2 publication Critical patent/JP6701208B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2017536216A 2014-09-24 2015-09-23 脂質化アミド系インスリンプロドラッグ Expired - Fee Related JP6701208B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201462054670P 2014-09-24 2014-09-24
US62/054,670 2014-09-24
PCT/US2015/051705 WO2016049174A1 (en) 2014-09-24 2015-09-23 Lipidated amide-based insulin prodrugs

Publications (3)

Publication Number Publication Date
JP2017534675A JP2017534675A (ja) 2017-11-24
JP2017534675A5 true JP2017534675A5 (https=) 2018-10-25
JP6701208B2 JP6701208B2 (ja) 2020-05-27

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ID=55581947

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JP2017536216A Expired - Fee Related JP6701208B2 (ja) 2014-09-24 2015-09-23 脂質化アミド系インスリンプロドラッグ

Country Status (6)

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US (1) US10385107B2 (https=)
EP (1) EP3197912B1 (https=)
JP (1) JP6701208B2 (https=)
CN (1) CN107001441A (https=)
ES (1) ES2947409T3 (https=)
WO (1) WO2016049174A1 (https=)

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MY206918A (en) 2020-11-06 2025-01-17 Novo Nordisk As Glp-1 prodrugs and uses hereof
WO2023012263A1 (en) 2021-08-04 2023-02-09 Novo Nordisk A/S Solid oral peptide formulations
TW202330584A (zh) 2022-01-20 2023-08-01 丹麥商諾佛 儂迪克股份有限公司 前藥及其用途
JP2025517672A (ja) 2022-05-10 2025-06-10 ノヴォ ノルディスク アー/エス プロドラッグおよびその使用
TW202421645A (zh) 2022-11-25 2024-06-01 丹麥商諾佛 儂迪克股份有限公司 如glp—1之肽治療劑的口服投與

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