JP2017516772A5 - - Google Patents

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Publication number
JP2017516772A5
JP2017516772A5 JP2016568812A JP2016568812A JP2017516772A5 JP 2017516772 A5 JP2017516772 A5 JP 2017516772A5 JP 2016568812 A JP2016568812 A JP 2016568812A JP 2016568812 A JP2016568812 A JP 2016568812A JP 2017516772 A5 JP2017516772 A5 JP 2017516772A5
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JP
Japan
Prior art keywords
dodeca
oxo
triazatricyclo
trifluoromethyl
tetraen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2016568812A
Other languages
English (en)
Japanese (ja)
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JP2017516772A (ja
JP6580074B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2015/061468 external-priority patent/WO2015177367A1/en
Publication of JP2017516772A publication Critical patent/JP2017516772A/ja
Publication of JP2017516772A5 publication Critical patent/JP2017516772A5/ja
Application granted granted Critical
Publication of JP6580074B2 publication Critical patent/JP6580074B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2016568812A 2014-05-23 2015-05-22 S100阻害薬として有用な新規化合物 Expired - Fee Related JP6580074B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14169757 2014-05-23
EP14169757.3 2014-05-23
PCT/EP2015/061468 WO2015177367A1 (en) 2014-05-23 2015-05-22 Novel compounds useful as s100-inhibitors

Publications (3)

Publication Number Publication Date
JP2017516772A JP2017516772A (ja) 2017-06-22
JP2017516772A5 true JP2017516772A5 (en:Method) 2018-05-10
JP6580074B2 JP6580074B2 (ja) 2019-09-25

Family

ID=50774707

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2016568812A Expired - Fee Related JP6580074B2 (ja) 2014-05-23 2015-05-22 S100阻害薬として有用な新規化合物

Country Status (12)

Country Link
US (1) US9771372B2 (en:Method)
EP (1) EP2991990B1 (en:Method)
JP (1) JP6580074B2 (en:Method)
KR (1) KR20170005868A (en:Method)
CN (1) CN106414448B (en:Method)
AU (1) AU2015261775B2 (en:Method)
BR (1) BR112016024749A2 (en:Method)
CA (1) CA2948436A1 (en:Method)
EA (1) EA030604B1 (en:Method)
ES (1) ES2620751T3 (en:Method)
MX (1) MX2016014483A (en:Method)
WO (1) WO2015177367A1 (en:Method)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7392951B2 (ja) 2018-04-27 2023-12-06 国立大学法人 岡山大学 抗s100a8/a9抗体とその用途
US11197908B2 (en) 2018-07-17 2021-12-14 The Board Of Trustees Of The University Of Arkansas Peptoids and methods for attenuating inflammatory response
US20230144545A1 (en) 2019-10-30 2023-05-11 National University Corporation Okayama University Prophylactic and/or therapeutic agent for inflammatory pulmonary disease
WO2023209141A1 (en) 2022-04-29 2023-11-02 Westfälische Wilhelms-Universität Münster Benzo[d]imidazo[1,2-a]imidazoles and their use in diagnosis
WO2025132458A1 (en) 2023-12-18 2025-06-26 Chiesi Farmaceutici S.P.A. Pyridazinyl amino derivatives as alk5 inhibitors

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6248755B1 (en) 1999-04-06 2001-06-19 Merck & Co., Inc. Pyrrolidine modulators of chemokine receptor activity
AR029489A1 (es) 2000-03-10 2003-07-02 Euro Celtique Sa Piridinas, pirimidinas, pirazinas, triazinas sustituidas por arilo, composiciones farmaceuticas y el uso de las mismas para la manufactura de un medicamento
HUP0300721A3 (en) 2000-07-26 2006-02-28 Smithkline Beecham Plc Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity, process for producing them, pharmaceutical compositions containing them and use thereof
CA2440037C (en) * 2001-03-05 2010-02-16 Transtech Pharma, Inc. Benzimidazole derivatives for modulating the rage receptor
GB0117506D0 (en) 2001-07-18 2001-09-12 Bayer Ag Imidazopyridinones
SE0104331D0 (sv) 2001-12-19 2001-12-19 Astrazeneca Ab Novel compounds
EP2324830A1 (en) * 2002-03-05 2011-05-25 TransTech Pharma Inc. Process for the preparation of a monocyclic azole derivative that inhibits the interaction of ligands with rage
US20060111416A1 (en) 2004-11-24 2006-05-25 Lane Charlotte A L Octahydropyrrolo[3,4-C]pyrrole derivatives
EP2061768A2 (en) 2006-09-28 2009-05-27 Exelixis, Inc. Imidazole-4,5-dicarboxamide derivatives as jak-2 modulators
JP2010522177A (ja) 2007-03-23 2010-07-01 アムジエン・インコーポレーテツド 複素環化合物およびその使用
EP1986009A1 (en) * 2007-04-26 2008-10-29 Active Biotech AB Screening method
WO2008157270A1 (en) 2007-06-13 2008-12-24 Smithkline Beecham Corporation Farnesoid x receptor agonists
WO2009093747A1 (en) * 2008-01-22 2009-07-30 Takeda Pharmaceutical Company Limited Tricyclic compounds having corticotropin-releasing factor antagonistic activity and pharmaceutical compositions containing them
TW201004941A (en) 2008-07-16 2010-02-01 Wyeth Corp Alpha7 nicotinic acetylcholine receptor inhibitors
EP2403833A4 (en) 2009-03-02 2012-08-29 Sirtris Pharmaceuticals Inc 8-SUBSTITUTED QUINOLINES AND RELATED ANALOGUES USED AS SIRTUINE MODULATORS
RU2628616C2 (ru) 2011-11-03 2017-08-21 Ф. Хоффманн-Ля Рош Аг Бициклические соединения пиперазина
GB201321728D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents

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