JP2016535019A5 - - Google Patents

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Publication number
JP2016535019A5
JP2016535019A5 JP2016525563A JP2016525563A JP2016535019A5 JP 2016535019 A5 JP2016535019 A5 JP 2016535019A5 JP 2016525563 A JP2016525563 A JP 2016525563A JP 2016525563 A JP2016525563 A JP 2016525563A JP 2016535019 A5 JP2016535019 A5 JP 2016535019A5
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JP
Japan
Prior art keywords
adenosine
pain
methyl
group
bromothien
Prior art date
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Application number
JP2016525563A
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English (en)
Japanese (ja)
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JP6534997B2 (ja
JP2016535019A (ja
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Priority claimed from PCT/US2014/061734 external-priority patent/WO2015061426A1/en
Publication of JP2016535019A publication Critical patent/JP2016535019A/ja
Publication of JP2016535019A5 publication Critical patent/JP2016535019A5/ja
Application granted granted Critical
Publication of JP6534997B2 publication Critical patent/JP6534997B2/ja
Active legal-status Critical Current
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JP2016525563A 2013-10-23 2014-10-22 神経変性疾患及び疼痛の予防及び治療における使用のための化合物 Active JP6534997B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361894699P 2013-10-23 2013-10-23
US61/894,699 2013-10-23
PCT/US2014/061734 WO2015061426A1 (en) 2013-10-23 2014-10-22 Compounds for use in prevention and treatment of neurodegenerative diseases and pain

Publications (3)

Publication Number Publication Date
JP2016535019A JP2016535019A (ja) 2016-11-10
JP2016535019A5 true JP2016535019A5 (https=) 2017-11-09
JP6534997B2 JP6534997B2 (ja) 2019-06-26

Family

ID=52993493

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2016525563A Active JP6534997B2 (ja) 2013-10-23 2014-10-22 神経変性疾患及び疼痛の予防及び治療における使用のための化合物

Country Status (14)

Country Link
US (1) US10301348B2 (https=)
EP (1) EP3060566B1 (https=)
JP (1) JP6534997B2 (https=)
KR (1) KR102313314B1 (https=)
CN (1) CN106414456B (https=)
AU (1) AU2014340114B2 (https=)
BR (1) BR112016008901B1 (https=)
CA (1) CA2927699C (https=)
IL (1) IL245103B (https=)
MX (1) MX367707B (https=)
RU (1) RU2695358C2 (https=)
SG (1) SG11201603063WA (https=)
WO (1) WO2015061426A1 (https=)
ZA (1) ZA201603118B (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG11201707513QA (en) * 2015-05-29 2017-10-30 Univ Leland Stanford Junior Nucleoside agents for the reduction of the deleterious activity of extended nucleotide repeat containing genes
US11753432B2 (en) 2017-01-27 2023-09-12 Academia Sinica Compound with analgesic effect for use in prevention and treatment of pain
CA3250090A1 (en) * 2022-02-10 2023-08-17 Academia Sinica METHOD FOR TREATMENT OF A SPINAL CORD INJURY AND CORRESPONDING COMPOSITION
TWI910441B (zh) * 2022-07-07 2026-01-01 中央研究院 治療思覺失調症之方法及用於其中之組成物
JP2026503973A (ja) * 2022-12-29 2026-02-03 中央研究院 睡眠障害を処置する方法及びそれに使用するための組成物
EP4680230A1 (en) * 2023-03-17 2026-01-21 Academia Sinica Method of treating tuberous sclerosis complex or epilepsy and composition for use therein

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1988003148A2 (en) 1986-10-31 1988-05-05 Warner-Lambert Company Heteroaromatic derivatives of adenoside
US5034381A (en) * 1988-01-07 1991-07-23 Ciba-Geigy Corporation 2-(substituted amino) adenosines as antihypertensives
AU654507B2 (en) * 1990-09-25 1994-11-10 Rhone-Poulenc Rorer International (Holdings) Inc. Compounds having antihypertensive and anti-ischemic properties
US5561134A (en) * 1990-09-25 1996-10-01 Rhone-Poulenc Rorer Pharmaceuticals Inc. Compounds having antihypertensive, cardioprotective, anti-ischemic and antilipolytic properties
UY27939A1 (es) * 2002-08-21 2004-03-31 Glaxo Group Ltd Compuestos
US20120295863A1 (en) 2009-11-13 2012-11-22 Yun-Lian Lin Dual-Action Compounds Targeting Adenosine A2A Receptor and Adenosine Transporter for Prevention and Treatment of Neurodegenerative Diseases
CN102812033B (zh) 2009-12-10 2015-11-25 中国医学科学院药物研究所 N6-取代腺苷衍生物和n6-取代腺嘌呤衍生物及其用途
CA2897675C (en) 2012-02-09 2017-07-18 Brandbumps, Llc Decorative detectable warning panel having improved grip
CN104363757B (zh) 2012-02-11 2017-05-24 中央研究院 治疗疼痛的方法及组合物

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