JP2016520095A5 - - Google Patents
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- Publication number
- JP2016520095A5 JP2016520095A5 JP2016514971A JP2016514971A JP2016520095A5 JP 2016520095 A5 JP2016520095 A5 JP 2016520095A5 JP 2016514971 A JP2016514971 A JP 2016514971A JP 2016514971 A JP2016514971 A JP 2016514971A JP 2016520095 A5 JP2016520095 A5 JP 2016520095A5
- Authority
- JP
- Japan
- Prior art keywords
- crystallized
- isolated
- compound
- seed crystals
- polymorph form
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 229940125904 compound 1 Drugs 0.000 description 2
- 239000013078 crystal Substances 0.000 description 2
- 150000003556 thioamides Chemical class 0.000 description 2
- 239000002904 solvent Substances 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361825139P | 2013-05-20 | 2013-05-20 | |
| US61/825,139 | 2013-05-20 | ||
| PCT/US2014/038132 WO2014189753A1 (en) | 2013-05-20 | 2014-05-15 | Solid forms of fungicidal pyrazoles |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2016520095A JP2016520095A (ja) | 2016-07-11 |
| JP2016520095A5 true JP2016520095A5 (OSRAM) | 2017-06-01 |
Family
ID=50885022
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016514971A Pending JP2016520095A (ja) | 2013-05-20 | 2014-05-15 | 殺菌・殺カビ性ピラゾールの固体形態 |
Country Status (16)
| Country | Link |
|---|---|
| US (2) | US9688639B2 (OSRAM) |
| EP (1) | EP2999695A1 (OSRAM) |
| JP (1) | JP2016520095A (OSRAM) |
| KR (1) | KR20160009657A (OSRAM) |
| CN (1) | CN105308025A (OSRAM) |
| AR (1) | AR096365A1 (OSRAM) |
| AU (1) | AU2014268872A1 (OSRAM) |
| BR (1) | BR112015029006A2 (OSRAM) |
| CA (1) | CA2912067A1 (OSRAM) |
| MX (1) | MX2015015828A (OSRAM) |
| MY (1) | MY172149A (OSRAM) |
| RU (1) | RU2652138C2 (OSRAM) |
| TW (1) | TWI652012B (OSRAM) |
| UA (1) | UA120837C2 (OSRAM) |
| WO (1) | WO2014189753A1 (OSRAM) |
| ZA (1) | ZA201508015B (OSRAM) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI504350B (zh) | 2010-09-01 | 2015-10-21 | Du Pont | 殺真菌吡唑及其混合物 |
| CN104673605A (zh) * | 2014-12-04 | 2015-06-03 | 贵州宝洞酱藏酒业有限公司 | 一种养生酒及其制备方法 |
| AR106472A1 (es) | 2015-10-26 | 2018-01-17 | Gilead Apollo Llc | Inhibidores de acc y usos de los mismos |
| JP2019502660A (ja) | 2015-11-25 | 2019-01-31 | ギリアド アポロ, エルエルシー | ピラゾールacc阻害剤およびその使用 |
| BR112018010453B1 (pt) | 2015-11-25 | 2022-06-14 | Gilead Apollo, Llc | Compostos triazólicos inibindores de acetil coa carboxilase (acc) |
| EA201890910A1 (ru) * | 2015-11-25 | 2018-11-30 | Джилид Аполло, Ллс | ФУНГИЦИДНЫЕ КОМПОЗИЦИИ, СОДЕРЖАЩИЕ ПРОИЗВОДНЫЕ 2,4-ДИОКСО-1,4-ДИГИДРОТИЕНО[2,3-d]ПИРИМИДИНА |
| EA201890949A1 (ru) | 2015-11-25 | 2018-12-28 | Джилид Аполло, Ллс | СЛОЖНОЭФИРНЫЕ ИНГИБИТОРЫ АЦЕТИЛ-КоА-КАРБОКСИЛАЗЫ И ВАРИАНТЫ ИХ ПРИМЕНЕНИЯ |
| MA49639A (fr) * | 2017-07-17 | 2020-05-27 | Adama Makhteshim Ltd | Polymorphes de 5-fluoro-4-imino-3-méthyl-1-tosyl-3,4-dihydropyrimidin-2-one |
| KR20220034818A (ko) | 2019-07-10 | 2022-03-18 | 바이엘 악티엔게젤샤프트 | 2-(페닐이미노)-1,3-티아졸리딘-4-온의 제조 방법 |
| KR20220034151A (ko) | 2019-07-10 | 2022-03-17 | 바이엘 악티엔게젤샤프트 | 2-(페닐이미노)-1,3-티아졸리딘-4-온의 제조 방법 |
| CN115583898A (zh) * | 2021-07-06 | 2023-01-10 | 苏州开拓药业股份有限公司 | 一种异硫氰酸芳基酯的制备方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2004002393A (ja) * | 2002-04-19 | 2004-01-08 | Nissan Chem Ind Ltd | 結晶多形インド−ル化合物およびその製造方法 |
| UY30645A1 (es) * | 2006-10-13 | 2008-05-02 | Basf Ag | Forma cristalina de 2-cloro-5-[3,6-dihidro-3-metil-2,6-dioxo-4-(trifluorometil)-1-(2h)-pirimidinil]-4-fluoro-n-[ [metil(1-metiletil) amino]sulfonil]benzamida |
| KR20100043069A (ko) * | 2007-07-12 | 2010-04-27 | 바스프 에스이 | 3-(디플루오르메틸)-1-메틸-n-(3',4',5'-트리플루오르[1,1'-바이페닐]-2-일)-1h-피라졸-4-카르복사미드의 신규 결정질 형태 |
| AR075713A1 (es) * | 2009-03-03 | 2011-04-20 | Du Pont | Pirazoles fungicidas |
| TWI504350B (zh) * | 2010-09-01 | 2015-10-21 | Du Pont | 殺真菌吡唑及其混合物 |
| TW201245155A (en) * | 2010-09-01 | 2012-11-16 | Du Pont | Fungicidal pyrazoles |
| TWI568721B (zh) * | 2012-02-01 | 2017-02-01 | 杜邦股份有限公司 | 殺真菌之吡唑混合物 |
-
2014
- 2014-04-22 TW TW103114460A patent/TWI652012B/zh not_active IP Right Cessation
- 2014-05-15 BR BR112015029006A patent/BR112015029006A2/pt not_active Application Discontinuation
- 2014-05-15 MY MYPI2015703865A patent/MY172149A/en unknown
- 2014-05-15 CA CA2912067A patent/CA2912067A1/en not_active Abandoned
- 2014-05-15 MX MX2015015828A patent/MX2015015828A/es unknown
- 2014-05-15 EP EP14728397.2A patent/EP2999695A1/en not_active Withdrawn
- 2014-05-15 UA UAA201512219A patent/UA120837C2/uk unknown
- 2014-05-15 AU AU2014268872A patent/AU2014268872A1/en not_active Abandoned
- 2014-05-15 JP JP2016514971A patent/JP2016520095A/ja active Pending
- 2014-05-15 RU RU2015154479A patent/RU2652138C2/ru not_active IP Right Cessation
- 2014-05-15 WO PCT/US2014/038132 patent/WO2014189753A1/en not_active Ceased
- 2014-05-15 US US14/888,835 patent/US9688639B2/en not_active Expired - Fee Related
- 2014-05-15 CN CN201480029192.7A patent/CN105308025A/zh active Pending
- 2014-05-15 KR KR1020157035586A patent/KR20160009657A/ko not_active Withdrawn
- 2014-05-20 AR ARP140102009A patent/AR096365A1/es unknown
-
2015
- 2015-10-28 ZA ZA2015/08015A patent/ZA201508015B/en unknown
-
2017
- 2017-05-25 US US15/604,712 patent/US20170260142A1/en not_active Abandoned
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