JP2016508506A5 - - Google Patents

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Publication number
JP2016508506A5
JP2016508506A5 JP2015556454A JP2015556454A JP2016508506A5 JP 2016508506 A5 JP2016508506 A5 JP 2016508506A5 JP 2015556454 A JP2015556454 A JP 2015556454A JP 2015556454 A JP2015556454 A JP 2015556454A JP 2016508506 A5 JP2016508506 A5 JP 2016508506A5
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JP
Japan
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JP2015556454A
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English (en)
Japanese (ja)
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JP2016508506A (ja
JP6314335B2 (ja
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Priority claimed from PCT/EP2014/051878 external-priority patent/WO2014122067A1/en
Publication of JP2016508506A publication Critical patent/JP2016508506A/ja
Publication of JP2016508506A5 publication Critical patent/JP2016508506A5/ja
Application granted granted Critical
Publication of JP6314335B2 publication Critical patent/JP6314335B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2015556454A 2013-02-06 2014-01-31 新しいインダニルオキシジヒドロベンゾフラニル酢酸 Expired - Fee Related JP6314335B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP13154261 2013-02-06
EP13154261.5 2013-02-06
PCT/EP2014/051878 WO2014122067A1 (en) 2013-02-06 2014-01-31 New indanyloxydihydrobenzofuranylacetic acids

Publications (3)

Publication Number Publication Date
JP2016508506A JP2016508506A (ja) 2016-03-22
JP2016508506A5 true JP2016508506A5 (enExample) 2017-03-09
JP6314335B2 JP6314335B2 (ja) 2018-04-25

Family

ID=47681765

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015556454A Expired - Fee Related JP6314335B2 (ja) 2013-02-06 2014-01-31 新しいインダニルオキシジヒドロベンゾフラニル酢酸

Country Status (7)

Country Link
US (1) US8927531B2 (enExample)
EP (1) EP2953681B1 (enExample)
JP (1) JP6314335B2 (enExample)
AR (1) AR095163A1 (enExample)
TW (1) TW201518284A (enExample)
UY (1) UY35312A (enExample)
WO (1) WO2014122067A1 (enExample)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3068788A1 (en) 2013-11-14 2016-09-21 Cadila Healthcare Limited Novel heterocyclic compounds
CN105566263A (zh) * 2016-01-27 2016-05-11 中国药科大学 一类新型含氮杂环衍生物、其制备方法及其作为药物的用途
JOP20190060A1 (ar) 2016-09-26 2019-03-26 Chugai Pharmaceutical Co Ltd مشتق بيرازولو بيريدين له تأثير مساعد لمستقبل glp-1
BR102018007822A2 (pt) 2017-04-20 2018-11-06 Gilead Sciences, Inc. composto, métodos para inibir pd-1, pd-l1 e/ou interação de pd-1/pd-l1 e para tratamento de câncer, composição farmacêutica, e, kit para tratamento de ou prevenção de câncer ou uma doença ou condição
JP7461104B2 (ja) * 2017-11-29 2024-04-03 中外製薬株式会社 Glp-1受容体アゴニスト作用を持つピラゾロピリジン誘導体を含有する医薬組成物
KR102708681B1 (ko) 2018-02-13 2024-09-26 길리애드 사이언시즈, 인코포레이티드 Pd-1/pd-l1 억제제
EP4600247A3 (en) 2018-04-19 2025-11-19 Gilead Sciences, Inc. Pd-1/pd-l1 inhibitors
UA126421C2 (uk) 2018-07-13 2022-09-28 Гіліад Сайєнсіз, Інк. Інгібітори pd-1/pd-l1
US11236085B2 (en) 2018-10-24 2022-02-01 Gilead Sciences, Inc. PD-1/PD-L1 inhibitors
BR112022006546A2 (pt) 2019-10-07 2022-08-30 Kallyope Inc Agonistas de gpr119
PE20231066A1 (es) 2020-02-07 2023-07-17 Gasherbrum Bio Inc Agonistas heterociclicos de glp-1
CA3173731A1 (en) 2020-02-28 2021-09-02 Kallyope, Inc. Gpr40 agonists
CN116323608A (zh) 2020-05-19 2023-06-23 卡尔优普公司 Ampk活化剂
EP4172162A4 (en) 2020-06-26 2024-08-07 Kallyope, Inc. AMPK ACTIVATORS
JP7858636B2 (ja) 2020-09-10 2026-05-14 ガシャーブラム・バイオ・インコーポレイテッド ヘテロ環glp-1アゴニスト
IL322686A (en) 2023-02-16 2025-10-01 Gasherbrum Bio Inc Heterocyclic glp-1 agonists

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4594611B2 (ja) * 2002-11-08 2010-12-08 武田薬品工業株式会社 受容体機能調節剤
EP1559422B1 (en) 2002-11-08 2014-04-30 Takeda Pharmaceutical Company Limited Receptor function controlling agent
JP4805552B2 (ja) * 2003-05-30 2011-11-02 武田薬品工業株式会社 縮合環化合物
EP1924546A1 (en) 2005-09-14 2008-05-28 Amgen, Inc Conformationally constrained 3- (4-hydroxy-phenyl) - substituted-propanoic acids useful for treating metabolic disorders
CA2646430A1 (en) * 2006-03-14 2007-09-20 Amgen Inc. Bicyclic carboxylic acid derivatives useful for treating metabolic disorders
CL2007001873A1 (es) 2006-06-27 2008-01-04 Takeda Pharmaceutical Acido((3s))-6-((¨2,6-dimetil-4-(3-(metilsulfonil)-propoxi)bifenil-3-il)metoxi-2,3-dihidro-1-benzofuran-3-il)acetico o una sal del mismo
CA2727340A1 (en) 2008-06-25 2009-12-30 Daiichi Sankyo Company, Limited Carboxylic acid compound
WO2010143733A1 (en) * 2009-06-09 2010-12-16 Takeda Pharmaceutical Company Limited Novel fused cyclic compound and use thereof
EP2646425B1 (en) 2010-12-01 2015-06-10 Boehringer Ingelheim International Gmbh Indanyloxydihydrobenzofuranylacetic acids useful for the treatment of metabolic syndrome
US8809376B2 (en) * 2012-04-30 2014-08-19 Boehringer Ingelheim International Gmbh Indanyloxydihydrobenzofuranylacetic acids

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