JP2015523337A5 - - Google Patents
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- Publication number
- JP2015523337A5 JP2015523337A5 JP2015514142A JP2015514142A JP2015523337A5 JP 2015523337 A5 JP2015523337 A5 JP 2015523337A5 JP 2015514142 A JP2015514142 A JP 2015514142A JP 2015514142 A JP2015514142 A JP 2015514142A JP 2015523337 A5 JP2015523337 A5 JP 2015523337A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- contacted
- solution
- tms
- acetonitrile
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261650553P | 2012-05-23 | 2012-05-23 | |
| US61/650,553 | 2012-05-23 | ||
| PCT/US2013/042150 WO2013177243A1 (en) | 2012-05-23 | 2013-05-22 | Sulfilimine and sulphoxide methods for producing festinavir |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2015523337A JP2015523337A (ja) | 2015-08-13 |
| JP2015523337A5 true JP2015523337A5 (https=) | 2016-07-07 |
Family
ID=48534517
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015514142A Pending JP2015523337A (ja) | 2012-05-23 | 2013-05-22 | フェスチナビルを製造するためのスルフィリミンおよびスルホキシド方法 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US9249171B2 (https=) |
| EP (1) | EP2852583A1 (https=) |
| JP (1) | JP2015523337A (https=) |
| CN (1) | CN104379571A (https=) |
| WO (1) | WO2013177243A1 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20160060252A1 (en) | 2013-04-16 | 2016-03-03 | Bristol-Myers Squibb Company | 5-methyluridine method for producing festinavir |
| WO2014201122A1 (en) | 2013-06-13 | 2014-12-18 | Bristol-Myers Squibb Company | Tert-butyl-sulphoxide method for producing festinavir |
| US10301624B2 (en) | 2014-06-25 | 2019-05-28 | The General Hospital Corporation | Targeting human satellite II (HSATII) |
| JP7025064B2 (ja) * | 2018-08-09 | 2022-02-24 | ヤマサ醤油株式会社 | ４’－置換ヌクレオシド誘導体の立体選択的合成法 |
| SG11202107145SA (en) | 2019-01-25 | 2021-08-30 | Univ Brown | Compositions and methods for treating, preventing or reversing age-associated inflammation and disorders |
| IL316425A (en) * | 2022-04-22 | 2024-12-01 | Rome Therapeutics Inc | Dihydro-3'-deoxy-4'-ethynylthymidines and related compounds and their uses in the treatment of medical conditions |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0454193A (ja) * | 1990-05-25 | 1992-02-21 | Japan Tobacco Inc | ２’，３’―ジデオキシ―２’，３’―ジデヒドロ―β―リボヌクレオシドの製造方法 |
| EA012844B1 (ru) * | 2003-02-19 | 2009-12-30 | Йельский Университет | Аналоги противовирусных нуклеозидов и способы лечения вирусных инфекций, в частности вич-инфекций |
| NZ567272A (en) | 2005-09-26 | 2012-02-24 | Pharmasset Inc | Modified 4'-nucleosides as antiviral agents |
| CN101784532B (zh) | 2007-06-29 | 2014-10-22 | 韩国化学研究院 | Hiv逆转录酶抑制剂 |
| US20090318380A1 (en) | 2007-11-20 | 2009-12-24 | Pharmasset, Inc. | 2',4'-substituted nucleosides as antiviral agents |
| WO2009084655A1 (ja) * | 2007-12-27 | 2009-07-09 | Oncolys Biopharma Inc. | 4'-エチニルd4Tの製造方法 |
| JP5485138B2 (ja) | 2008-03-28 | 2014-05-07 | 浜理薬品工業株式会社 | エチニルチミジン化合物の精製方法 |
| US8445669B2 (en) | 2008-04-10 | 2013-05-21 | Hamari Chemicals, Ltd. | Production process of ethynylthymidine compounds from 5-methyluridine as a starting material |
| DE102009034346B4 (de) | 2009-07-23 | 2013-01-24 | Kone Corp. | Antriebssystem für eine Personenförderanlage |
| EP2537851B1 (en) | 2010-02-15 | 2015-06-10 | Nissan Chemical Industries, Ltd. | Process for preparation of b-glycoside compounds |
| EP2537839B1 (en) | 2010-02-15 | 2016-12-14 | Nissan Chemical Industries, Ltd. | B-dihydrofuran deriving compound, method for producing b-dihydrofuran deriving compound or b-tetrahydrofuran deriving compound, b -glycoside compound, method for producing b-glycoside compound, and method for producing 4'-ethynyl d4t and analogue compounds thereof |
-
2013
- 2013-05-22 EP EP13725545.1A patent/EP2852583A1/en not_active Withdrawn
- 2013-05-22 WO PCT/US2013/042150 patent/WO2013177243A1/en not_active Ceased
- 2013-05-22 CN CN201380027023.5A patent/CN104379571A/zh active Pending
- 2013-05-22 JP JP2015514142A patent/JP2015523337A/ja active Pending
- 2013-05-22 US US14/402,231 patent/US9249171B2/en active Active
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