JP2015522544A5 - - Google Patents
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- Publication number
- JP2015522544A5 JP2015522544A5 JP2015513123A JP2015513123A JP2015522544A5 JP 2015522544 A5 JP2015522544 A5 JP 2015522544A5 JP 2015513123 A JP2015513123 A JP 2015513123A JP 2015513123 A JP2015513123 A JP 2015513123A JP 2015522544 A5 JP2015522544 A5 JP 2015522544A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- optionally substituted
- group
- aromatic heterocycle
- phenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 *C(*)N(C*CC(*)(NC(N)=NC(c1nc(*)c(N)nc1N)=O)N1)C*1=* Chemical compound *C(*)N(C*CC(*)(NC(N)=NC(c1nc(*)c(N)nc1N)=O)N1)C*1=* 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP12169577 | 2012-05-25 | ||
| EP12169577.9 | 2012-05-25 | ||
| PCT/EP2013/060282 WO2013174757A1 (en) | 2012-05-25 | 2013-05-17 | Tertiary amines, medicaments containing said amines, use thereof and processes for the preparation thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2015522544A JP2015522544A (ja) | 2015-08-06 |
| JP2015522544A5 true JP2015522544A5 (OSRAM) | 2016-07-07 |
| JP6204977B2 JP6204977B2 (ja) | 2017-09-27 |
Family
ID=48539098
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015513123A Active JP6204977B2 (ja) | 2012-05-25 | 2013-05-17 | 三級アミン、前記アミンを含む薬物、その使用及びその調製方法 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US9078909B2 (OSRAM) |
| EP (1) | EP2861577B1 (OSRAM) |
| JP (1) | JP6204977B2 (OSRAM) |
| WO (1) | WO2013174757A1 (OSRAM) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK3219705T3 (da) | 2005-12-28 | 2020-04-14 | Vertex Pharma | Farmaceutiske sammensætninger af den amorfe form af n-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinolin-3-carboxamid |
| JP6353032B2 (ja) * | 2013-04-30 | 2018-07-04 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ジアミノピラジン化合物、前記化合物を含有する医薬、その使用、およびその調製方法 |
| JP6543268B2 (ja) | 2014-04-15 | 2019-07-10 | バーテックス ファーマシューティカルズ インコーポレイテッドＶｅｒｔｅｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃｏｒｐｏｒａｔｅｄ | 嚢胞性線維症膜コンダクタンス調節因子が媒介する疾患を処置するための医薬組成物 |
| CN107250113B (zh) | 2014-10-07 | 2019-03-29 | 弗特克斯药品有限公司 | 囊性纤维化跨膜传导调节蛋白的调节剂的共晶 |
| CN115028661A (zh) * | 2022-05-19 | 2022-09-09 | 上海应用技术大学 | 一种4-氨基哌啶-1-甲基磷酸酯及其制备方法 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL6812003A (OSRAM) | 1967-09-07 | 1969-03-11 | ||
| US3953476A (en) | 1971-12-27 | 1976-04-27 | Merck & Co., Inc. | 3-Amino-5-sulfonylbenzoic acids |
| AU2001229501A1 (en) | 2000-01-24 | 2001-07-31 | Isis Pharmaceuticals, Inc. | Antisense modulation of inducible nitric oxide synthase expression |
| AU2004264441A1 (en) * | 2003-08-18 | 2005-02-24 | Parion Sciences, Inc. | Cyclic pyrazinoylguanidine sodium channel blockers |
| GB0526240D0 (en) * | 2005-12-22 | 2006-02-01 | Novartis Ag | Organic compounds |
| KR20100005730A (ko) | 2007-05-07 | 2010-01-15 | 노파르티스 아게 | 유기 화합물 |
| JP2011520831A (ja) | 2008-05-13 | 2011-07-21 | ノバルティス アーゲー | ３，５−ジアミノ−６−クロロ−ピラジン−２−カルボン酸誘導体および気道疾患処置用上皮性ナトリウムチャネルブロッカーとしてのその使用 |
| AR086745A1 (es) | 2011-06-27 | 2014-01-22 | Parion Sciences Inc | 3,5-diamino-6-cloro-n-(n-(4-(4-(2-(hexil(2,3,4,5,6-pentahidroxihexil)amino)etoxi)fenil)butil)carbamimidoil)pirazina-2-carboxamida |
| PL2723176T3 (pl) | 2011-06-27 | 2018-01-31 | Parion Sciences Inc | Chemicznie i metabolicznie stabilny dipeptyd o silnej aktywności blokera kanału sodowego |
-
2013
- 2013-05-17 JP JP2015513123A patent/JP6204977B2/ja active Active
- 2013-05-17 EP EP13726129.3A patent/EP2861577B1/en active Active
- 2013-05-17 WO PCT/EP2013/060282 patent/WO2013174757A1/en not_active Ceased
- 2013-05-22 US US13/899,762 patent/US9078909B2/en active Active
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