JP2014525432A5 - - Google Patents

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Publication number
JP2014525432A5
JP2014525432A5 JP2014527767A JP2014527767A JP2014525432A5 JP 2014525432 A5 JP2014525432 A5 JP 2014525432A5 JP 2014527767 A JP2014527767 A JP 2014527767A JP 2014527767 A JP2014527767 A JP 2014527767A JP 2014525432 A5 JP2014525432 A5 JP 2014525432A5
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Japan
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alkyl
hydrogen
cycloalkyl
independently
substituted
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JP2014527767A
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Japanese (ja)
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JP2014525432A (ja
JP6043355B2 (ja
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Priority claimed from PCT/IB2012/054198 external-priority patent/WO2013030713A1/en
Publication of JP2014525432A publication Critical patent/JP2014525432A/ja
Publication of JP2014525432A5 publication Critical patent/JP2014525432A5/ja
Application granted granted Critical
Publication of JP6043355B2 publication Critical patent/JP6043355B2/ja
Expired - Fee Related legal-status Critical Current
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JP2014527767A 2011-08-31 2012-08-17 ヘキサヒドロピラノ［３，４−ｄ］［１，３］チアジン−２−アミン化合物 Expired - Fee Related JP6043355B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161529367P 2011-08-31 2011-08-31
US61/529,367 2011-08-31
PCT/IB2012/054198 WO2013030713A1 (en) 2011-08-31 2012-08-17 Hexahydropyrano [3,4-d][1,3] thiazin-2-amine compounds

Publications (3)

Publication Number Publication Date
JP2014525432A JP2014525432A (ja) 2014-09-29
JP2014525432A5 true JP2014525432A5 (https=) 2015-09-24
JP6043355B2 JP6043355B2 (ja) 2016-12-14

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JP2014527767A Expired - Fee Related JP6043355B2 (ja) 2011-08-31 2012-08-17 ヘキサヒドロピラノ［３，４−ｄ］［１，３］チアジン−２−アミン化合物

Country Status (8)

Country Link
US (2) US8933221B2 (https=)
EP (1) EP2751116B1 (https=)
JP (1) JP6043355B2 (https=)
AR (1) AR087742A1 (https=)
ES (1) ES2605565T3 (https=)
TW (1) TW201326182A (https=)
UY (1) UY34302A (https=)
WO (1) WO2013030713A1 (https=)

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JP7149271B2 (ja) 2016-12-15 2022-10-06 アムジエン・インコーポレーテツド β－セクレターゼ阻害剤としての１，４－チアジンジオキシドおよび１，２，４－チアジアジンジオキシド誘導体ならびに使用方法
US10947223B2 (en) 2016-12-15 2021-03-16 Amgen Inc. Substituted oxazines as beta-secretase inhibitors
JP7149272B2 (ja) 2016-12-15 2022-10-06 アムジエン・インコーポレーテツド β－セクレターゼ阻害剤としてのチアジン誘導体および使用方法
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