JP2014508784A5 - - Google Patents
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- Publication number
- JP2014508784A5 JP2014508784A5 JP2014500216A JP2014500216A JP2014508784A5 JP 2014508784 A5 JP2014508784 A5 JP 2014508784A5 JP 2014500216 A JP2014500216 A JP 2014500216A JP 2014500216 A JP2014500216 A JP 2014500216A JP 2014508784 A5 JP2014508784 A5 JP 2014508784A5
- Authority
- JP
- Japan
- Prior art keywords
- treatment
- radiolabeled compound
- cancer
- radioactive imaging
- breast cancer
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 206010006187 Breast cancer Diseases 0.000 claims 1
- 208000026310 Breast neoplasm Diseases 0.000 claims 1
- 206010060862 Prostate cancer Diseases 0.000 claims 1
- 208000000236 Prostatic Neoplasms Diseases 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 238000003384 imaging method Methods 0.000 claims 1
- 230000002285 radioactive effect Effects 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161467764P | 2011-03-25 | 2011-03-25 | |
| US61/467,764 | 2011-03-25 | ||
| PCT/CA2012/000316 WO2012129673A1 (en) | 2011-03-25 | 2012-03-26 | INHIBITORS OF 17ß-HSD1, 17ß-HSD3 AND 17ß-HSD10 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017253315A Division JP6727184B2 (ja) | 2011-03-25 | 2017-12-28 | １７β−ＨＳＤ１、１７β−ＨＳＤ３、および１７β−ＨＳＤ１０の阻害剤 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2014508784A JP2014508784A (ja) | 2014-04-10 |
| JP2014508784A5 true JP2014508784A5 (enExample) | 2016-10-27 |
Family
ID=46929260
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014500216A Withdrawn JP2014508784A (ja) | 2011-03-25 | 2012-03-26 | １７β−ＨＳＤ１、１７β−ＨＳＤ３、および１７β−ＨＳＤ１０の阻害剤 |
| JP2017253315A Expired - Fee Related JP6727184B2 (ja) | 2011-03-25 | 2017-12-28 | １７β−ＨＳＤ１、１７β−ＨＳＤ３、および１７β−ＨＳＤ１０の阻害剤 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017253315A Expired - Fee Related JP6727184B2 (ja) | 2011-03-25 | 2017-12-28 | １７β−ＨＳＤ１、１７β−ＨＳＤ３、および１７β−ＨＳＤ１０の阻害剤 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US11072632B2 (enExample) |
| EP (1) | EP2688901B1 (enExample) |
| JP (2) | JP2014508784A (enExample) |
| AU (1) | AU2012234682A1 (enExample) |
| CA (1) | CA2830984C (enExample) |
| WO (1) | WO2012129673A1 (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW201522359A (zh) * | 2013-06-25 | 2015-06-16 | Forendo Pharma Ltd | 治療用活性雌三烯噻唑衍生物 |
| CN105518016B (zh) * | 2013-06-25 | 2020-10-23 | 佛恩多制药有限公司 | 治疗活性的作为1型17β-羟基类固醇脱氢酶抑制剂的雌三烯噻唑衍生物 |
| CA2950800C (en) * | 2014-05-09 | 2023-01-10 | Tangent Reprofiling Limited | Modulators of androgen synthesis |
| CN106687471B (zh) * | 2014-09-11 | 2018-10-30 | 拜耳医药股份公司 | 3-氮或者硫取代的雌甾-1,3,5(10),16-四烯akr1c3抑制剂 |
| CZ307437B6 (cs) * | 2016-06-07 | 2018-08-22 | Ăšstav organickĂ© chemie a biochemie AV ÄŚR, v.v.i. | 15β-substituované deriváty estronu jako selektivní inhibitory 17β-hydroxysteoiddehydrogenáz |
| IL294140B2 (en) | 2017-06-08 | 2024-09-01 | Forendo Pharma Ltd | 15beta-(3-PROPANAMIDO)-SUBSTITUTED ESTRA-1,3,5(10)-TRIEN-17-OXIMES FOR USE IN INHIBITION OF 17beta-HYDROXYSTEROID DEHYDROGENASES |
| WO2024020520A2 (en) * | 2022-07-20 | 2024-01-25 | Board Of Regents, The University Of Texas System | Enzyme compositions, steroid derivatives, enzyme inhibitors, and methods of making same for pharmaceutical applications |
| WO2025035212A1 (en) * | 2023-08-15 | 2025-02-20 | UNIVERSITé LAVAL | Irreversible 17beta-hsd1 inhibitors |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5232917A (en) * | 1987-08-25 | 1993-08-03 | University Of Southern California | Methods, compositions, and compounds for allosteric modulation of the GABA receptor by members of the androstane and pregnane series |
| FI101601B1 (fi) | 1987-09-24 | 1998-07-31 | Jencap Research Ltd | Ehkäisyvalmiste sekä estrogeenin ja progestiinin käyttö ehkäisyvalmisteen valmistusmenetelmässä |
| IL112778A0 (en) * | 1994-03-04 | 1995-05-26 | Merck & Co Inc | Substituted heterocycles, their preparation and pharmaceutical compositions containing them |
| US5952319A (en) * | 1997-11-26 | 1999-09-14 | Research Triangle Institute | Androgenic steroid compounds and a method of making and using the same |
| US6933312B2 (en) * | 2002-10-07 | 2005-08-23 | Agouron Pharmaceuticals, Inc. | Pyrazole derivatives |
| TWI331154B (en) | 2003-11-12 | 2010-10-01 | Solvay Pharm Gmbh | Novel 17-hydroxysteroid dehydrogenase type i inhibitors |
| BRPI0611623A2 (pt) | 2005-05-26 | 2010-09-21 | Solvay Pharm Gmbh | inibidores das 17beta-hsd1 e sts |
| US10174070B2 (en) * | 2005-09-30 | 2019-01-08 | Endece Llc | 6-substituted estradiol derivatives and methods of use |
| WO2008034796A2 (en) | 2006-09-19 | 2008-03-27 | Solvay Pharmaceuticals Gmbh | Estratriene derivatives and their uses as 17beta-hydr0xyster0id dehydrogenase inhibitors |
| JP5264760B2 (ja) * | 2006-11-30 | 2013-08-14 | アボット プロダクツ ゲゼルシャフト ミット ベシュレンクテル ハフツング | １７β−ＨＳＤインヒビターとしての置換エストラトリエン誘導体 |
| WO2008089093A2 (en) | 2007-01-12 | 2008-07-24 | Quatrx Pharmaceuticals Company | Efficient processes for preparing steroids and vitamin d derivatives with the unnatural configuration at c20 (20 alpha-methyl) from pregnenolone |
| EP2014672A1 (en) * | 2007-07-12 | 2009-01-14 | Bayer Schering Pharma Aktiengesellschaft | 8-beta-substituted estratrienes as selectively active estrogens |
-
2012
- 2012-03-26 EP EP12765822.7A patent/EP2688901B1/en active Active
- 2012-03-26 US US14/007,577 patent/US11072632B2/en not_active Expired - Fee Related
- 2012-03-26 JP JP2014500216A patent/JP2014508784A/ja not_active Withdrawn
- 2012-03-26 CA CA2830984A patent/CA2830984C/en active Active
- 2012-03-26 WO PCT/CA2012/000316 patent/WO2012129673A1/en not_active Ceased
- 2012-03-26 AU AU2012234682A patent/AU2012234682A1/en not_active Abandoned
-
2017
- 2017-12-28 JP JP2017253315A patent/JP6727184B2/ja not_active Expired - Fee Related
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