JP2014508784A5 - - Google Patents
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- Publication number
- JP2014508784A5 JP2014508784A5 JP2014500216A JP2014500216A JP2014508784A5 JP 2014508784 A5 JP2014508784 A5 JP 2014508784A5 JP 2014500216 A JP2014500216 A JP 2014500216A JP 2014500216 A JP2014500216 A JP 2014500216A JP 2014508784 A5 JP2014508784 A5 JP 2014508784A5
- Authority
- JP
- Japan
- Prior art keywords
- treatment
- radiolabeled compound
- cancer
- radioactive imaging
- breast cancer
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 206010006187 Breast cancer Diseases 0.000 claims 1
- 208000026310 Breast neoplasm Diseases 0.000 claims 1
- 206010060862 Prostate cancer Diseases 0.000 claims 1
- 208000000236 Prostatic Neoplasms Diseases 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 238000003384 imaging method Methods 0.000 claims 1
- 230000002285 radioactive effect Effects 0.000 claims 1
Claims (1)
- 放射性イメージングまたは乳癌または前立腺癌の治療のための、請求項45に記載の放
射標識化合物。
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201161467764P | 2011-03-25 | 2011-03-25 | |
US61/467,764 | 2011-03-25 | ||
PCT/CA2012/000316 WO2012129673A1 (en) | 2011-03-25 | 2012-03-26 | INHIBITORS OF 17ß-HSD1, 17ß-HSD3 AND 17ß-HSD10 |
Related Child Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2017253315A Division JP6727184B2 (ja) | 2011-03-25 | 2017-12-28 | 17β−HSD1、17β−HSD3、および17β−HSD10の阻害剤 |
Publications (2)
Publication Number | Publication Date |
---|---|
JP2014508784A JP2014508784A (ja) | 2014-04-10 |
JP2014508784A5 true JP2014508784A5 (ja) | 2016-10-27 |
Family
ID=46929260
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2014500216A Withdrawn JP2014508784A (ja) | 2011-03-25 | 2012-03-26 | 17β−HSD1、17β−HSD3、および17β−HSD10の阻害剤 |
JP2017253315A Active JP6727184B2 (ja) | 2011-03-25 | 2017-12-28 | 17β−HSD1、17β−HSD3、および17β−HSD10の阻害剤 |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2017253315A Active JP6727184B2 (ja) | 2011-03-25 | 2017-12-28 | 17β−HSD1、17β−HSD3、および17β−HSD10の阻害剤 |
Country Status (6)
Country | Link |
---|---|
US (1) | US11072632B2 (ja) |
EP (1) | EP2688901B1 (ja) |
JP (2) | JP2014508784A (ja) |
AU (1) | AU2012234682A1 (ja) |
CA (1) | CA2830984C (ja) |
WO (1) | WO2012129673A1 (ja) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US9850272B2 (en) | 2013-06-25 | 2017-12-26 | Forendo Pharma Ltd. | Therapeutically active estratrienthiazole derivatives as inhibitors of 17.beta-hydroxy-steroid dehydrogenase, type 1 |
US10377791B2 (en) | 2013-06-25 | 2019-08-13 | Forendo Pharma Ltd. | Therapeutically active estratrienthiazole derivatives as inhibitors of 17 B-hydroxysteroid dehydrogenase, type 1 |
WO2015169971A1 (en) * | 2014-05-09 | 2015-11-12 | Tangent Reprofiling Limited | Modulators of androgen synthesis |
JP6407415B2 (ja) * | 2014-09-11 | 2018-10-17 | バイエル・ファルマ・アクティエンゲゼルシャフト | 3−窒素または硫黄置換エストラ−1,3,5(10),16−テトラエンakr1c3阻害剤 |
CZ307437B6 (cs) | 2016-06-07 | 2018-08-22 | Ăšstav organickĂ© chemie a biochemie AV ÄŚR, v.v.i. | 15β-substituované deriváty estronu jako selektivní inhibitory 17β-hydroxysteoiddehydrogenáz |
UA126342C2 (uk) | 2017-06-08 | 2022-09-21 | Форендо Фарма Лтд | 15-бета-[3-пропанамідо]-заміщені естра-1,3,5(10)-трієн-17-он-сполуки і їх 17-оксими для використання в інгібуванні 17-бета-гідроксистероїддегідрогеназ |
WO2024020520A2 (en) * | 2022-07-20 | 2024-01-25 | Board Of Regents, The University Of Texas System | Enzyme compositions, steroid derivatives, enzyme inhibitors, and methods of making same for pharmaceutical applications |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5232917A (en) * | 1987-08-25 | 1993-08-03 | University Of Southern California | Methods, compositions, and compounds for allosteric modulation of the GABA receptor by members of the androstane and pregnane series |
EP0559240B1 (en) * | 1987-09-24 | 2001-12-05 | Jencap Research Limited | Contraceptive packages containing oestrogen and progestin |
TW385308B (en) * | 1994-03-04 | 2000-03-21 | Merck & Co Inc | Prodrugs of morpholine tachykinin receptor antagonists |
US5952319A (en) * | 1997-11-26 | 1999-09-14 | Research Triangle Institute | Androgenic steroid compounds and a method of making and using the same |
US6933312B2 (en) * | 2002-10-07 | 2005-08-23 | Agouron Pharmaceuticals, Inc. | Pyrazole derivatives |
TWI331154B (en) | 2003-11-12 | 2010-10-01 | Solvay Pharm Gmbh | Novel 17-hydroxysteroid dehydrogenase type i inhibitors |
CN102796160A (zh) | 2005-05-26 | 2012-11-28 | 索尔瓦药物有限公司 | 17β-HSD1和STS抑制剂 |
US10174070B2 (en) * | 2005-09-30 | 2019-01-08 | Endece Llc | 6-substituted estradiol derivatives and methods of use |
AU2007299010B2 (en) * | 2006-09-19 | 2013-01-31 | Solvay Pharmaceuticals Gmbh | Estratriene derivatives and their uses as 17beta-hydroxysteroid dehydrogenase inhibitors |
RU2453554C2 (ru) | 2006-11-30 | 2012-06-20 | Зольвай Фармасьютиклз Гмбх | Замещенные производные эстратриена как ингибиторы 17бета hsd |
US20080171728A1 (en) | 2007-01-12 | 2008-07-17 | Quatrx Pharmaceuticals Co. | Efficient Process for Preparing Steroids and Vitamin D Derivatives With the Unnatural Configuration at C20 (20 Alpha-Methyl) from Pregnenolone |
EP2014672A1 (en) * | 2007-07-12 | 2009-01-14 | Bayer Schering Pharma Aktiengesellschaft | 8-beta-substituted estratrienes as selectively active estrogens |
-
2012
- 2012-03-26 EP EP12765822.7A patent/EP2688901B1/en active Active
- 2012-03-26 US US14/007,577 patent/US11072632B2/en active Active
- 2012-03-26 JP JP2014500216A patent/JP2014508784A/ja not_active Withdrawn
- 2012-03-26 CA CA2830984A patent/CA2830984C/en active Active
- 2012-03-26 WO PCT/CA2012/000316 patent/WO2012129673A1/en active Application Filing
- 2012-03-26 AU AU2012234682A patent/AU2012234682A1/en not_active Abandoned
-
2017
- 2017-12-28 JP JP2017253315A patent/JP6727184B2/ja active Active
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