JP2014508784A5 - - Google Patents

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Publication number
JP2014508784A5
JP2014508784A5 JP2014500216A JP2014500216A JP2014508784A5 JP 2014508784 A5 JP2014508784 A5 JP 2014508784A5 JP 2014500216 A JP2014500216 A JP 2014500216A JP 2014500216 A JP2014500216 A JP 2014500216A JP 2014508784 A5 JP2014508784 A5 JP 2014508784A5
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JP
Japan
Prior art keywords
treatment
radiolabeled compound
cancer
radioactive imaging
breast cancer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2014500216A
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English (en)
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JP2014508784A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/CA2012/000316 external-priority patent/WO2012129673A1/en
Publication of JP2014508784A publication Critical patent/JP2014508784A/ja
Publication of JP2014508784A5 publication Critical patent/JP2014508784A5/ja
Withdrawn legal-status Critical Current

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Claims (1)

  1. 射性イメージングまたは乳癌または前立腺癌の治療のための、請求項45に記載の放
    射標識化合物。
JP2014500216A 2011-03-25 2012-03-26 17β−HSD1、17β−HSD3、および17β−HSD10の阻害剤 Withdrawn JP2014508784A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161467764P 2011-03-25 2011-03-25
US61/467,764 2011-03-25
PCT/CA2012/000316 WO2012129673A1 (en) 2011-03-25 2012-03-26 INHIBITORS OF 17ß-HSD1, 17ß-HSD3 AND 17ß-HSD10

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2017253315A Division JP6727184B2 (ja) 2011-03-25 2017-12-28 17β−HSD1、17β−HSD3、および17β−HSD10の阻害剤

Publications (2)

Publication Number Publication Date
JP2014508784A JP2014508784A (ja) 2014-04-10
JP2014508784A5 true JP2014508784A5 (ja) 2016-10-27

Family

ID=46929260

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2014500216A Withdrawn JP2014508784A (ja) 2011-03-25 2012-03-26 17β−HSD1、17β−HSD3、および17β−HSD10の阻害剤
JP2017253315A Active JP6727184B2 (ja) 2011-03-25 2017-12-28 17β−HSD1、17β−HSD3、および17β−HSD10の阻害剤

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2017253315A Active JP6727184B2 (ja) 2011-03-25 2017-12-28 17β−HSD1、17β−HSD3、および17β−HSD10の阻害剤

Country Status (6)

Country Link
US (1) US11072632B2 (ja)
EP (1) EP2688901B1 (ja)
JP (2) JP2014508784A (ja)
AU (1) AU2012234682A1 (ja)
CA (1) CA2830984C (ja)
WO (1) WO2012129673A1 (ja)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9850272B2 (en) 2013-06-25 2017-12-26 Forendo Pharma Ltd. Therapeutically active estratrienthiazole derivatives as inhibitors of 17.beta-hydroxy-steroid dehydrogenase, type 1
US10377791B2 (en) 2013-06-25 2019-08-13 Forendo Pharma Ltd. Therapeutically active estratrienthiazole derivatives as inhibitors of 17 B-hydroxysteroid dehydrogenase, type 1
WO2015169971A1 (en) * 2014-05-09 2015-11-12 Tangent Reprofiling Limited Modulators of androgen synthesis
JP6407415B2 (ja) * 2014-09-11 2018-10-17 バイエル・ファルマ・アクティエンゲゼルシャフト 3−窒素または硫黄置換エストラ−1,3,5(10),16−テトラエンakr1c3阻害剤
CZ307437B6 (cs) 2016-06-07 2018-08-22 Ăšstav organickĂ© chemie a biochemie AV ÄŚR, v.v.i. 15β-substituované deriváty estronu jako selektivní inhibitory 17β-hydroxysteoiddehydrogenáz
UA126342C2 (uk) 2017-06-08 2022-09-21 Форендо Фарма Лтд 15-бета-[3-пропанамідо]-заміщені естра-1,3,5(10)-трієн-17-он-сполуки і їх 17-оксими для використання в інгібуванні 17-бета-гідроксистероїддегідрогеназ
WO2024020520A2 (en) * 2022-07-20 2024-01-25 Board Of Regents, The University Of Texas System Enzyme compositions, steroid derivatives, enzyme inhibitors, and methods of making same for pharmaceutical applications

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5232917A (en) * 1987-08-25 1993-08-03 University Of Southern California Methods, compositions, and compounds for allosteric modulation of the GABA receptor by members of the androstane and pregnane series
EP0559240B1 (en) * 1987-09-24 2001-12-05 Jencap Research Limited Contraceptive packages containing oestrogen and progestin
TW385308B (en) * 1994-03-04 2000-03-21 Merck & Co Inc Prodrugs of morpholine tachykinin receptor antagonists
US5952319A (en) * 1997-11-26 1999-09-14 Research Triangle Institute Androgenic steroid compounds and a method of making and using the same
US6933312B2 (en) * 2002-10-07 2005-08-23 Agouron Pharmaceuticals, Inc. Pyrazole derivatives
TWI331154B (en) 2003-11-12 2010-10-01 Solvay Pharm Gmbh Novel 17-hydroxysteroid dehydrogenase type i inhibitors
CN102796160A (zh) 2005-05-26 2012-11-28 索尔瓦药物有限公司 17β-HSD1和STS抑制剂
US10174070B2 (en) * 2005-09-30 2019-01-08 Endece Llc 6-substituted estradiol derivatives and methods of use
AU2007299010B2 (en) * 2006-09-19 2013-01-31 Solvay Pharmaceuticals Gmbh Estratriene derivatives and their uses as 17beta-hydroxysteroid dehydrogenase inhibitors
RU2453554C2 (ru) 2006-11-30 2012-06-20 Зольвай Фармасьютиклз Гмбх Замещенные производные эстратриена как ингибиторы 17бета hsd
US20080171728A1 (en) 2007-01-12 2008-07-17 Quatrx Pharmaceuticals Co. Efficient Process for Preparing Steroids and Vitamin D Derivatives With the Unnatural Configuration at C20 (20 Alpha-Methyl) from Pregnenolone
EP2014672A1 (en) * 2007-07-12 2009-01-14 Bayer Schering Pharma Aktiengesellschaft 8-beta-substituted estratrienes as selectively active estrogens

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