JP2013520473A5 - - Google Patents

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Publication number
JP2013520473A5
JP2013520473A5 JP2012554348A JP2012554348A JP2013520473A5 JP 2013520473 A5 JP2013520473 A5 JP 2013520473A5 JP 2012554348 A JP2012554348 A JP 2012554348A JP 2012554348 A JP2012554348 A JP 2012554348A JP 2013520473 A5 JP2013520473 A5 JP 2013520473A5
Authority
JP
Japan
Prior art keywords
alkyl
group
methyl
substituted
thieno
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP2012554348A
Other languages
English (en)
Japanese (ja)
Other versions
JP2013520473A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2011/052811 external-priority patent/WO2011104338A1/en
Publication of JP2013520473A publication Critical patent/JP2013520473A/ja
Publication of JP2013520473A5 publication Critical patent/JP2013520473A5/ja
Ceased legal-status Critical Current

Links

JP2012554348A 2010-02-26 2011-02-25 医薬組成物用のＭｎｋ１／Ｍｎｋ２阻害活性を有するハロゲン又はシアノ置換されたチエノ［２，３−ｄ］ピリミジン Ceased JP2013520473A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP10154928 2010-02-26
EP10154928.5 2010-02-26
PCT/EP2011/052811 WO2011104338A1 (en) 2010-02-26 2011-02-25 Halogen or cyano substituted thieno [2,3-d]pyrimidines having mnk1/mnk2 inhibiting activity for pharmaceutical compositions

Publications (2)

Publication Number Publication Date
JP2013520473A JP2013520473A (ja) 2013-06-06
JP2013520473A5 true JP2013520473A5 (OSRAM) 2014-04-03

Family

ID=43907102

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012554348A Ceased JP2013520473A (ja) 2010-02-26 2011-02-25 医薬組成物用のＭｎｋ１／Ｍｎｋ２阻害活性を有するハロゲン又はシアノ置換されたチエノ［２，３−ｄ］ピリミジン

Country Status (4)

Country Link
US (1) US20130065914A1 (OSRAM)
EP (1) EP2539344B1 (OSRAM)
JP (1) JP2013520473A (OSRAM)
WO (1) WO2011104338A1 (OSRAM)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4518378B2 (ja) * 2001-10-29 2010-08-04 ベーリンガー インゲルハイム インテルナツィオナール ゲゼルシャフト ミット ベシュレンクテル ハフツング エネルギー恒常性および細胞小器官代謝の調節に関与するＭｎｋキナーゼ相同性タンパク質
EP2004656B1 (en) 2006-04-07 2013-07-10 Boehringer Ingelheim International GmbH Thienopyrimidines having mnk1 /mnk2 inhibiting activity for pharmaceutical compositions
EP1889847A1 (en) 2006-07-10 2008-02-20 DeveloGen Aktiengesellschaft Pyrrolopyrimidines for pharmaceutical compositions
AU2009286734A1 (en) 2008-08-26 2010-03-04 Boehringer Ingelheim International Gmbh Thienopyrimidines for pharmaceutical compositions
UY33245A (es) 2010-02-26 2011-09-30 Boehringer Ingelheim Int Tienopirimidinas que contienen un grupo alquilo sustituido para composiciones farmacéuticas
UY33241A (es) 2010-02-26 2011-09-30 Boehringer Ingelheim Int ?Tienopirimidinas que contienen heterocicloalquilo para composiciones farmacéuticas?.
US8754079B2 (en) * 2010-02-26 2014-06-17 Boehringer Ingelheim International Gmbh Cycloalkyl containing thienopyrimidines for pharmaceutical compositions
ES2754774T3 (es) * 2010-03-24 2020-04-20 Progastrine Et Cancers S A R L Profilaxis de cáncer colorrectal y gastrointestinal
CA2873967A1 (en) 2012-05-21 2013-11-28 Bayer Pharma Aktiengesellschaft Substituted benzothienopyrimidines
CA2873975A1 (en) 2012-05-21 2013-11-28 Bayer Pharma Aktiengesellschaft Thienopyrimidines
TW201412740A (zh) 2012-09-20 2014-04-01 Bayer Pharma AG 經取代之吡咯并嘧啶胺基苯并噻唑酮
US9556181B2 (en) 2013-02-01 2017-01-31 Bayer Pharma Aktiengesellschaft Substituted pyrazolopyrimidinylamino-indazoles
EP2951187A1 (en) 2013-02-01 2015-12-09 Bayer Pharma Aktiengesellschaft Substituted thienopyrimidines and pharmaceutical use thereof
US9675612B2 (en) 2013-03-06 2017-06-13 Bayer Pharma Aktiengesellschaft Substituted thiazolopyrimidines
CN109069865A (zh) * 2016-03-31 2018-12-21 南澳大利亚卫生与医学研究所有限公司 抑制高脂肪饮食相关病症的方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6643277B2 (en) 2000-06-29 2003-11-04 Harris Broadband Wireless Access, Inc. Frequency re-use for point to multipoint applications
SE0102147D0 (sv) 2001-06-18 2001-06-18 Pharmacia Ab New methods
JP4518378B2 (ja) 2001-10-29 2010-08-04 ベーリンガー インゲルハイム インテルナツィオナール ゲゼルシャフト ミット ベシュレンクテル ハフツング エネルギー恒常性および細胞小器官代謝の調節に関与するＭｎｋキナーゼ相同性タンパク質
US20050012622A1 (en) 2003-05-19 2005-01-20 Sutton William R. Monitoring and control of sleep cycles
EP1746099A1 (en) 2004-12-23 2007-01-24 DeveloGen Aktiengesellschaft Mnk1 or Mnk2 inhibitors
US20100143341A1 (en) * 2005-06-22 2010-06-10 Develogen Aktiengesellschaft Thienopyrimidines for pharmaceutical compositions
WO2007056215A2 (en) * 2005-11-02 2007-05-18 Cytovia, Inc. N-aryl-thienopyrimidin-4-amines and the use thereof
WO2007059905A2 (en) * 2005-11-25 2007-05-31 Develogen Aktiengesellschaft Thienopyrimidines treating inflammatory diseases
EP2004656B1 (en) 2006-04-07 2013-07-10 Boehringer Ingelheim International GmbH Thienopyrimidines having mnk1 /mnk2 inhibiting activity for pharmaceutical compositions
EP1889847A1 (en) 2006-07-10 2008-02-20 DeveloGen Aktiengesellschaft Pyrrolopyrimidines for pharmaceutical compositions
AU2009286734A1 (en) * 2008-08-26 2010-03-04 Boehringer Ingelheim International Gmbh Thienopyrimidines for pharmaceutical compositions

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