JP2013508413A - ｍＧｌｕＲ４アロステリック増強剤、組成物、および神経機能不全を治療する方法 - Google Patents

ｍＧｌｕＲ４アロステリック増強剤、組成物、および神経機能不全を治療する方法 Download PDF

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JP2013508413A
JP2013508413A JP2012535430A JP2012535430A JP2013508413A JP 2013508413 A JP2013508413 A JP 2013508413A JP 2012535430 A JP2012535430 A JP 2012535430A JP 2012535430 A JP2012535430 A JP 2012535430A JP 2013508413 A JP2013508413 A JP 2013508413A
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optionally substituted
cycloalkyl
alkyl
thiocarbonyl
carbonyl
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JP2013508413A5 (https=
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ジェフリー コン，ピー．
ダブリュ． リンズリー，クレイグ
アール． ホプキンス，コーリー
エム． ニスウェンダー，コリーン
ディー． ゴグリオッティ，ロッコ
エム． サロヴィッチ，ジェームス
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Vanderbilt University
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JP2012535430A 2009-10-22 2010-10-22 ｍＧｌｕＲ４アロステリック増強剤、組成物、および神経機能不全を治療する方法 Withdrawn JP2013508413A (ja)

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US25406209P 2009-10-22 2009-10-22
US61/254,062 2009-10-22
US29272510P 2010-01-06 2010-01-06
US61/292,725 2010-01-06
PCT/US2010/053837 WO2011050316A1 (en) 2009-10-22 2010-10-22 Mglur4 allosteric potentiators, compositions, and methods of treating neurological dysfunction

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JP2013508413A5 JP2013508413A5 (https=) 2013-12-05

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JP2012535428A Pending JP2013508412A (ja) 2009-10-22 2010-10-22 ｍＧｌｕＲ４アロステリック増強剤、組成物、および神経機能不全を治療する方法

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US (2) US9180192B2 (https=)
EP (2) EP2490529A4 (https=)
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KR (2) KR20120129869A (https=)
CN (2) CN102665411A (https=)
AU (2) AU2010310440A1 (https=)
BR (2) BR112012009574A2 (https=)
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AU2010208176A1 (en) 2009-01-28 2011-09-15 Vanderbilt University Substituted 1,1,3,3-tetraoxidobenzo[d][1,3,2]dithiazoles as mGluR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction
US8759377B2 (en) 2009-11-23 2014-06-24 Vanderbilt University Substituted dioxopiperidines and dioxopyrrolidines as MGLUR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction
JP6161537B2 (ja) 2010-04-07 2017-07-12 エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト ピラゾール−４−イル−ヘテロシクリル−カルボキサミド化合物及び使用の方法
EP2760857A1 (en) 2011-09-27 2014-08-06 F.Hoffmann-La Roche Ag Pyrazol-4-yl-heterocyclyl-carboxamide compounds and methods of use
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