JP2013500255A5 - - Google Patents

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Publication number
JP2013500255A5
JP2013500255A5 JP2012521755A JP2012521755A JP2013500255A5 JP 2013500255 A5 JP2013500255 A5 JP 2013500255A5 JP 2012521755 A JP2012521755 A JP 2012521755A JP 2012521755 A JP2012521755 A JP 2012521755A JP 2013500255 A5 JP2013500255 A5 JP 2013500255A5
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JP
Japan
Prior art keywords
lower alkyl
autophagy
cancer
cells
mbcq
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2012521755A
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English (en)
Japanese (ja)
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JP2013500255A (ja
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Publication date
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Priority claimed from PCT/US2010/042759 external-priority patent/WO2011011522A2/en
Publication of JP2013500255A publication Critical patent/JP2013500255A/ja
Publication of JP2013500255A5 publication Critical patent/JP2013500255A5/ja
Pending legal-status Critical Current

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JP2012521755A 2009-07-21 2010-07-21 自食作用の強力な小分子阻害剤、およびそれの使用方法 Pending JP2013500255A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US22716409P 2009-07-21 2009-07-21
US61/227,164 2009-07-21
US29673510P 2010-01-20 2010-01-20
US61/296,735 2010-01-20
PCT/US2010/042759 WO2011011522A2 (en) 2009-07-21 2010-07-21 Potent small molecule inhibitors of autophagy, and methods of use thereof

Publications (2)

Publication Number Publication Date
JP2013500255A JP2013500255A (ja) 2013-01-07
JP2013500255A5 true JP2013500255A5 (enExample) 2013-08-22

Family

ID=42829077

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012521755A Pending JP2013500255A (ja) 2009-07-21 2010-07-21 自食作用の強力な小分子阻害剤、およびそれの使用方法

Country Status (18)

Country Link
US (1) US20120258975A1 (enExample)
EP (1) EP2456761A2 (enExample)
JP (1) JP2013500255A (enExample)
KR (1) KR20120100886A (enExample)
CN (1) CN102574816A (enExample)
AU (1) AU2010276223A1 (enExample)
BR (1) BR112012001316A2 (enExample)
CA (1) CA2767772A1 (enExample)
CL (1) CL2012000163A1 (enExample)
IL (1) IL217502A0 (enExample)
IN (1) IN2012DN01478A (enExample)
MX (1) MX2012000940A (enExample)
PE (1) PE20120798A1 (enExample)
PH (1) PH12012500097A1 (enExample)
RU (1) RU2012105914A (enExample)
SG (1) SG177486A1 (enExample)
WO (1) WO2011011522A2 (enExample)
ZA (1) ZA201201224B (enExample)

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JP7633676B2 (ja) 2018-07-26 2025-02-20 ドメイン・セラピューティクス 置換キナゾリノン誘導体、及びmGluR4のポジティブアロステリック調節剤としてのその使用
CN109721554A (zh) * 2019-01-08 2019-05-07 贵州大学 一类4-氨基喹唑啉类化合物及其制备方法和应用
IL287795B2 (en) 2019-05-10 2025-05-01 Deciphera Pharmaceuticals Llc Heteroarylaminopyrimidine amides as autophagy inhibitors and methods of using them
CN118878519A (zh) 2019-05-10 2024-11-01 德西费拉制药有限责任公司 苯基氨基嘧啶酰胺自噬抑制剂及其使用方法
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JP2024504587A (ja) * 2021-01-14 2024-02-01 ジョージタウン ユニバーシティ Usp13阻害剤及びその使用方法
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