JP2012530113A5 - - Google Patents
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- Publication number
- JP2012530113A5 JP2012530113A5 JP2012515500A JP2012515500A JP2012530113A5 JP 2012530113 A5 JP2012530113 A5 JP 2012530113A5 JP 2012515500 A JP2012515500 A JP 2012515500A JP 2012515500 A JP2012515500 A JP 2012515500A JP 2012530113 A5 JP2012530113 A5 JP 2012530113A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- formula
- branched
- linear
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP09305562A EP2270021A1 (en) | 2009-06-18 | 2009-06-18 | Phosphonates synthons for the synthesis of phosphonates derivatives showing better bioavailability |
| EP09305562.2 | 2009-06-18 | ||
| PCT/EP2010/058567 WO2010146127A1 (en) | 2009-06-18 | 2010-06-17 | Phosphonates synthons for the synthesis of phosphonates derivatives showing better bioavailability |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2012530113A JP2012530113A (ja) | 2012-11-29 |
| JP2012530113A5 true JP2012530113A5 (https=) | 2013-08-01 |
Family
ID=41171101
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012515500A Pending JP2012530113A (ja) | 2009-06-18 | 2010-06-17 | より良好な生物学的利用能を示すホスホネート誘導体の合成のためのホスホネートシントン |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US8785629B2 (https=) |
| EP (2) | EP2270021A1 (https=) |
| JP (1) | JP2012530113A (https=) |
| CA (1) | CA2764827C (https=) |
| ES (1) | ES2601849T3 (https=) |
| WO (1) | WO2010146127A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012034719A1 (en) * | 2010-09-14 | 2012-03-22 | Centre National De La Recherche Scientifique | Novel antiviral acyclic nucleoside phosphonates |
| EP4116310A4 (en) * | 2020-03-04 | 2024-07-17 | FUJIFILM Wako Pure Chemical Corporation | PROCESS FOR PRODUCING PHOSPHONE ACID ESTERS AND PROCESS FOR PRODUCING PHOSPHATE ESTERS |
| EP4370136A4 (en) * | 2021-07-15 | 2025-10-29 | Alnylam Pharmaceuticals Inc | SIMPLE CHEMICAL APPROACHES TO INTRODUCE 2,6-DIAMINOPURINE AND 2-AMINOADENINE CONJUGATES INTO OLIGONUCLEOTIDES |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL6814978A (https=) | 1967-10-30 | 1969-05-02 | ||
| BR6914868D0 (pt) * | 1969-01-23 | 1973-03-20 | & Co Inc Merck | Processos quimicos |
| JPS6069089A (ja) | 1983-09-26 | 1985-04-19 | Nissan Chem Ind Ltd | ジヒドロピリジン−５−ホスホネ−ト誘導体およびその製造法 |
| EP0533833B1 (en) * | 1990-06-13 | 1995-12-20 | GLAZIER, Arnold | Phosphorous produgs |
| EP0521622B1 (en) | 1991-07-03 | 1997-08-13 | PHARMACIA & UPJOHN COMPANY | Pyrazolopyrimidine and pyrimidinyl bisphosphonic esters as anti-inflammatories |
| ZA941088B (en) * | 1993-02-19 | 1995-09-27 | Symphar Sa | Substituted ketophosphonates the processes for their preparation and pharmaceutical compositions containing them |
| DE4343599A1 (de) | 1993-12-21 | 1995-06-22 | Bayer Ag | Verwendung von Phosphonsäureestern zur Behandlung von Hirnleistungsstörungen und Depressionen |
| US5635449A (en) * | 1995-04-07 | 1997-06-03 | American Cyanamid Company | Arylthioalkyl- and arylthioalkenylphosphonic acids and derivatives thereof useful as herbicidal agents |
| IT1281498B1 (it) * | 1995-06-07 | 1998-02-18 | Sardinian Antiviral Research C | Pirazolo - derivati ad attivita' antitumorale, processo per la loro preparazione e composizioni farmaceutiche che li contengono , e |
| NZ330216A (en) * | 1996-01-16 | 2000-09-29 | Bristol Myers Squibb Co | Conformationally restricted aromatic inhibitors of microsomal triglyceride transfer protein and use in treatment of atherosclerosis |
| IT1290444B1 (it) | 1997-03-27 | 1998-12-03 | Boehringer Mannheim Italia | Coniugati di bis-fosfonati con funzionalita' alchilanti aventi attivita' antitumorale |
| CA2747954C (en) * | 1999-12-03 | 2014-02-25 | The Regents Of The University Of California | Phosphonate compounds |
| WO2003091264A2 (en) | 2002-04-26 | 2003-11-06 | Gilead Sciences, Inc. | Non nucleoside reverse transcriptase inhibitors |
| WO2004026315A1 (en) | 2002-09-19 | 2004-04-01 | Ilex Oncology Research, Sarl | Substituted ketophosphonate compounds having bone anabolic activity |
| WO2004035577A2 (en) * | 2002-10-16 | 2004-04-29 | Gilead Sciences, Inc. | Pre-organized tricyclic integrase inhibitor compounds |
| JP2010535701A (ja) * | 2003-04-25 | 2010-11-25 | ギリアード サイエンシーズ， インコーポレイテッド | 抗癌ホスホネートアナログ |
| CN1882327A (zh) | 2003-11-19 | 2006-12-20 | 症变治疗公司 | 含磷的新的拟甲状腺素药 |
| US20080261923A1 (en) * | 2004-08-04 | 2008-10-23 | Etzkorn Felicia A | Alkene Mimics |
| WO2008096002A1 (en) | 2007-02-08 | 2008-08-14 | Tibotec Pharmaceuticals Ltd. | Hcv inhibiting macrocyclic phosphonates and amidophosphates |
-
2009
- 2009-06-18 EP EP09305562A patent/EP2270021A1/en not_active Withdrawn
-
2010
- 2010-06-17 US US13/377,652 patent/US8785629B2/en not_active Expired - Fee Related
- 2010-06-17 WO PCT/EP2010/058567 patent/WO2010146127A1/en not_active Ceased
- 2010-06-17 JP JP2012515500A patent/JP2012530113A/ja active Pending
- 2010-06-17 EP EP10725716.4A patent/EP2443130B1/en not_active Not-in-force
- 2010-06-17 ES ES10725716.4T patent/ES2601849T3/es active Active
- 2010-06-17 CA CA2764827A patent/CA2764827C/en not_active Expired - Fee Related
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