JP2012526854A5 - - Google Patents
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- Publication number
- JP2012526854A5 JP2012526854A5 JP2012511068A JP2012511068A JP2012526854A5 JP 2012526854 A5 JP2012526854 A5 JP 2012526854A5 JP 2012511068 A JP2012511068 A JP 2012511068A JP 2012511068 A JP2012511068 A JP 2012511068A JP 2012526854 A5 JP2012526854 A5 JP 2012526854A5
- Authority
- JP
- Japan
- Prior art keywords
- dispensing device
- pharmaceutical composition
- analgesic pharmaceutical
- dexmedetomidine
- pharmaceutically acceptable
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 230000000202 analgesic effect Effects 0.000 claims 8
- 239000008194 pharmaceutical composition Substances 0.000 claims 8
- 229960004253 dexmedetomidine Drugs 0.000 claims 4
- HRLIOXLXPOHXTA-NSHDSACASA-N dexmedetomidine Chemical compound C1([C@@H](C)C=2C(=C(C)C=CC=2)C)=CN=C[N]1 HRLIOXLXPOHXTA-NSHDSACASA-N 0.000 claims 4
- 210000000214 mouth Anatomy 0.000 claims 3
- 150000003839 salts Chemical class 0.000 claims 3
- 206010039897 Sedation Diseases 0.000 claims 1
- 229960002746 dexmedetomidine hydrochloride Drugs 0.000 claims 1
- VPNGEIHDPSLNMU-MERQFXBCSA-N dexmedetomidine hydrochloride Chemical group Cl.C1([C@@H](C)C=2C(=C(C)C=CC=2)C)=CNC=N1 VPNGEIHDPSLNMU-MERQFXBCSA-N 0.000 claims 1
- 210000004877 mucosa Anatomy 0.000 claims 1
- 239000008203 oral pharmaceutical composition Substances 0.000 claims 1
- 230000036280 sedation Effects 0.000 claims 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US17873009P | 2009-05-15 | 2009-05-15 | |
| US61/178,730 | 2009-05-15 | ||
| PCT/US2010/035136 WO2010132882A2 (en) | 2009-05-15 | 2010-05-17 | Sublingual dexmedetomidine compositions and methods of use thereof |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015179975A Division JP2016029055A (ja) | 2009-05-15 | 2015-09-11 | デクスメデトミジンの舌下組成物およびその使用方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2012526854A JP2012526854A (ja) | 2012-11-01 |
| JP2012526854A5 true JP2012526854A5 (enExample) | 2013-07-04 |
| JP6172938B2 JP6172938B2 (ja) | 2017-08-02 |
Family
ID=43085620
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012511068A Expired - Fee Related JP6172938B2 (ja) | 2009-05-15 | 2010-05-17 | デクスメデトミジンの舌下組成物およびその使用方法 |
| JP2015179975A Pending JP2016029055A (ja) | 2009-05-15 | 2015-09-11 | デクスメデトミジンの舌下組成物およびその使用方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015179975A Pending JP2016029055A (ja) | 2009-05-15 | 2015-09-11 | デクスメデトミジンの舌下組成物およびその使用方法 |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US20110021588A1 (enExample) |
| EP (2) | EP2429521B1 (enExample) |
| JP (2) | JP6172938B2 (enExample) |
| KR (1) | KR101859486B1 (enExample) |
| CN (2) | CN102639131A (enExample) |
| AU (1) | AU2010248776B2 (enExample) |
| BR (1) | BRPI1010567A2 (enExample) |
| CA (1) | CA2762107A1 (enExample) |
| CL (1) | CL2011002858A1 (enExample) |
| CO (1) | CO6460767A2 (enExample) |
| CR (1) | CR20110596A (enExample) |
| DO (1) | DOP2011000354A (enExample) |
| EC (1) | ECSP11011459A (enExample) |
| HN (1) | HN2011003011A (enExample) |
| IL (1) | IL216159A (enExample) |
| MX (1) | MX2011011950A (enExample) |
| NZ (1) | NZ596976A (enExample) |
| PE (1) | PE20120713A1 (enExample) |
| RU (1) | RU2572692C2 (enExample) |
| SG (1) | SG175979A1 (enExample) |
| WO (1) | WO2010132882A2 (enExample) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20130096170A1 (en) | 2011-10-14 | 2013-04-18 | Hospira, Inc. | Methods of treating pediatric patients using dexmedetomidine |
| CN104470516A (zh) * | 2011-12-11 | 2015-03-25 | 瑞克欧制药有限公司 | 鼻内右美托咪定组合物和其使用方法 |
| US8242158B1 (en) | 2012-01-04 | 2012-08-14 | Hospira, Inc. | Dexmedetomidine premix formulation |
| CA2865593A1 (en) * | 2012-02-27 | 2013-09-06 | Eye Therapies Llc | Compositions and methods for the treatment of migraine |
| NZ706990A (en) * | 2012-10-15 | 2017-12-22 | Orion Corp | A veterinary method of alleviating noise aversion |
| EP2792352A1 (en) * | 2013-04-16 | 2014-10-22 | Laboratorios Del. Dr. Esteve, S.A. | Alpha-2 adrenoreceptor and sigma receptor ligand combinations |
| US20150273215A1 (en) * | 2014-03-26 | 2015-10-01 | Pacesetter, Inc. | Systems and methods for assessment of pain and other parameters during trial neurostimulation |
| TWI704933B (zh) * | 2013-10-07 | 2020-09-21 | 美商帝國製藥美國股份有限公司 | 右美托咪啶經皮輸送裝置及使用其之方法 |
| TWI709417B (zh) | 2013-10-07 | 2020-11-11 | 美商帝國製藥美國股份有限公司 | 使用右美托咪啶經皮組成物用於治療注意力不足過動症、焦慮及失眠的方法及組成物 |
| CN105764496B (zh) | 2013-10-07 | 2020-09-25 | 帝国制药美国公司 | 用于经皮递送非镇静量的右旋美托咪啶的方法和组合物 |
| RU2557882C1 (ru) * | 2014-07-08 | 2015-07-27 | Государственное бюджетное образовательное учреждение высшего профессионального образования "Астраханская государственная медицинская академия" Министерства здравоохранения Российской Федерации (ГБОУ ВПО АГМА Минздрава России) | Способ проведения премедикации при плановом хирургическом лечении |
| MA41689A (fr) * | 2014-10-15 | 2017-08-22 | Bioxcel Corp | Prévention ou traitement de troubles du sommeil au moyen d'une formulation de dexmédétomidine |
| ES2879298T3 (es) * | 2016-12-13 | 2021-11-22 | Orion Corp | Dexmedetomidina o medetomidina para su uso en el tratamiento de la ansiedad por separación en perro |
| CA3045043A1 (en) * | 2016-12-31 | 2018-07-05 | Bioxcel Therapeutics, Inc. | Use of sublingual dexmedetomidine for the treatment of agitation |
| CN115154440A (zh) | 2018-06-27 | 2022-10-11 | 比奥克斯塞尔医疗股份有限公司 | 含右美托咪定的膜制剂及其制造方法 |
| WO2020176807A1 (en) | 2019-02-27 | 2020-09-03 | Vanderbilt University | Methods of treating trigeminal nerve pain |
| CN116474218A (zh) * | 2019-06-28 | 2023-07-25 | 四川普锐特药业有限公司 | 保持给药均一度的药物流体分配器及右美托咪定鼻喷器 |
| WO2021016112A2 (en) | 2019-07-19 | 2021-01-28 | Bioxcel Therapeutics, Inc. | Non-sedating dexmedetomidine treatment regimens |
| CN113827590A (zh) * | 2020-06-08 | 2021-12-24 | 四川普锐特药业有限公司 | 右美托咪定在助眠药物制备中的应用 |
| US20220031664A1 (en) * | 2020-07-28 | 2022-02-03 | Melt Pharmaceuticals, Inc. | Pharmaceutical compositions comprising antiemetics and alpha-2-adrenergic receptor agonists and methods of using the same for anesthesiological applications |
| EP4583871A1 (en) * | 2022-09-11 | 2025-07-16 | BioXcel Therapeutics, Inc. | Methods for treating agitation in community settings |
| US11806334B1 (en) | 2023-01-12 | 2023-11-07 | Bioxcel Therapeutics, Inc. | Non-sedating dexmedetomidine treatment regimens |
| CN118542852B (zh) * | 2024-07-30 | 2024-10-01 | 山东则正医药技术有限公司 | 包含经口给药的右美托咪定舌下膜组合物及其制备方法和应用 |
Family Cites Families (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2206880B (en) * | 1987-07-16 | 1991-04-24 | Farmos Oy | Optical isomers of an imidazole derivative |
| US5124157A (en) * | 1989-08-18 | 1992-06-23 | Cygnus Therapeutic Systems | Method and device for administering dexmedetomidine transdermally |
| US5217718A (en) * | 1989-08-18 | 1993-06-08 | Cygnus Therapeutic Systems | Method and device for administering dexmedetomidine transdermally |
| FI894911A0 (fi) * | 1989-10-17 | 1989-10-17 | Farmos Oy | En terapeutiskt vaerdefull foerening. |
| DE122007000103I1 (de) * | 1990-12-05 | 2008-04-03 | Gen Hospital Corp | Verwendung von NO zur Behandlung der persistenten pulmonalen Hypertonie des Neugeborenen |
| GB9111732D0 (en) * | 1991-05-31 | 1991-07-24 | Orion Yhtymae Oy | The use of certain salts of medetomidine and its optically active enantiomers to regulate the rate of transdermal administration of the drugs |
| US5571840A (en) * | 1993-06-22 | 1996-11-05 | The Regents Of The University Of Michigan | Method for treating central nervous system ischemia |
| US5713907A (en) * | 1995-07-20 | 1998-02-03 | Endotex Interventional Systems, Inc. | Apparatus and method for dilating a lumen and for inserting an intraluminal graft |
| GB9520150D0 (en) | 1995-10-03 | 1995-12-06 | Orion Yhtymae Oy | New imidazole derivatives |
| US20050281752A1 (en) * | 1997-10-01 | 2005-12-22 | Dugger Harry A Iii | Buccal, polar and non-polar spray or capsule containing drugs for treating disorders of the central nervous system |
| US20030077227A1 (en) * | 1997-10-01 | 2003-04-24 | Dugger Harry A. | Buccal, polar and non-polar spray or capsule containing drugs for treating disorders of the central nervous system |
| US6716867B1 (en) | 1998-04-01 | 2004-04-06 | Orion Corporation | Use of dexmedetomidine for ICU sedation |
| AR015744A1 (es) * | 1998-04-01 | 2001-05-16 | Orion Corp | Uso de dexmedetomidina para sedacion en terapia intensiva |
| US7001609B1 (en) * | 1998-10-02 | 2006-02-21 | Regents Of The University Of Minnesota | Mucosal originated drug delivery systems and animal applications |
| CN1321086A (zh) * | 1998-10-02 | 2001-11-07 | 3M创新有限公司 | 粘膜型药物送递系统及其动物运用 |
| GB9913677D0 (en) * | 1999-06-11 | 1999-08-11 | Imperial College | Formulation |
| AUPR184500A0 (en) * | 2000-12-01 | 2001-01-04 | Drug Delivery Solutions Pty Ltd | Dispensing device |
| US20030022926A1 (en) * | 2001-05-07 | 2003-01-30 | Lavand'homme Patricia | Method for treating neuropathic pain and pharmaceutical preparation therefor |
| WO2002094238A1 (en) * | 2001-05-24 | 2002-11-28 | Alexza Molecular Delivery Corporation | Delivery of anti-migraine compounds through an inhalation route |
| FR2834212B1 (fr) * | 2001-12-27 | 2004-07-09 | Besins Int Belgique | Utilisation d'une poudre a liberation immediate dans des compositions pharmaceutiques et nutraceutiques |
| IL147921A0 (en) * | 2002-01-31 | 2002-08-14 | Abdulrazik Mohammad | A method for treating central nervous system disorders by ocular dosing |
| US7439241B2 (en) * | 2003-05-27 | 2008-10-21 | Galderma Laboratories, Inc. | Compounds, formulations, and methods for treating or preventing rosacea |
| US20090117054A1 (en) * | 2005-03-29 | 2009-05-07 | University Of Kentucky Research Foundation | Sublingual spray for the treatment of pain |
| MX374396B (es) * | 2006-01-25 | 2025-03-06 | Insys Therapeutics Inc | Rocio de fentanilo sublingual. |
| EP1986642B1 (en) * | 2006-02-13 | 2013-11-13 | Orient Pharma (Samoa) Co, Ltd | Combination of alpha-2 receptor agonist (clonidine) and an anti-muscarinic agent (oxybutynin) for the treatment of sialorrhoea |
| WO2008003093A2 (en) * | 2006-06-29 | 2008-01-03 | Questcor Pharmaceuticals, Inc. | Pharmaceutical compositions and related methods of treatment |
| CN101057830A (zh) * | 2007-05-10 | 2007-10-24 | 北京天川军威医药技术开发有限公司 | 盐酸纳洛酮舌下喷雾给药系统或组合物及其制备方法 |
-
2010
- 2010-05-17 EP EP10775671.0A patent/EP2429521B1/en active Active
- 2010-05-17 SG SG2011082666A patent/SG175979A1/en unknown
- 2010-05-17 CN CN2010800211820A patent/CN102639131A/zh active Pending
- 2010-05-17 CN CN201610753813.7A patent/CN106511273A/zh active Pending
- 2010-05-17 BR BRPI1010567A patent/BRPI1010567A2/pt not_active IP Right Cessation
- 2010-05-17 NZ NZ596976A patent/NZ596976A/en not_active IP Right Cessation
- 2010-05-17 PE PE2011001958A patent/PE20120713A1/es not_active Application Discontinuation
- 2010-05-17 AU AU2010248776A patent/AU2010248776B2/en not_active Ceased
- 2010-05-17 MX MX2011011950A patent/MX2011011950A/es active IP Right Grant
- 2010-05-17 RU RU2011151059/15A patent/RU2572692C2/ru active
- 2010-05-17 EP EP17187813.5A patent/EP3305281A1/en not_active Withdrawn
- 2010-05-17 WO PCT/US2010/035136 patent/WO2010132882A2/en not_active Ceased
- 2010-05-17 KR KR1020117027466A patent/KR101859486B1/ko not_active Expired - Fee Related
- 2010-05-17 CA CA2762107A patent/CA2762107A1/en not_active Abandoned
- 2010-05-17 US US12/781,628 patent/US20110021588A1/en not_active Abandoned
- 2010-05-17 JP JP2012511068A patent/JP6172938B2/ja not_active Expired - Fee Related
-
2011
- 2011-11-06 IL IL216159A patent/IL216159A/en active IP Right Grant
- 2011-11-14 EC EC2011011459A patent/ECSP11011459A/es unknown
- 2011-11-14 HN HN2011003011A patent/HN2011003011A/es unknown
- 2011-11-14 CL CL2011002858A patent/CL2011002858A1/es unknown
- 2011-11-14 DO DO2011000354A patent/DOP2011000354A/es unknown
- 2011-11-14 CR CR20110596A patent/CR20110596A/es unknown
- 2011-11-15 CO CO11155150A patent/CO6460767A2/es active IP Right Grant
-
2015
- 2015-09-11 JP JP2015179975A patent/JP2016029055A/ja active Pending
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