MX2011011950A - Composiciones de dexmedetomidina sublinguales y metodos de uso de las mismas. - Google Patents

Composiciones de dexmedetomidina sublinguales y metodos de uso de las mismas.

Info

Publication number
MX2011011950A
MX2011011950A MX2011011950A MX2011011950A MX2011011950A MX 2011011950 A MX2011011950 A MX 2011011950A MX 2011011950 A MX2011011950 A MX 2011011950A MX 2011011950 A MX2011011950 A MX 2011011950A MX 2011011950 A MX2011011950 A MX 2011011950A
Authority
MX
Mexico
Prior art keywords
methods
dexmedetomidine compositions
sublingual
sublingual dexmedetomidine
compositions
Prior art date
Application number
MX2011011950A
Other languages
English (en)
Inventor
Geraldine Anne Henwood
Christopher Thomas Sharr
John Joseph Koleng Jr
Randall Jerome Mack
Original Assignee
Recro Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43085620&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2011011950(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Recro Pharma Inc filed Critical Recro Pharma Inc
Publication of MX2011011950A publication Critical patent/MX2011011950A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4174—Arylalkylimidazoles, e.g. oxymetazolin, naphazoline, miconazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/12—Aerosols; Foams
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61M—DEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
    • A61M31/00—Devices for introducing or retaining media, e.g. remedies, in cavities of the body
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00—Preparations for use in therapy
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61M—DEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
    • A61M2210/00—Anatomical parts of the body
    • A61M2210/06—Head
    • A61M2210/0625—Mouth

Abstract

La presente invención se relaciona con formulaciones sublinguales analgésicas de dexmedetomidina y con métodos de uso de las mismas, para el uso en la prevención, tratamiento y manejo del dolor y otras afecciones.
MX2011011950A 2009-05-15 2010-05-17 Composiciones de dexmedetomidina sublinguales y metodos de uso de las mismas. MX2011011950A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17873009P 2009-05-15 2009-05-15
PCT/US2010/035136 WO2010132882A2 (en) 2009-05-15 2010-05-17 Sublingual dexmedetomidine compositions and methods of use thereof

Publications (1)

Publication Number Publication Date
MX2011011950A true MX2011011950A (es) 2012-02-21

Family

ID=43085620

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2011011950A MX2011011950A (es) 2009-05-15 2010-05-17 Composiciones de dexmedetomidina sublinguales y metodos de uso de las mismas.

Country Status (21)

Country Link
US (1) US20110021588A1 (es)
EP (2) EP2429521B1 (es)
JP (2) JP6172938B2 (es)
KR (1) KR101859486B1 (es)
CN (2) CN106511273A (es)
AU (1) AU2010248776B2 (es)
BR (1) BRPI1010567A2 (es)
CA (1) CA2762107A1 (es)
CL (1) CL2011002858A1 (es)
CO (1) CO6460767A2 (es)
CR (1) CR20110596A (es)
DO (1) DOP2011000354A (es)
EC (1) ECSP11011459A (es)
HN (1) HN2011003011A (es)
IL (1) IL216159A (es)
MX (1) MX2011011950A (es)
NZ (1) NZ596976A (es)
PE (1) PE20120713A1 (es)
RU (1) RU2572692C2 (es)
SG (1) SG175979A1 (es)
WO (1) WO2010132882A2 (es)

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US20130096170A1 (en) 2011-10-14 2013-04-18 Hospira, Inc. Methods of treating pediatric patients using dexmedetomidine
WO2013090278A2 (en) 2011-12-11 2013-06-20 Recro Pharma, Inc. Intranasal dexmedetomidine compositions and methods of use thereof
US8242158B1 (en) 2012-01-04 2012-08-14 Hospira, Inc. Dexmedetomidine premix formulation
WO2013130577A2 (en) * 2012-02-27 2013-09-06 Eye Therapies, Llc Compositions and methods for the treatment of migraine
US10780079B2 (en) * 2012-10-15 2020-09-22 Orion Corporation Veterinary method of alleviating noise aversion
EP2792352A1 (en) * 2013-04-16 2014-10-22 Laboratorios Del. Dr. Esteve, S.A. Alpha-2 adrenoreceptor and sigma receptor ligand combinations
US20150273215A1 (en) * 2014-03-26 2015-10-01 Pacesetter, Inc. Systems and methods for assessment of pain and other parameters during trial neurostimulation
CA2924236C (en) 2013-10-07 2020-01-07 Teikoku Pharma Usa, Inc. Methods and compositions for transdermal delivery of a non-sedative amount of dexmedetomidine
RU2018105761A (ru) 2013-10-07 2019-02-26 ТЕЙКОКУ ФАРМА ЮЭсЭй, ИНК. Устройства для трансдермальной доставки дексмедетомидина и способы их применения
EP3054935B1 (en) 2013-10-07 2020-12-09 Teikoku Pharma USA, Inc. Methods and compositions for treating attention deficit hyperactivity disorder, anxiety and insomnia using dexmedetomidine transdermal compositions
RU2557882C1 (ru) * 2014-07-08 2015-07-27 Государственное бюджетное образовательное учреждение высшего профессионального образования "Астраханская государственная медицинская академия" Министерства здравоохранения Российской Федерации (ГБОУ ВПО АГМА Минздрава России) Способ проведения премедикации при плановом хирургическом лечении
MA41689A (fr) * 2014-10-15 2017-08-22 Bioxcel Corp Prévention ou traitement de troubles du sommeil au moyen d'une formulation de dexmédétomidine
US20200069650A1 (en) * 2016-12-13 2020-03-05 Orion Corporation Dexmedetomidine or medetomidine for use in treating separation anxiety in dogs
CA3045043A1 (en) * 2016-12-31 2018-07-05 Bioxcel Therapeutics, Inc. Use of sublingual dexmedetomidine for the treatment of agitation
US10792246B2 (en) * 2018-06-27 2020-10-06 Bioxcel Therapeutics, Inc. Film formulations containing dexmedetomidine and methods of producing them
CN112138250B (zh) * 2019-06-28 2023-04-14 四川普锐特药业有限公司 保持给药均一度的药物流体分配器及右美托咪定鼻喷器
KR20220049526A (ko) 2019-07-19 2022-04-21 바이오엑셀 테라퓨틱스 인코포레이티드 비-진정성 덱스메데토미딘 치료 양생법
CN113827590A (zh) * 2020-06-08 2021-12-24 四川普锐特药业有限公司 右美托咪定在助眠药物制备中的应用
US20220031664A1 (en) * 2020-07-28 2022-02-03 Melt Pharmaceuticals, Inc. Pharmaceutical compositions comprising antiemetics and alpha-2-adrenergic receptor agonists and methods of using the same for anesthesiological applications
WO2024055042A1 (en) * 2022-09-11 2024-03-14 Bioxcel Therapeutics, Inc. Methods for treating agitation in community settings
US11806334B1 (en) 2023-01-12 2023-11-07 Bioxcel Therapeutics, Inc. Non-sedating dexmedetomidine treatment regimens

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Also Published As

Publication number Publication date
CA2762107A1 (en) 2010-11-18
NZ596976A (en) 2014-05-30
AU2010248776A1 (en) 2012-01-12
ECSP11011459A (es) 2012-01-31
EP2429521A4 (en) 2013-08-21
HN2011003011A (es) 2014-12-01
CL2011002858A1 (es) 2012-06-22
JP6172938B2 (ja) 2017-08-02
AU2010248776B2 (en) 2013-06-06
WO2010132882A2 (en) 2010-11-18
PE20120713A1 (es) 2012-07-08
WO2010132882A8 (en) 2011-12-29
US20110021588A1 (en) 2011-01-27
WO2010132882A3 (en) 2011-03-31
KR101859486B1 (ko) 2018-06-28
CN102639131A (zh) 2012-08-15
EP2429521B1 (en) 2017-10-18
KR20120008058A (ko) 2012-01-25
JP2012526854A (ja) 2012-11-01
EP2429521A2 (en) 2012-03-21
RU2011151059A (ru) 2013-06-20
SG175979A1 (en) 2011-12-29
EP3305281A1 (en) 2018-04-11
IL216159A0 (en) 2012-01-31
BRPI1010567A2 (pt) 2016-03-15
RU2572692C2 (ru) 2016-01-20
CR20110596A (es) 2012-03-26
CN106511273A (zh) 2017-03-22
JP2016029055A (ja) 2016-03-03
DOP2011000354A (es) 2012-07-15
CO6460767A2 (es) 2012-06-15
IL216159A (en) 2015-10-29

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