JP2012502978A5 - - Google Patents

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Publication number
JP2012502978A5
JP2012502978A5 JP2011527463A JP2011527463A JP2012502978A5 JP 2012502978 A5 JP2012502978 A5 JP 2012502978A5 JP 2011527463 A JP2011527463 A JP 2011527463A JP 2011527463 A JP2011527463 A JP 2011527463A JP 2012502978 A5 JP2012502978 A5 JP 2012502978A5
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JP
Japan
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alkyl
alkenyl
aryl
heteroaryl
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JP2011527463A
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English (en)
Japanese (ja)
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JP5666454B2 (ja
JP2012502978A (ja
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Priority claimed from EP08164847A external-priority patent/EP2166008A1/en
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Publication of JP2012502978A5 publication Critical patent/JP2012502978A5/ja
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Publication of JP5666454B2 publication Critical patent/JP5666454B2/ja
Expired - Fee Related legal-status Critical Current
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JP2011527463A 2008-09-23 2009-09-22 Nadphオキシダーゼインヒビターとしてのピラゾロピリジン誘導体 Expired - Fee Related JP5666454B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP08164847A EP2166008A1 (en) 2008-09-23 2008-09-23 Pyrazolo pyridine derivatives as NADPH oxidase inhibitors
EP08164847.9 2008-09-23
PCT/IB2009/054148 WO2010035217A1 (en) 2008-09-23 2009-09-22 Pyrazolo pyridine derivatives as nadph oxidase inhibitors

Publications (3)

Publication Number Publication Date
JP2012502978A JP2012502978A (ja) 2012-02-02
JP2012502978A5 true JP2012502978A5 (enExample) 2012-11-08
JP5666454B2 JP5666454B2 (ja) 2015-02-12

Family

ID=40325411

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011527463A Expired - Fee Related JP5666454B2 (ja) 2008-09-23 2009-09-22 Nadphオキシダーゼインヒビターとしてのピラゾロピリジン誘導体

Country Status (12)

Country Link
US (2) US8481562B2 (enExample)
EP (2) EP2166008A1 (enExample)
JP (1) JP5666454B2 (enExample)
KR (1) KR101703360B1 (enExample)
CN (1) CN102137863B (enExample)
AU (1) AU2009298004B2 (enExample)
BR (1) BRPI0919329A2 (enExample)
CA (1) CA2737457C (enExample)
ES (1) ES2565436T3 (enExample)
IL (1) IL211889A (enExample)
RU (1) RU2569303C2 (enExample)
WO (1) WO2010035217A1 (enExample)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2002835A1 (en) 2007-06-04 2008-12-17 GenKyo Tex Pyrazolo pyridine derivatives as NADPH oxidase inhibitors
EP2000176A1 (en) 2007-06-04 2008-12-10 GenKyo Tex Tetrahydroindole derivatives as NADPH Oxidase inhibitors
EP2165707A1 (en) 2008-09-23 2010-03-24 Genkyo Tex Sa Pyrazolo pyridine derivatives as NADPH oxidase inhibitors
EP2166009A1 (en) 2008-09-23 2010-03-24 Genkyo Tex Sa Pyrazolo pyridine derivatives as nadph oxidase inhibitors
EP2166010A1 (en) 2008-09-23 2010-03-24 Genkyo Tex Sa Pyrazolo pyridine derivatives as NADPH oxidase inhibitors
EP2305679A1 (en) 2009-09-28 2011-04-06 GenKyoTex SA Pyrazoline dione derivatives as nadph oxidase inhibitors
EP2361911A1 (en) 2010-02-18 2011-08-31 GenKyoTex SA Pyrazolo piperidine derivatives as NADPH oxidase inhibitors
CN104918616A (zh) 2012-10-24 2015-09-16 格卢科克斯生物科技有限公司 用于治疗与烟酰胺腺嘌呤二核苷酸磷酸氧化酶相关的病况的三嗪衍生物
US20140212891A1 (en) 2013-01-29 2014-07-31 Amina El Jamali Compositions and Methods Using NOX5
EP2857399A1 (en) * 2013-10-03 2015-04-08 GenKyoTex SA Compounds useful for the treatment of PDE5 inhibitor-poorly responsive erectile dysfunction
JP6783224B2 (ja) 2014-04-04 2020-11-11 デル マー ファーマシューティカルズ 肺の非小細胞癌腫及び卵巣癌を処置するためのジアンヒドロガラクチトール及びその類縁体又は誘導体の使用
JP2018505226A (ja) 2015-02-16 2018-02-22 グルコックス・バイオテック・アーベー N2−(3,4−ジメチルフェニル)−6−((4−(p−トリル)ピペラジン−1−イル)メチル)−1,3,5−トリアジン−2,4−ジアミン
US20180072718A1 (en) 2016-09-09 2018-03-15 Incyte Corporation Pyrazolopyridine compounds and uses thereof
US10280164B2 (en) 2016-09-09 2019-05-07 Incyte Corporation Pyrazolopyridone compounds and uses thereof
IL292977A (en) 2016-09-09 2022-07-01 Incyte Corp Pyrazolopyridine derivatives as modulators of hpk1 and their use in cancer therapy
AR109595A1 (es) 2016-09-09 2018-12-26 Incyte Corp Compuestos de pirazolopirimidina y usos de estos como inhibidores de hpk1
WO2018152220A1 (en) 2017-02-15 2018-08-23 Incyte Corporation Pyrazolopyridine compounds and uses thereof
BR112019023109A2 (pt) 2017-05-04 2020-05-26 Glenmark Pharmaceuticals S.A. Composto, composição farmacêutica e método para tratar uma doença, distúrbio, síndrome ou afecção mediada por nadph oxidase em um indivíduo
US10722495B2 (en) 2017-09-08 2020-07-28 Incyte Corporation Cyanoindazole compounds and uses thereof
EP3479843A1 (en) 2017-11-01 2019-05-08 GenKyoTex Suisse SA Use of nox inhibitors for treatment of cancer
US10752635B2 (en) 2018-02-20 2020-08-25 Incyte Corporation Indazole compounds and uses thereof
US10745388B2 (en) 2018-02-20 2020-08-18 Incyte Corporation Indazole compounds and uses thereof
JP7526673B2 (ja) 2018-02-20 2024-08-01 インサイト・コーポレイション がんを治療するためのhpk1阻害剤としてのn-(フェニル)-2-(フェニル)ピリミジン-4-カルボキサミド誘導体及び関連化合物
US11299473B2 (en) 2018-04-13 2022-04-12 Incyte Corporation Benzimidazole and indole compounds and uses thereof
US10899755B2 (en) 2018-08-08 2021-01-26 Incyte Corporation Benzothiazole compounds and uses thereof
ES2973117T3 (es) 2018-09-25 2024-06-18 Incyte Corp Compuestos de pirazolo[4,3-d]pirimidina como moduladores de ALK2 y/o FGFR
KR20220059480A (ko) 2019-08-06 2022-05-10 인사이트 코포레이션 고체 형태의 hpk1 억제제
US11896719B2 (en) 2022-01-24 2024-02-13 Calliditas Therapeutics Ab Pharmaceutical compositions

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US3931407A (en) 1973-03-01 1976-01-06 American Hoechst Corporation Method of treatment with and compositions containing condensed pyrroles bearing an N-phenyl substituent
DE3728278A1 (de) 1986-12-17 1988-06-23 Bayer Ag Herbizide und fungizide mittel auf basis von substituierten pyrazolin-5-on derivaten
DE19518082A1 (de) 1995-05-17 1996-11-21 Merck Patent Gmbh 4(-Arylaminomethylen)-2,4-dihydropyrazol-3-one
WO1998037068A1 (en) 1997-02-21 1998-08-27 Bristol-Myers Squibb Company Benzoic acid derivatives and related compounds as antiarrhythmic agents
JP4196678B2 (ja) 2001-04-26 2008-12-17 味の素株式会社 複素環化合物
KR20040097375A (ko) * 2002-04-23 2004-11-17 시오노기 앤드 컴파니, 리미티드 피라졸로[1, 5-에이]피리미딘 유도체 및 이를 함유한엔에이디(피)에이취 산화효소 저해제
WO2005080378A1 (ja) 2004-02-24 2005-09-01 Mitsubishi Pharma Corporation 縮合ピリダジン誘導体
KR20070060156A (ko) 2004-10-04 2007-06-12 미리어드 제네틱스, 인크. 알츠하이머병 치료용 화합물
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EP2002835A1 (en) 2007-06-04 2008-12-17 GenKyo Tex Pyrazolo pyridine derivatives as NADPH oxidase inhibitors
EP2000176A1 (en) 2007-06-04 2008-12-10 GenKyo Tex Tetrahydroindole derivatives as NADPH Oxidase inhibitors
EP2165707A1 (en) 2008-09-23 2010-03-24 Genkyo Tex Sa Pyrazolo pyridine derivatives as NADPH oxidase inhibitors
EP2166010A1 (en) 2008-09-23 2010-03-24 Genkyo Tex Sa Pyrazolo pyridine derivatives as NADPH oxidase inhibitors
EP2166009A1 (en) 2008-09-23 2010-03-24 Genkyo Tex Sa Pyrazolo pyridine derivatives as nadph oxidase inhibitors
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CN102216309B (zh) * 2008-11-19 2014-05-07 沃泰克斯药物股份有限公司 C-met蛋白激酶的三唑并噻二唑抑制剂
EP2361911A1 (en) 2010-02-18 2011-08-31 GenKyoTex SA Pyrazolo piperidine derivatives as NADPH oxidase inhibitors
EP2361912A1 (en) 2010-02-18 2011-08-31 GenKyoTex SA Pyrazolo piperidine derivatives as NADPH oxidase inhibitors

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