JP2011529857A - 選択的グリコシダーゼインヒビターおよびその使用 - Google Patents
選択的グリコシダーゼインヒビターおよびその使用 Download PDFInfo
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- JP2011529857A JP2011529857A JP2011520296A JP2011520296A JP2011529857A JP 2011529857 A JP2011529857 A JP 2011529857A JP 2011520296 A JP2011520296 A JP 2011520296A JP 2011520296 A JP2011520296 A JP 2011520296A JP 2011529857 A JP2011529857 A JP 2011529857A
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- C12Q—MEASURING OR TESTING PROCESSES INVOLVING ENZYMES, NUCLEIC ACIDS OR MICROORGANISMS; COMPOSITIONS OR TEST PAPERS THEREFOR; PROCESSES OF PREPARING SUCH COMPOSITIONS; CONDITION-RESPONSIVE CONTROL IN MICROBIOLOGICAL OR ENZYMOLOGICAL PROCESSES
- C12Q1/00—Measuring or testing processes involving enzymes, nucleic acids or microorganisms; Compositions therefor; Processes of preparing such compositions
- C12Q1/34—Measuring or testing processes involving enzymes, nucleic acids or microorganisms; Compositions therefor; Processes of preparing such compositions involving hydrolase
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- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N2500/00—Screening for compounds of potential therapeutic value
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| US8552708P | 2008-08-01 | 2008-08-01 | |
| US61/085,527 | 2008-08-01 | ||
| PCT/CA2009/001087 WO2010012106A1 (en) | 2008-08-01 | 2009-07-31 | Selective glycosidase inhibitors and uses thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2011529857A true JP2011529857A (ja) | 2011-12-15 |
| JP2011529857A5 JP2011529857A5 (enExample) | 2012-09-06 |
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| JP2011520296A Pending JP2011529857A (ja) | 2008-08-01 | 2009-07-31 | 選択的グリコシダーゼインヒビターおよびその使用 |
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| US (2) | US8541441B2 (enExample) |
| EP (1) | EP2340250B1 (enExample) |
| JP (1) | JP2011529857A (enExample) |
| AU (1) | AU2009276222B2 (enExample) |
| CA (1) | CA2732335A1 (enExample) |
| WO (1) | WO2010012106A1 (enExample) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2436687A1 (en) * | 2005-03-01 | 2012-04-04 | Simon Fraser University | Selective glycosidase inhibitors, methods of making inhibitors, and uses thereof |
| EP2322529B1 (en) | 2006-08-31 | 2017-12-06 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| AU2009276223B2 (en) * | 2008-08-01 | 2015-04-02 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| WO2011140640A1 (en) | 2010-05-11 | 2011-11-17 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| TW201249848A (en) | 2010-11-08 | 2012-12-16 | Merck Sharp & Dohme | Selective glycosidase inhibitors and uses thereof |
| US8901087B2 (en) | 2010-11-08 | 2014-12-02 | Merck Sharp & Dohme Corp. | Selective glycosidase inhibitors and uses thereof |
| WO2012061927A1 (en) | 2010-11-08 | 2012-05-18 | Alectos Therapeutics, Inc. | Selective glycosidase inhibitors and uses thereof |
| LT2655388T (lt) | 2010-12-23 | 2016-11-10 | Alectos Therapeutics Inc. | Selektyvieji glikozidazės inhibitoriai ir jų panaudojimas |
| WO2012126091A1 (en) | 2011-03-24 | 2012-09-27 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| EP2691407B1 (en) | 2011-03-31 | 2017-02-22 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| WO2013000084A1 (en) | 2011-06-27 | 2013-01-03 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| EP2726468B1 (en) | 2011-06-27 | 2017-04-12 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| WO2013000086A1 (en) | 2011-06-27 | 2013-01-03 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| US9861686B2 (en) | 2011-12-05 | 2018-01-09 | Ben-Gurion University Of The Negev Research & Development Authority | Diagnostic and therapeutic methods and their application in amyotrophic lateral sclerosis (ALS) |
| CA2871920C (en) | 2012-05-08 | 2021-03-09 | Merck Sharp & Dohme Corp. | Permeable glycosidase inhibitors and uses thereof |
| US9670195B2 (en) | 2012-08-31 | 2017-06-06 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| US9809537B2 (en) | 2012-08-31 | 2017-11-07 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| US9695197B2 (en) | 2012-10-31 | 2017-07-04 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| WO2024083820A1 (en) | 2022-10-18 | 2024-04-25 | Institut National de la Santé et de la Recherche Médicale | Method and composition for determining the level of o-glcnacylation in horses |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH05507474A (ja) * | 1990-06-04 | 1993-10-28 | メレルダウファーマス―ティカルズ インコーポレイテッド | ６―アミノオクタヒドロインドリジントリオールの誘導体 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5300265A (en) | 1989-06-26 | 1994-04-05 | Fluid Dynamics Pty Ltd. | Controlled atmosphere generating equipment |
| US20080166323A1 (en) | 2004-04-14 | 2008-07-10 | Uab Research Foundation | Activators of Hexosamine Biosynthesis as Inhibitors of Injury Induced by Ischemia or Hermorrhagic Shock |
| EP2436687A1 (en) | 2005-03-01 | 2012-04-04 | Simon Fraser University | Selective glycosidase inhibitors, methods of making inhibitors, and uses thereof |
| EP2322529B1 (en) | 2006-08-31 | 2017-12-06 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
-
2009
- 2009-07-31 EP EP09802332.8A patent/EP2340250B1/en not_active Not-in-force
- 2009-07-31 WO PCT/CA2009/001087 patent/WO2010012106A1/en not_active Ceased
- 2009-07-31 AU AU2009276222A patent/AU2009276222B2/en not_active Ceased
- 2009-07-31 US US13/057,062 patent/US8541441B2/en not_active Expired - Fee Related
- 2009-07-31 JP JP2011520296A patent/JP2011529857A/ja active Pending
- 2009-07-31 CA CA2732335A patent/CA2732335A1/en not_active Abandoned
-
2013
- 2013-08-15 US US13/967,818 patent/US20140051719A1/en not_active Abandoned
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH05507474A (ja) * | 1990-06-04 | 1993-10-28 | メレルダウファーマス―ティカルズ インコーポレイテッド | ６―アミノオクタヒドロインドリジントリオールの誘導体 |
Non-Patent Citations (1)
| Title |
|---|
| JPN6013061794; Ｔｅｔｒａｈｅｄｒｏｎ ５０，７, 1994, ２１３１-２１６０ * |
Also Published As
| Publication number | Publication date |
|---|---|
| US8541441B2 (en) | 2013-09-24 |
| US20120095033A1 (en) | 2012-04-19 |
| EP2340250A1 (en) | 2011-07-06 |
| AU2009276222A1 (en) | 2010-02-04 |
| AU2009276222B2 (en) | 2015-03-05 |
| WO2010012106A1 (en) | 2010-02-04 |
| EP2340250A4 (en) | 2011-10-26 |
| EP2340250B1 (en) | 2019-06-26 |
| CA2732335A1 (en) | 2010-02-04 |
| US20140051719A1 (en) | 2014-02-20 |
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