JP2011514339A5 - - Google Patents
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- Publication number
- JP2011514339A5 JP2011514339A5 JP2010547919A JP2010547919A JP2011514339A5 JP 2011514339 A5 JP2011514339 A5 JP 2011514339A5 JP 2010547919 A JP2010547919 A JP 2010547919A JP 2010547919 A JP2010547919 A JP 2010547919A JP 2011514339 A5 JP2011514339 A5 JP 2011514339A5
- Authority
- JP
- Japan
- Prior art keywords
- optionally substituted
- oxo
- methyl
- substituted
- diazepan
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US3289808P | 2008-02-29 | 2008-02-29 | |
| US61/032,898 | 2008-02-29 | ||
| PCT/AU2009/000232 WO2009105825A1 (en) | 2008-02-29 | 2009-02-27 | 3-substituted-1,4-diazepan-2-one melanocortin-5 receptor antagonists |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011514339A JP2011514339A (ja) | 2011-05-06 |
| JP2011514339A5 true JP2011514339A5 (https=) | 2014-02-20 |
| JP5503559B2 JP5503559B2 (ja) | 2014-05-28 |
Family
ID=41015442
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010547919A Expired - Fee Related JP5503559B2 (ja) | 2008-02-29 | 2009-02-27 | ３−置換−１，４−ジアゼパン−２−オンメラノコルチン−５受容体アンタゴニスト |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US8440653B2 (https=) |
| EP (1) | EP2257533B1 (https=) |
| JP (1) | JP5503559B2 (https=) |
| KR (1) | KR101620116B1 (https=) |
| CN (1) | CN102007106B (https=) |
| AU (1) | AU2009219108B2 (https=) |
| BR (1) | BRPI0907898B8 (https=) |
| CA (1) | CA2716256C (https=) |
| ES (1) | ES2439964T3 (https=) |
| IL (1) | IL207701A (https=) |
| MX (1) | MX2010009486A (https=) |
| NZ (1) | NZ587362A (https=) |
| RU (1) | RU2524245C2 (https=) |
| WO (1) | WO2009105825A1 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5503558B2 (ja) * | 2008-02-29 | 2014-05-28 | ミメチカ ピーティーワイ エルティーディー | Ｍｃ５受容体の活性を調節する方法およびこの受容体と関連する症状の治療 |
| WO2016149628A1 (en) * | 2015-03-19 | 2016-09-22 | Chembridge Corporation | Tgr5 agonists |
| US11485725B2 (en) | 2017-12-15 | 2022-11-01 | Auransa Inc. | Derivatives of piperlongumine and uses thereof |
| CN116262115B (zh) * | 2021-12-15 | 2026-02-24 | 深圳先进技术研究院 | 释放氨基酸及其衍生物类药物的医用材料及其应用方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AUPP254898A0 (en) * | 1998-03-24 | 1998-04-23 | University Of Queensland, The | Peptide turn mimetics |
| IL152701A0 (en) * | 2000-05-25 | 2003-06-24 | Hoffmann La Roche | Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists |
| AU2002331064B2 (en) * | 2001-08-10 | 2007-08-23 | Palatin Technologies, Inc. | Peptidomimetics of biologically active metallopeptides |
| US6916812B2 (en) | 2001-10-09 | 2005-07-12 | Bristol-Myers Squibb Company | Alpha-aminoamide derivatives as melanocortin agonists |
| AU2003216274A1 (en) * | 2002-02-11 | 2003-09-04 | Neurocrine Biosciences, Inc. | Pyrrole derivatives as ligands of melanocortin receptors |
| WO2008017852A1 (en) * | 2006-08-11 | 2008-02-14 | Palatin Technologies, Inc. | Diamine-containing, tetra- substituted piperazine compounds as melanocortin receptor modulators |
| JP5503558B2 (ja) * | 2008-02-29 | 2014-05-28 | ミメチカ ピーティーワイ エルティーディー | Ｍｃ５受容体の活性を調節する方法およびこの受容体と関連する症状の治療 |
-
2009
- 2009-02-27 US US12/919,973 patent/US8440653B2/en not_active Expired - Fee Related
- 2009-02-27 CN CN200980113158.7A patent/CN102007106B/zh not_active Expired - Fee Related
- 2009-02-27 WO PCT/AU2009/000232 patent/WO2009105825A1/en not_active Ceased
- 2009-02-27 AU AU2009219108A patent/AU2009219108B2/en not_active Ceased
- 2009-02-27 MX MX2010009486A patent/MX2010009486A/es active IP Right Grant
- 2009-02-27 KR KR1020107021385A patent/KR101620116B1/ko not_active Expired - Fee Related
- 2009-02-27 JP JP2010547919A patent/JP5503559B2/ja not_active Expired - Fee Related
- 2009-02-27 ES ES09716109.5T patent/ES2439964T3/es active Active
- 2009-02-27 CA CA2716256A patent/CA2716256C/en not_active Expired - Fee Related
- 2009-02-27 RU RU2010137033/04A patent/RU2524245C2/ru active
- 2009-02-27 NZ NZ587362A patent/NZ587362A/en not_active IP Right Cessation
- 2009-02-27 EP EP09716109.5A patent/EP2257533B1/en not_active Not-in-force
- 2009-02-27 BR BRPI0907898A patent/BRPI0907898B8/pt not_active IP Right Cessation
-
2010
- 2010-08-19 IL IL207701A patent/IL207701A/en active IP Right Grant
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