JP2011510972A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2011510972A5 JP2011510972A5 JP2010544816A JP2010544816A JP2011510972A5 JP 2011510972 A5 JP2011510972 A5 JP 2011510972A5 JP 2010544816 A JP2010544816 A JP 2010544816A JP 2010544816 A JP2010544816 A JP 2010544816A JP 2011510972 A5 JP2011510972 A5 JP 2011510972A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- oxo
- triaza
- hexahydro
- carboxylic acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP08290076A EP2090579A1 (en) | 2008-01-29 | 2008-01-29 | Substituted heteroarylamide diazepinopyrimidone derivatives |
| EP08290076.2 | 2008-01-29 | ||
| PCT/IB2009/000397 WO2009095792A2 (en) | 2008-01-29 | 2009-01-27 | Substituted heteroarylamide diazepinopyrimidone derivatives |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011510972A JP2011510972A (ja) | 2011-04-07 |
| JP2011510972A5 true JP2011510972A5 (enExample) | 2012-01-19 |
| JP5611837B2 JP5611837B2 (ja) | 2014-10-22 |
Family
ID=39540691
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010544816A Expired - Fee Related JP5611837B2 (ja) | 2008-01-29 | 2009-01-27 | 置換へテロアリールアミドジアゼピノピリミドン誘導体 |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US8507475B2 (enExample) |
| EP (2) | EP2090579A1 (enExample) |
| JP (1) | JP5611837B2 (enExample) |
| KR (1) | KR20100117583A (enExample) |
| CN (1) | CN101986782A (enExample) |
| AR (1) | AR070273A1 (enExample) |
| AU (1) | AU2009208731A1 (enExample) |
| BR (1) | BRPI0906359A2 (enExample) |
| CA (1) | CA2713289A1 (enExample) |
| EA (1) | EA201070891A1 (enExample) |
| IL (1) | IL207192A0 (enExample) |
| MX (1) | MX2010008362A (enExample) |
| NZ (1) | NZ587068A (enExample) |
| TW (1) | TW200936588A (enExample) |
| WO (1) | WO2009095792A2 (enExample) |
| ZA (1) | ZA201005382B (enExample) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2085399A1 (en) * | 2008-01-29 | 2009-08-05 | Sanofi-Aventis | substituted arylamide oxazepinopyrimidone derivatives |
| EP2085400A1 (en) * | 2008-01-29 | 2009-08-05 | Sanofi-Aventis | Substituted heteroarylamide oxazepinopyrimidone derivatives |
| EP2090578A1 (en) * | 2008-01-29 | 2009-08-19 | Sanofi-Aventis | Substituted arylamide diazepinopyrimidone derivatives for the treatment of neurodegenerative diseases caused by abnormal activity of GSK3-beta |
| EP2138494A1 (en) * | 2008-06-26 | 2009-12-30 | Sanofi-Aventis | Substituted alkyl pyrimidin-4-one derivatives |
| WO2011107494A1 (de) | 2010-03-03 | 2011-09-09 | Sanofi | Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung |
| US8530413B2 (en) | 2010-06-21 | 2013-09-10 | Sanofi | Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments |
| TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
| TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
| TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
| WO2013037390A1 (en) | 2011-09-12 | 2013-03-21 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
| EP2760862B1 (en) | 2011-09-27 | 2015-10-21 | Sanofi | 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
| PE20181893A1 (es) * | 2016-02-15 | 2018-12-11 | Sanofi Sa | Nuevos compuestos de 6,7-dihidro-5h-benzo[7]anuleno sustituidos, procesos para su preparacion y usos terapeuticos de los mismos |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EG13192A (en) | 1976-02-10 | 1982-12-31 | Rhone Poulenc Ind | Nouveaux derives du dithiole-1,2 leur preparation et les compositions qui les contiennent |
| US5629322A (en) | 1994-11-15 | 1997-05-13 | Merck & Co., Inc. | Cyclic amidine analogs as inhibitors of nitric oxide synthase |
| JP3188715B2 (ja) | 1995-11-01 | 2001-07-16 | メルク エンド カンパニー インコーポレーテッド | 一酸化窒素シンターゼの阻害物質としてのヘキサヒドロ−５−イミノ−１，４−ヘテロアゼピン誘導体 |
| US20030096813A1 (en) * | 2001-04-20 | 2003-05-22 | Jingrong Cao | Compositions useful as inhibitors of GSK-3 |
| CN1247586C (zh) * | 2001-09-21 | 2006-03-29 | 赛诺菲安万特 | 治疗神经退化性疾病的取代的2－嘧啶基－6,7,8,9－四氢嘧啶并[1,2－a]嘧啶－4－酮及7－嘧啶基－2,3－二氢咪唑并[1,2－a]嘧啶－5(1h)酮衍生物 |
| EP1557417B1 (en) * | 2003-12-19 | 2007-03-07 | Sanofi-Aventis | Substituted 8'-pyri(mi)dinyl-dihydrospiro-[cycloalkylamine]-pyrimido[1,2-a] pyrimidin-6-one derivatives |
| EP1790649A1 (en) * | 2005-11-21 | 2007-05-30 | Sanofi-Aventis | Substituted bicyclic pyrimidone derivatives |
| EP2085399A1 (en) * | 2008-01-29 | 2009-08-05 | Sanofi-Aventis | substituted arylamide oxazepinopyrimidone derivatives |
| EP2085400A1 (en) * | 2008-01-29 | 2009-08-05 | Sanofi-Aventis | Substituted heteroarylamide oxazepinopyrimidone derivatives |
| EP2090578A1 (en) * | 2008-01-29 | 2009-08-19 | Sanofi-Aventis | Substituted arylamide diazepinopyrimidone derivatives for the treatment of neurodegenerative diseases caused by abnormal activity of GSK3-beta |
-
2008
- 2008-01-29 EP EP08290076A patent/EP2090579A1/en not_active Withdrawn
-
2009
- 2009-01-23 TW TW098103040A patent/TW200936588A/zh unknown
- 2009-01-27 EA EA201070891A patent/EA201070891A1/ru unknown
- 2009-01-27 EP EP09705869.7A patent/EP2238140B1/en active Active
- 2009-01-27 MX MX2010008362A patent/MX2010008362A/es not_active Application Discontinuation
- 2009-01-27 JP JP2010544816A patent/JP5611837B2/ja not_active Expired - Fee Related
- 2009-01-27 KR KR1020107016905A patent/KR20100117583A/ko not_active Withdrawn
- 2009-01-27 WO PCT/IB2009/000397 patent/WO2009095792A2/en not_active Ceased
- 2009-01-27 CN CN2009801106975A patent/CN101986782A/zh active Pending
- 2009-01-27 AU AU2009208731A patent/AU2009208731A1/en not_active Abandoned
- 2009-01-27 CA CA2713289A patent/CA2713289A1/en not_active Abandoned
- 2009-01-27 BR BRPI0906359A patent/BRPI0906359A2/pt not_active IP Right Cessation
- 2009-01-27 NZ NZ587068A patent/NZ587068A/en not_active IP Right Cessation
- 2009-01-28 AR ARP090100256A patent/AR070273A1/es unknown
-
2010
- 2010-07-25 IL IL207192A patent/IL207192A0/en unknown
- 2010-07-27 US US12/844,273 patent/US8507475B2/en not_active Expired - Fee Related
- 2010-07-28 ZA ZA2010/05382A patent/ZA201005382B/en unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2011510972A5 (enExample) | ||
| AU2015222584B2 (en) | 2,4-disubstituted phenylene-1,5-diamine derivatives and applications thereof, and pharmaceutical compositions and pharmaceutically acceptable compositions prepared therefrom | |
| AU2020302338A1 (en) | 2,3-dihydroquinazolin compounds as NAV1.8 inhibitors | |
| EP4277901A1 (en) | Isoindolinone compounds | |
| JP2016512823A5 (enExample) | ||
| JP6951406B2 (ja) | フラバグリン誘導体 | |
| CN108290867B (zh) | 一种制备酪氨酸激酶抑制剂及其衍生物的方法 | |
| JP6965478B2 (ja) | ２−アミノキナゾリノン誘導体 | |
| EA031614B1 (ru) | Трициклические атропоизомерные соединения | |
| Ma et al. | Discovery of novel quinoline-based mTOR inhibitors via introducing intra-molecular hydrogen bonding scaffold (iMHBS): The design, synthesis and biological evaluation | |
| JP2018536698A (ja) | Ｅｇｆｒキナーゼ阻害剤およびその製造方法と使用 | |
| JP2024001109A (ja) | Ｊａｋ阻害化合物のキシナホ酸塩 | |
| JP2016124825A (ja) | 多置換７−デアザプリン誘導体合成のための２，６−ジクロロ−８−ヨード−７−デアザプリン | |
| CA3159211A1 (en) | Fluorinated quinoline, quinoxaline and benzo[b][1,4]oxazine derivatives as dihydroorotate dehydrogenase (dhodh) inhibitors for the treatment of cancer, autoimmune and inflammatory diseases | |
| MX2009010243A (es) | Compuestos de quinolina apropiados para tratar trastornos que responden a la modulacion del receptor de serotonina 5-ht6. | |
| AU2009267828A1 (en) | Antineoplastic derivatives of 4-OXO-L, 4-dihydro-quinoline, preparation thereof, and therapeutic use thereof | |
| CN102249982B (zh) | 新型截短侧耳素类化合物、其药物组合物及其制备方法和用途 | |
| DK3189060T3 (en) | DERIVATIVES OF MACROCYCLIC N-ARYL-2-AMINO-4-ARYL-PYRIMIDINE POLYETHERS AS FTL3 AND JAK INHIBITORS | |
| Xin et al. | Synthesis and pharmacological evaluation of trifluoromethyl containing 4-(2-pyrimidinylamino) benzamides as Hedgehog signaling pathway inhibitors | |
| JPWO2019059344A1 (ja) | 化学活性化型水溶性プロドラッグ | |
| KR20150117123A (ko) | 블로난세린의 온화한 제조방법 | |
| US20120157482A1 (en) | Compounds and methods | |
| JP5017101B2 (ja) | 不斉四置換炭素原子含有化合物の製法 | |
| JP7787063B2 (ja) | オーロラキナーゼ阻害剤およびその使用 | |
| JP5536771B2 (ja) | セロトニン作動性活性を有する化合物、その製造方法およびそれを含む医薬組成物 |