JP2011506323A5 - - Google Patents
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- Publication number
- JP2011506323A5 JP2011506323A5 JP2010536949A JP2010536949A JP2011506323A5 JP 2011506323 A5 JP2011506323 A5 JP 2011506323A5 JP 2010536949 A JP2010536949 A JP 2010536949A JP 2010536949 A JP2010536949 A JP 2010536949A JP 2011506323 A5 JP2011506323 A5 JP 2011506323A5
- Authority
- JP
- Japan
- Prior art keywords
- hydrogen
- group
- formula
- alkyl
- oxygen protecting
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US1240907P | 2007-12-07 | 2007-12-07 | |
| US1240807P | 2007-12-07 | 2007-12-07 | |
| US1241107P | 2007-12-07 | 2007-12-07 | |
| US61/012,411 | 2007-12-07 | ||
| US61/012,408 | 2007-12-07 | ||
| US61/012,409 | 2007-12-07 | ||
| US8004808P | 2008-07-11 | 2008-07-11 | |
| US61/080,048 | 2008-07-11 | ||
| PCT/US2008/013498 WO2009075818A1 (en) | 2007-12-07 | 2008-12-08 | Intermediates and methods for making zearalenone macrolide analogs |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014042331A Division JP2014141498A (ja) | 2007-12-07 | 2014-03-05 | ゼラレノンマクロライドアナログを作製するための中間体および方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011506323A JP2011506323A (ja) | 2011-03-03 |
| JP2011506323A5 true JP2011506323A5 (OSRAM) | 2012-02-02 |
| JP5496908B2 JP5496908B2 (ja) | 2014-05-21 |
Family
ID=40445478
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010536949A Active JP5496908B2 (ja) | 2007-12-07 | 2008-12-08 | ゼラレノンマクロライドアナログを作製するための中間体および方法 |
| JP2010536950A Active JP5492786B2 (ja) | 2007-12-07 | 2008-12-08 | ゼラレノンマクロライドアナログを作製するための中間体および方法 |
| JP2014042331A Withdrawn JP2014141498A (ja) | 2007-12-07 | 2014-03-05 | ゼラレノンマクロライドアナログを作製するための中間体および方法 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010536950A Active JP5492786B2 (ja) | 2007-12-07 | 2008-12-08 | ゼラレノンマクロライドアナログを作製するための中間体および方法 |
| JP2014042331A Withdrawn JP2014141498A (ja) | 2007-12-07 | 2014-03-05 | ゼラレノンマクロライドアナログを作製するための中間体および方法 |
Country Status (10)
| Country | Link |
|---|---|
| US (3) | US8350059B2 (OSRAM) |
| EP (2) | EP2231635B1 (OSRAM) |
| JP (3) | JP5496908B2 (OSRAM) |
| CN (2) | CN101889006B (OSRAM) |
| BR (2) | BRPI0820958B1 (OSRAM) |
| CA (2) | CA2708141C (OSRAM) |
| IL (2) | IL205954A (OSRAM) |
| MX (2) | MX2010006091A (OSRAM) |
| RU (2) | RU2478630C2 (OSRAM) |
| WO (2) | WO2009075818A1 (OSRAM) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN104876904A (zh) * | 2002-03-08 | 2015-09-02 | 卫材R&D管理株式会社 | 用作医药品的大环化合物 |
| US8609640B2 (en) | 2007-07-25 | 2013-12-17 | Eisai, Inc. | Multikinase inhibitors for use in the treatment of cancer |
| EP2231635B1 (en) * | 2007-12-07 | 2014-03-19 | Eisai R&D Management Co., Ltd. | Intermediates and methods for making zearalenone macrolide analogs |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU561147B2 (en) * | 1982-09-13 | 1987-04-30 | Eli Lilly And Company | 20-amino macrolide antibiotics |
| GB9225396D0 (en) | 1992-12-04 | 1993-01-27 | Sandoz Ltd | Improvements in or relating to organic compounds |
| US5795910A (en) | 1994-10-28 | 1998-08-18 | Cor Therapeutics, Inc. | Method and compositions for inhibiting protein kinases |
| RU2213741C2 (ru) * | 1997-07-08 | 2003-10-10 | Бристол-Маерс Сквибб Компани | Производные эпотилона |
| JP2004292315A (ja) | 2000-12-14 | 2004-10-21 | Chugai Pharmaceut Co Ltd | Ｔａｋ１阻害剤 |
| JP2004292314A (ja) | 2000-12-14 | 2004-10-21 | Chugai Pharmaceut Co Ltd | ケラチノサイト増殖抑制剤 |
| CN104876904A (zh) * | 2002-03-08 | 2015-09-02 | 卫材R&D管理株式会社 | 用作医药品的大环化合物 |
| US7915306B2 (en) * | 2002-03-08 | 2011-03-29 | Eisai Co., Ltd. | Macrocyclic compounds useful as pharmaceuticals |
| CA2696021C (en) | 2006-08-11 | 2015-09-29 | Nicolas Winssinger | Macrocyclic compounds useful as inhibitors of kinases and hsp90 |
| US8513440B2 (en) * | 2007-06-05 | 2013-08-20 | Universite De Strasbourg | Compositions and methods comprising analogues of radicicol A |
| TW200924749A (en) * | 2007-07-25 | 2009-06-16 | Eisai R & Amp D Man Co Ltd | Zearalenone macrolide derivatives and uses of the same |
| US8609640B2 (en) * | 2007-07-25 | 2013-12-17 | Eisai, Inc. | Multikinase inhibitors for use in the treatment of cancer |
| EP2231635B1 (en) * | 2007-12-07 | 2014-03-19 | Eisai R&D Management Co., Ltd. | Intermediates and methods for making zearalenone macrolide analogs |
-
2008
- 2008-12-08 EP EP08860534.0A patent/EP2231635B1/en active Active
- 2008-12-08 MX MX2010006091A patent/MX2010006091A/es active IP Right Grant
- 2008-12-08 JP JP2010536949A patent/JP5496908B2/ja active Active
- 2008-12-08 RU RU2010128103/04A patent/RU2478630C2/ru active
- 2008-12-08 MX MX2010005999A patent/MX2010005999A/es active IP Right Grant
- 2008-12-08 BR BRPI0820958-8A patent/BRPI0820958B1/pt active IP Right Grant
- 2008-12-08 BR BRPI0820953-7A patent/BRPI0820953B1/pt active IP Right Grant
- 2008-12-08 US US12/746,672 patent/US8350059B2/en active Active
- 2008-12-08 CA CA2708141A patent/CA2708141C/en active Active
- 2008-12-08 CN CN2008801195442A patent/CN101889006B/zh active Active
- 2008-12-08 CA CA2708143A patent/CA2708143C/en active Active
- 2008-12-08 US US12/746,675 patent/US8507696B2/en active Active
- 2008-12-08 WO PCT/US2008/013498 patent/WO2009075818A1/en not_active Ceased
- 2008-12-08 CN CN200880119543.8A patent/CN101889005B/zh active Active
- 2008-12-08 EP EP08860344.4A patent/EP2231634B1/en active Active
- 2008-12-08 WO PCT/US2008/013512 patent/WO2009075823A1/en not_active Ceased
- 2008-12-08 RU RU2010128096/04A patent/RU2497803C2/ru active
- 2008-12-08 JP JP2010536950A patent/JP5492786B2/ja active Active
-
2010
- 2010-05-25 IL IL205954A patent/IL205954A/en active IP Right Grant
- 2010-05-26 IL IL205983A patent/IL205983A/en active IP Right Grant
-
2013
- 2013-01-03 US US13/733,562 patent/US20130211103A1/en not_active Abandoned
-
2014
- 2014-03-05 JP JP2014042331A patent/JP2014141498A/ja not_active Withdrawn
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