JP2011500513A5 - - Google Patents
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- Publication number
- JP2011500513A5 JP2011500513A5 JP2010525229A JP2010525229A JP2011500513A5 JP 2011500513 A5 JP2011500513 A5 JP 2011500513A5 JP 2010525229 A JP2010525229 A JP 2010525229A JP 2010525229 A JP2010525229 A JP 2010525229A JP 2011500513 A5 JP2011500513 A5 JP 2011500513A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- alkyl
- general formula
- arylalkyl
- haloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 125000000217 alkyl group Chemical group 0.000 claims description 13
- 125000003710 aryl alkyl group Chemical group 0.000 claims description 11
- 125000001188 haloalkyl group Chemical group 0.000 claims description 11
- 125000003118 aryl group Chemical group 0.000 claims description 10
- 125000000753 cycloalkyl group Chemical group 0.000 claims description 9
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims description 4
- 150000001875 compounds Chemical class 0.000 claims 13
- 238000000034 method Methods 0.000 claims 8
- 229910052801 chlorine Inorganic materials 0.000 claims 7
- 239000000460 chlorine Chemical group 0.000 claims 7
- -1 4-aminobut-2-enolide compound Chemical class 0.000 claims 5
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical group [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 claims 5
- 229910052731 fluorine Inorganic materials 0.000 claims 5
- 239000011737 fluorine Substances 0.000 claims 5
- 125000001153 fluoro group Chemical group F* 0.000 claims 4
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 3
- 125000001424 substituent group Chemical group 0.000 claims 3
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical group [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 claims 2
- 229910052783 alkali metal Inorganic materials 0.000 claims 2
- 150000001340 alkali metals Chemical class 0.000 claims 2
- 229910052784 alkaline earth metal Inorganic materials 0.000 claims 2
- 150000001342 alkaline earth metals Chemical class 0.000 claims 2
- 239000002585 base Substances 0.000 claims 2
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Chemical group BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 claims 2
- 229910052794 bromium Inorganic materials 0.000 claims 2
- 125000001309 chloro group Chemical group Cl* 0.000 claims 2
- 125000004093 cyano group Chemical group *C#N 0.000 claims 2
- 229910052736 halogen Inorganic materials 0.000 claims 2
- 150000002367 halogens Chemical group 0.000 claims 2
- 229910052739 hydrogen Inorganic materials 0.000 claims 2
- 239000001257 hydrogen Substances 0.000 claims 2
- 125000004435 hydrogen atom Chemical class [H]* 0.000 claims 2
- 238000002360 preparation method Methods 0.000 claims 2
- 125000004504 1,2,4-oxadiazolyl group Chemical group 0.000 claims 1
- 125000001376 1,2,4-triazolyl group Chemical group N1N=C(N=C1)* 0.000 claims 1
- 125000004517 1,2,5-thiadiazolyl group Chemical group 0.000 claims 1
- 125000004105 2-pyridyl group Chemical group N1=C([*])C([H])=C([H])C([H])=C1[H] 0.000 claims 1
- 125000003349 3-pyridyl group Chemical group N1=C([H])C([*])=C([H])C([H])=C1[H] 0.000 claims 1
- 125000000339 4-pyridyl group Chemical group N1=C([H])C([H])=C([*])C([H])=C1[H] 0.000 claims 1
- VGCXGMAHQTYDJK-UHFFFAOYSA-N Chloroacetyl chloride Chemical compound ClCC(Cl)=O VGCXGMAHQTYDJK-UHFFFAOYSA-N 0.000 claims 1
- IYXGSMUGOJNHAZ-UHFFFAOYSA-N Ethyl malonate Chemical compound CCOC(=O)CC(=O)OCC IYXGSMUGOJNHAZ-UHFFFAOYSA-N 0.000 claims 1
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 claims 1
- 125000003342 alkenyl group Chemical group 0.000 claims 1
- 150000004703 alkoxides Chemical class 0.000 claims 1
- 125000004183 alkoxy alkyl group Chemical group 0.000 claims 1
- 125000003545 alkoxy group Chemical group 0.000 claims 1
- 125000000304 alkynyl group Chemical group 0.000 claims 1
- 150000001540 azides Chemical group 0.000 claims 1
- 229940089960 chloroacetate Drugs 0.000 claims 1
- 125000001316 cycloalkyl alkyl group Chemical group 0.000 claims 1
- VEUUMBGHMNQHGO-UHFFFAOYSA-N ethyl chloroacetate Chemical compound CCOC(=O)CCl VEUUMBGHMNQHGO-UHFFFAOYSA-N 0.000 claims 1
- 125000000262 haloalkenyl group Chemical group 0.000 claims 1
- 125000004438 haloalkoxy group Chemical group 0.000 claims 1
- 125000005347 halocycloalkyl group Chemical group 0.000 claims 1
- 125000004461 halocycloalkylalkyl group Chemical group 0.000 claims 1
- 125000001786 isothiazolyl group Chemical group 0.000 claims 1
- 125000000842 isoxazolyl group Chemical group 0.000 claims 1
- 238000004519 manufacturing process Methods 0.000 claims 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 1
- 125000002971 oxazolyl group Chemical group 0.000 claims 1
- LPNYRYFBWFDTMA-UHFFFAOYSA-N potassium tert-butoxide Chemical compound [K+].CC(C)(C)[O-] LPNYRYFBWFDTMA-UHFFFAOYSA-N 0.000 claims 1
- 125000004944 pyrazin-3-yl group Chemical group [H]C1=C([H])N=C(*)C([H])=N1 0.000 claims 1
- 125000003226 pyrazolyl group Chemical group 0.000 claims 1
- 125000002206 pyridazin-3-yl group Chemical group [H]C1=C([H])C([H])=C(*)N=N1 0.000 claims 1
- 125000000714 pyrimidinyl group Chemical group 0.000 claims 1
- 229910052708 sodium Inorganic materials 0.000 claims 1
- 239000011734 sodium Substances 0.000 claims 1
- 239000007858 starting material Substances 0.000 claims 1
- 125000001544 thienyl group Chemical group 0.000 claims 1
- 125000000876 trifluoromethoxy group Chemical group FC(F)(F)O* 0.000 claims 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07116639A EP2042496A1 (de) | 2007-09-18 | 2007-09-18 | Verfahren zur Herstellung von 4-Aminobut-2-enoliden |
| EP07116639.1 | 2007-09-18 | ||
| PCT/EP2008/007270 WO2009036899A1 (de) | 2007-09-18 | 2008-09-05 | Verfahren zur herstellung von 4-aminobut-2-enoliden |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011500513A JP2011500513A (ja) | 2011-01-06 |
| JP2011500513A5 true JP2011500513A5 (enExample) | 2013-11-14 |
| JP5611043B2 JP5611043B2 (ja) | 2014-10-22 |
Family
ID=39167552
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010525229A Active JP5611043B2 (ja) | 2007-09-18 | 2008-09-05 | ４−アミノブタ−２−エノリド類を調製する方法 |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US8273904B2 (enExample) |
| EP (2) | EP2042496A1 (enExample) |
| JP (1) | JP5611043B2 (enExample) |
| KR (1) | KR101516606B1 (enExample) |
| CN (2) | CN101801948B (enExample) |
| BR (1) | BRPI0816911B1 (enExample) |
| DK (1) | DK2193128T3 (enExample) |
| ES (1) | ES2612058T3 (enExample) |
| IL (1) | IL203761A (enExample) |
| MX (1) | MX2010001963A (enExample) |
| TW (1) | TWI432419B (enExample) |
| WO (1) | WO2009036899A1 (enExample) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2230237A1 (de) | 2009-03-16 | 2010-09-22 | Bayer CropScience AG | Neues Verfahren zur Herstellung von Enaminocarbonyl-Verbindungen |
| EP2230236A1 (de) | 2009-03-16 | 2010-09-22 | Bayer CropScience AG | Neues Verfahren zur Herstellung von Enaminocarbonyl-Verbindungen |
| MX2012001675A (es) * | 2009-08-11 | 2012-03-06 | Bayer Cropscience Ag | Procedimiento para preparar 2,4-dioxotetrahidrofuran-3-carboxilato s. |
| TW201111370A (en) * | 2009-08-18 | 2011-04-01 | Bayer Cropscience Ag | Novel process for the preparation of 4-aminobut-2-enolides |
| CN102741244A (zh) | 2009-10-26 | 2012-10-17 | 拜耳作物科学公司 | 4-[[(6-氯吡啶-3-基)甲基](2,2-二氟乙基)氨基]呋喃-2(5h)-酮的新固体形式 |
| WO2011051242A1 (de) | 2009-10-27 | 2011-05-05 | Bayer Technology Services Gmbh | Co-kristall von 4- { [ (6-chlorpyrid-3-yl) methyl] (2,2-difluorethyl) amino} furan-2 (5h) -on mit salizylsäure und dessen verwendung als pestizid |
| US20120270904A1 (en) * | 2009-10-27 | 2012-10-25 | Bayer Technology Services Gmbh | Co-crystal of 4-furan-2(5h)-one with oxalic acid and use thereof as pesticide |
| US20120283294A1 (en) | 2009-10-27 | 2012-11-08 | Bayer Technology Services Gmbh | Co-crystal of 4-furan-2(5h)-one with benzoic acid and use thereof as pesticide |
| DK2516421T3 (en) * | 2009-12-23 | 2016-11-28 | Bayer Ip Gmbh | New process for the preparation of 4-aminobut-2-enoliden starting from 4-alkoxyfuran-2 (5H) -one or 4-arylalkoxyfuran-2- (5H) -one |
| US20130331417A1 (en) * | 2010-12-09 | 2013-12-12 | Bayer Intellectual Property Gmbh | Insecticidal mixtures with improved properties |
| EP2648515A1 (en) * | 2010-12-09 | 2013-10-16 | Bayer Intellectual Property GmbH | Pesticidal mixtures with improved properties |
| JP5970002B2 (ja) * | 2011-03-03 | 2016-08-17 | バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ ＧｍｂＨ | ４−ヒドロキシ−２−オキソ−２，５−ジヒドロフラン−３−カルボン酸化合物のナトリウム塩またはカリウム塩の製造方法 |
| KR101977919B1 (ko) * | 2012-08-01 | 2019-05-13 | 바이엘 크롭사이언스 악티엔게젤샤프트 | 특정 4-하이드록시-2-옥소-2,5-디하이드로푸란-3-카복실산 에스테르의 알칼리 금속 염의 다단 제조방법 |
| CN105503708B (zh) * | 2016-01-26 | 2018-05-29 | 南开大学 | 一类含二氟乙基的杂环化合物及其制备方法和用途 |
| EP4295683A1 (en) | 2022-06-21 | 2023-12-27 | Bayer Aktiengesellschaft | Agrochemical formulations comprising crystalline form a of 4-[(6-chloro-3-pyridylmethyl)(2,2-difluoroethyl)amino]furan-2(5h)-one |
| KR20250020435A (ko) | 2022-06-06 | 2025-02-11 | 바이엘 악티엔게젤샤프트 | 4-[(6-클로로-3-피리딜메틸)(2,2-디플루오로에틸)아미노]푸란-2(5h)-온의결정질 형태 a를 포함하는 농약 제제 |
| WO2025114238A1 (en) | 2023-12-01 | 2025-06-05 | Bayer Aktiengesellschaft | Solid agrochemical formulations comprising crystalline form a of 4-[(6-chloro-3-pyridylmethyl)(2,2- difluoroethyl)amino]furan-2(5h)-one |
| CN122476959A (zh) | 2023-12-05 | 2026-07-28 | 拜耳公司 | 包含氟吡呋喃酮的液体农用化学制剂 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH503722A (de) | 1969-05-28 | 1971-02-28 | Lonza Ag | Verfahren zur Herstellung von Tetronsäure |
| DE3311003A1 (de) | 1983-03-25 | 1984-09-27 | Bayer Ag, 5090 Leverkusen | Chromon- und thiochromonsubstituierte 1,4-dihydropyridinlactone, mehrere verfahren zu ihrer herstellung und ihre verwendung in arzneimitteln |
| CH658056A5 (de) | 1984-02-09 | 1986-10-15 | Lonza Ag | Verfahren zur herstellung von tetronsaeure. |
| US5010176A (en) | 1988-11-10 | 1991-04-23 | Eli Lilly And Company | Antibody-drug conjugates |
| WO1992000964A1 (fr) * | 1990-07-05 | 1992-01-23 | Nippon Soda Co., Ltd. | Derive d'amine |
| JPH054966A (ja) * | 1990-07-05 | 1993-01-14 | Nippon Soda Co Ltd | アミン誘導体、その製法及び殺虫剤 |
| DE102006015470A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
| DE102006015467A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
| DE102006015468A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
| CN1974532B (zh) * | 2006-12-13 | 2010-12-29 | 井冈山学院 | 羧酸二异丙基二乙基酯的制备方法及其应用 |
-
2007
- 2007-09-18 EP EP07116639A patent/EP2042496A1/de not_active Ceased
-
2008
- 2008-09-05 JP JP2010525229A patent/JP5611043B2/ja active Active
- 2008-09-05 CN CN200880107465XA patent/CN101801948B/zh active Active
- 2008-09-05 WO PCT/EP2008/007270 patent/WO2009036899A1/de not_active Ceased
- 2008-09-05 KR KR1020107007178A patent/KR101516606B1/ko active Active
- 2008-09-05 EP EP08801865.0A patent/EP2193128B1/de active Active
- 2008-09-05 MX MX2010001963A patent/MX2010001963A/es active IP Right Grant
- 2008-09-05 US US12/677,769 patent/US8273904B2/en active Active
- 2008-09-05 BR BRPI0816911-0A patent/BRPI0816911B1/pt active IP Right Grant
- 2008-09-05 CN CN2012102326181A patent/CN102775305A/zh active Pending
- 2008-09-05 DK DK08801865.0T patent/DK2193128T3/en active
- 2008-09-05 ES ES08801865.0T patent/ES2612058T3/es active Active
- 2008-09-17 TW TW097135546A patent/TWI432419B/zh active
-
2010
- 2010-02-07 IL IL203761A patent/IL203761A/en active IP Right Grant
-
2012
- 2012-08-22 US US13/591,431 patent/US9550745B2/en active Active
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