CN102775305A - 4-氨基丁-2-烯羟酸内酯的制备方法 - Google Patents
4-氨基丁-2-烯羟酸内酯的制备方法 Download PDFInfo
- Publication number
- CN102775305A CN102775305A CN2012102326181A CN201210232618A CN102775305A CN 102775305 A CN102775305 A CN 102775305A CN 2012102326181 A CN2012102326181 A CN 2012102326181A CN 201210232618 A CN201210232618 A CN 201210232618A CN 102775305 A CN102775305 A CN 102775305A
- Authority
- CN
- China
- Prior art keywords
- general formula
- base
- methyl
- compound
- acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 0 *N(CN)C(CO1)=CC1=O Chemical compound *N(CN)C(CO1)=CC1=O 0.000 description 3
- WTBIKLPLFXJWHV-UHFFFAOYSA-N CCNC(CNI)=C Chemical compound CCNC(CNI)=C WTBIKLPLFXJWHV-UHFFFAOYSA-N 0.000 description 1
- JCGNDDUYTRNOFT-UHFFFAOYSA-N O=C(C1)COC1=O Chemical compound O=C(C1)COC1=O JCGNDDUYTRNOFT-UHFFFAOYSA-N 0.000 description 1
- FUDDLSHBRSNCBV-UHFFFAOYSA-N OC(C1)COC1=O Chemical compound OC(C1)COC1=O FUDDLSHBRSNCBV-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07116639A EP2042496A1 (de) | 2007-09-18 | 2007-09-18 | Verfahren zur Herstellung von 4-Aminobut-2-enoliden |
| EP07116639.1 | 2007-09-18 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN200880107465XA Division CN101801948B (zh) | 2007-09-18 | 2008-09-05 | 4-氨基丁-2-烯羟酸内酯的制备方法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN102775305A true CN102775305A (zh) | 2012-11-14 |
Family
ID=39167552
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN200880107465XA Active CN101801948B (zh) | 2007-09-18 | 2008-09-05 | 4-氨基丁-2-烯羟酸内酯的制备方法 |
| CN2012102326181A Pending CN102775305A (zh) | 2007-09-18 | 2008-09-05 | 4-氨基丁-2-烯羟酸内酯的制备方法 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN200880107465XA Active CN101801948B (zh) | 2007-09-18 | 2008-09-05 | 4-氨基丁-2-烯羟酸内酯的制备方法 |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US8273904B2 (enExample) |
| EP (2) | EP2042496A1 (enExample) |
| JP (1) | JP5611043B2 (enExample) |
| KR (1) | KR101516606B1 (enExample) |
| CN (2) | CN101801948B (enExample) |
| BR (1) | BRPI0816911B1 (enExample) |
| DK (1) | DK2193128T3 (enExample) |
| ES (1) | ES2612058T3 (enExample) |
| IL (1) | IL203761A (enExample) |
| MX (1) | MX2010001963A (enExample) |
| TW (1) | TWI432419B (enExample) |
| WO (1) | WO2009036899A1 (enExample) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2230236A1 (de) | 2009-03-16 | 2010-09-22 | Bayer CropScience AG | Neues Verfahren zur Herstellung von Enaminocarbonyl-Verbindungen |
| EP2230237A1 (de) | 2009-03-16 | 2010-09-22 | Bayer CropScience AG | Neues Verfahren zur Herstellung von Enaminocarbonyl-Verbindungen |
| BR112012002871B1 (pt) * | 2009-08-11 | 2017-04-18 | Bayer Cropscience Ag | método para fabricação de 2,4-dióxo-tetrahidrofurano-3-carboxilatos |
| TW201111370A (en) * | 2009-08-18 | 2011-04-01 | Bayer Cropscience Ag | Novel process for the preparation of 4-aminobut-2-enolides |
| BR112012009808A2 (pt) | 2009-10-26 | 2015-09-29 | Bayer Cropscience Ag | nova forma sólida de 4-[[(6-cloropiridin - 3-il)metil]2,2-difluoroetil)amino] furan-2(5h)-ona |
| US20120283294A1 (en) | 2009-10-27 | 2012-11-08 | Bayer Technology Services Gmbh | Co-crystal of 4-furan-2(5h)-one with benzoic acid and use thereof as pesticide |
| EP2493884A1 (de) * | 2009-10-27 | 2012-09-05 | Bayer Technology Services GmbH | Co-kristall von 4- { [ (6-chlorpyrid-3-yl) methyl](2,2-difluorethyl) amino} furan-2 (5h) -on mit salizylsäure und dessen verwendung als pestizid |
| CN102712631A (zh) * | 2009-10-27 | 2012-10-03 | 拜尔技术服务有限责任公司 | 4-{[(6-氯吡啶-3-基)甲基](2,2-二氟乙基)-氨基}呋喃-2(5h)-酮与草酸的共结晶及其作为杀虫剂的用途 |
| ES2602028T3 (es) * | 2009-12-23 | 2017-02-17 | Bayer Intellectual Property Gmbh | Nuevo procedimiento para la preparación de 4-aminobut-2-enólidos partiendo de 4-alcoxifuran-2(5H)-ona o 4-arilalcoxifuran-2-(5H)-ona |
| US20130331417A1 (en) * | 2010-12-09 | 2013-12-12 | Bayer Intellectual Property Gmbh | Insecticidal mixtures with improved properties |
| EP2648515A1 (en) * | 2010-12-09 | 2013-10-16 | Bayer Intellectual Property GmbH | Pesticidal mixtures with improved properties |
| US9056848B2 (en) | 2011-03-03 | 2015-06-16 | Bayer Intellectual Property Gmbh | Process for preparing sodium salts or potassium salts of 4-hydroxy-2-oxo-2,5-dihydrofuran-3-carboxylate |
| CN104507920B (zh) * | 2012-08-01 | 2018-01-05 | 拜耳农作物科学股份公司 | 用于制备特定的4‑羟基‑2‑氧代‑2,5‑二氢呋喃‑3‑甲酸酯的碱金属盐的多步法 |
| CN105503708B (zh) * | 2016-01-26 | 2018-05-29 | 南开大学 | 一类含二氟乙基的杂环化合物及其制备方法和用途 |
| EP4295683A1 (en) | 2022-06-21 | 2023-12-27 | Bayer Aktiengesellschaft | Agrochemical formulations comprising crystalline form a of 4-[(6-chloro-3-pyridylmethyl)(2,2-difluoroethyl)amino]furan-2(5h)-one |
| KR20250020435A (ko) | 2022-06-06 | 2025-02-11 | 바이엘 악티엔게젤샤프트 | 4-[(6-클로로-3-피리딜메틸)(2,2-디플루오로에틸)아미노]푸란-2(5h)-온의결정질 형태 a를 포함하는 농약 제제 |
| WO2025114238A1 (en) | 2023-12-01 | 2025-06-05 | Bayer Aktiengesellschaft | Solid agrochemical formulations comprising crystalline form a of 4-[(6-chloro-3-pyridylmethyl)(2,2- difluoroethyl)amino]furan-2(5h)-one |
| WO2025119860A1 (en) | 2023-12-05 | 2025-06-12 | Bayer Aktiengesellschaft | Liquid agrochemical formulations comprising flupyradifurone |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0539588A1 (en) * | 1990-07-05 | 1993-05-05 | Nippon Soda Co., Ltd. | Amine derivative |
| CN1974532A (zh) * | 2006-12-13 | 2007-06-06 | 井冈山学院 | 羧酸二异丙基二乙基酯的制备方法及其应用 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH503722A (de) | 1969-05-28 | 1971-02-28 | Lonza Ag | Verfahren zur Herstellung von Tetronsäure |
| DE3311003A1 (de) | 1983-03-25 | 1984-09-27 | Bayer Ag, 5090 Leverkusen | Chromon- und thiochromonsubstituierte 1,4-dihydropyridinlactone, mehrere verfahren zu ihrer herstellung und ihre verwendung in arzneimitteln |
| CH658056A5 (de) | 1984-02-09 | 1986-10-15 | Lonza Ag | Verfahren zur herstellung von tetronsaeure. |
| US5010176A (en) | 1988-11-10 | 1991-04-23 | Eli Lilly And Company | Antibody-drug conjugates |
| JPH054966A (ja) * | 1990-07-05 | 1993-01-14 | Nippon Soda Co Ltd | アミン誘導体、その製法及び殺虫剤 |
| DE102006015470A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
| DE102006015467A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
| DE102006015468A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
-
2007
- 2007-09-18 EP EP07116639A patent/EP2042496A1/de not_active Ceased
-
2008
- 2008-09-05 KR KR1020107007178A patent/KR101516606B1/ko active Active
- 2008-09-05 EP EP08801865.0A patent/EP2193128B1/de active Active
- 2008-09-05 CN CN200880107465XA patent/CN101801948B/zh active Active
- 2008-09-05 CN CN2012102326181A patent/CN102775305A/zh active Pending
- 2008-09-05 MX MX2010001963A patent/MX2010001963A/es active IP Right Grant
- 2008-09-05 WO PCT/EP2008/007270 patent/WO2009036899A1/de not_active Ceased
- 2008-09-05 BR BRPI0816911-0A patent/BRPI0816911B1/pt active IP Right Grant
- 2008-09-05 JP JP2010525229A patent/JP5611043B2/ja active Active
- 2008-09-05 ES ES08801865.0T patent/ES2612058T3/es active Active
- 2008-09-05 DK DK08801865.0T patent/DK2193128T3/en active
- 2008-09-05 US US12/677,769 patent/US8273904B2/en active Active
- 2008-09-17 TW TW097135546A patent/TWI432419B/zh active
-
2010
- 2010-02-07 IL IL203761A patent/IL203761A/en active IP Right Grant
-
2012
- 2012-08-22 US US13/591,431 patent/US9550745B2/en active Active
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0539588A1 (en) * | 1990-07-05 | 1993-05-05 | Nippon Soda Co., Ltd. | Amine derivative |
| CN1974532A (zh) * | 2006-12-13 | 2007-06-06 | 井冈山学院 | 羧酸二异丙基二乙基酯的制备方法及其应用 |
Non-Patent Citations (1)
| Title |
|---|
| T.P.C.MULHOLLAND: "A SYNTHESIS OF TETRONIC ACID [FURAN-2(3H),4(5H)-DIONE] AND THREE ANALOGUES", 《J.C.S.PERKIN I》 * |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2009036899A1 (de) | 2009-03-26 |
| US20100190990A1 (en) | 2010-07-29 |
| CN101801948A (zh) | 2010-08-11 |
| TWI432419B (zh) | 2014-04-01 |
| EP2042496A1 (de) | 2009-04-01 |
| EP2193128B1 (de) | 2016-10-26 |
| BRPI0816911A2 (pt) | 2015-03-17 |
| ES2612058T3 (es) | 2017-05-11 |
| JP2011500513A (ja) | 2011-01-06 |
| TW200920741A (en) | 2009-05-16 |
| IL203761A (en) | 2015-09-24 |
| BRPI0816911A8 (pt) | 2015-10-27 |
| KR20100061826A (ko) | 2010-06-09 |
| DK2193128T3 (en) | 2017-01-30 |
| KR101516606B1 (ko) | 2015-04-30 |
| EP2193128A1 (de) | 2010-06-09 |
| US9550745B2 (en) | 2017-01-24 |
| CN101801948B (zh) | 2013-10-30 |
| JP5611043B2 (ja) | 2014-10-22 |
| US8273904B2 (en) | 2012-09-25 |
| BRPI0816911B1 (pt) | 2022-04-12 |
| MX2010001963A (es) | 2010-03-10 |
| US20120323023A1 (en) | 2012-12-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| C06 | Publication | ||
| PB01 | Publication | ||
| C10 | Entry into substantive examination | ||
| SE01 | Entry into force of request for substantive examination | ||
| C12 | Rejection of a patent application after its publication | ||
| RJ01 | Rejection of invention patent application after publication |
Application publication date: 20121114 |