BR112012009808A2 - nova forma sólida de 4-[[(6-cloropiridin - 3-il)metil]2,2-difluoroetil)amino] furan-2(5h)-ona - Google Patents
nova forma sólida de 4-[[(6-cloropiridin - 3-il)metil]2,2-difluoroetil)amino] furan-2(5h)-onaInfo
- Publication number
- BR112012009808A2 BR112012009808A2 BR112012009808A BR112012009808A BR112012009808A2 BR 112012009808 A2 BR112012009808 A2 BR 112012009808A2 BR 112012009808 A BR112012009808 A BR 112012009808A BR 112012009808 A BR112012009808 A BR 112012009808A BR 112012009808 A2 BR112012009808 A2 BR 112012009808A2
- Authority
- BR
- Brazil
- Prior art keywords
- chloropyridin
- difluoroethyl
- furan
- amino
- methyl
- Prior art date
Links
- -1 6-chloropyridin-3-yl Chemical group 0.000 title abstract 3
- VIHAEDVKXSOUAT-UHFFFAOYSA-N but-2-en-4-olide Chemical compound O=C1OCC=C1 VIHAEDVKXSOUAT-UHFFFAOYSA-N 0.000 title abstract 3
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 title abstract 3
- 239000007787 solid Substances 0.000 title abstract 3
- 125000004778 2,2-difluoroethyl group Chemical group [H]C([H])(*)C([H])(F)F 0.000 title abstract 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 title abstract 2
- 239000003905 agrochemical Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
- A01N43/04—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
- A01N43/06—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings
- A01N43/08—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings with oxygen as the ring hetero atom
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Dentistry (AREA)
- Agronomy & Crop Science (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- Engineering & Computer Science (AREA)
- Plant Pathology (AREA)
- Veterinary Medicine (AREA)
- Pest Control & Pesticides (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
nova forma sólida de 4-[[(6-cloropiridin - 3-il)metil]2,2-difluoroetil)amino] furan-2(5h)-ona a presente invenção refere-se a uma nova forma sólida de 4-[[(6-cloropiridin-3-il)metil]2,2-difluoroetil)amino]furan-2(5h)-ona, método para a fabricação destas e utilização das mesmas em preparações agroquímicas.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP09174046 | 2009-10-26 | ||
US25560009P | 2009-10-28 | 2009-10-28 | |
PCT/EP2010/065807 WO2011051151A1 (de) | 2009-10-26 | 2010-10-20 | Neue feste form von 4-[[(6-chlorpyridin-3-yl)methyl](2,2-difluorethyl)amino]furan-2(5h)-on |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112012009808A2 true BR112012009808A2 (pt) | 2015-09-29 |
Family
ID=41571314
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112012009808A BR112012009808A2 (pt) | 2009-10-26 | 2010-10-20 | nova forma sólida de 4-[[(6-cloropiridin - 3-il)metil]2,2-difluoroetil)amino] furan-2(5h)-ona |
Country Status (9)
Country | Link |
---|---|
US (2) | US8324392B2 (pt) |
EP (1) | EP2493881A1 (pt) |
JP (1) | JP2013508339A (pt) |
KR (1) | KR20120102060A (pt) |
CN (1) | CN102741244A (pt) |
BR (1) | BR112012009808A2 (pt) |
IL (1) | IL219013A0 (pt) |
MX (1) | MX2012004796A (pt) |
WO (1) | WO2011051151A1 (pt) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ703965A (en) * | 2012-08-03 | 2016-08-26 | Bayer Cropscience Ag | Composition comprising a pesticidal terpene mixture and a fungicide |
CN106561662A (zh) * | 2016-11-17 | 2017-04-19 | 佛山市盈辉作物科学有限公司 | 一种抗病杀虫复配种子处理剂 |
EP4295683A1 (en) | 2022-06-21 | 2023-12-27 | Bayer Aktiengesellschaft | Agrochemical formulations comprising crystalline form a of 4-[(6-chloro-3-pyridylmethyl)(2,2-difluoroethyl)amino]furan-2(5h)-one |
WO2023237444A1 (en) | 2022-06-06 | 2023-12-14 | Bayer Aktiengesellschaft | Agrochemical formulations comprising crystalline form a of 4-[(6-chloro-3-pyridylmethyl)(2,2-difluoroethyl)amino]furan-2(5h)-one |
Family Cites Families (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4272417A (en) | 1979-05-22 | 1981-06-09 | Cargill, Incorporated | Stable protective seed coating |
US4245432A (en) | 1979-07-25 | 1981-01-20 | Eastman Kodak Company | Seed coatings |
US4808430A (en) | 1987-02-27 | 1989-02-28 | Yazaki Corporation | Method of applying gel coating to plant seeds |
EP0539588A1 (en) | 1990-07-05 | 1993-05-05 | Nippon Soda Co., Ltd. | Amine derivative |
US5876739A (en) | 1996-06-13 | 1999-03-02 | Novartis Ag | Insecticidal seed coating |
EP1076053B1 (en) | 1998-04-27 | 2006-11-29 | Kumiai Chemical Industry Co., Ltd. | 3-arylphenyl sulfide derivatives and insecticides and miticides |
US6503904B2 (en) | 1998-11-16 | 2003-01-07 | Syngenta Crop Protection, Inc. | Pesticidal composition for seed treatment |
US6410583B1 (en) | 2000-07-25 | 2002-06-25 | Merck Frosst Canada & Co. | Cyclopentanoindoles, compositions containing such compounds and methods of treatment |
DE10119423A1 (de) | 2001-04-20 | 2002-10-24 | Bayer Ag | Neue insektizid wirkende Azole |
US6453683B1 (en) | 2001-05-22 | 2002-09-24 | Integrated Biosystems, Inc. | Tapered slot cryopreservation system with controlled dendritic freezing front velocity |
DE102004047922A1 (de) | 2004-10-01 | 2006-04-06 | Bayer Cropscience Ag | Wirkstoffe für die Saatgutbehandlung |
DE102005008021A1 (de) | 2005-02-22 | 2006-08-24 | Bayer Cropscience Ag | Spiroketal-substituierte cyclische Ketoenole |
DE602006007590D1 (de) | 2005-07-29 | 2009-08-13 | Basf Se | Cyanopyridinpestizide |
TWI398433B (zh) | 2006-02-10 | 2013-06-11 | Dow Agrosciences Llc | 殺蟲性之n-取代(6-鹵烷基吡啶-3-基)烷基磺醯亞胺 |
DE102006015467A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
DE102006015468A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
DE102006015470A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
TWI381811B (zh) | 2006-06-23 | 2013-01-11 | Dow Agrosciences Llc | 用以防治可抵抗一般殺蟲劑之昆蟲的方法 |
ATE439564T1 (de) | 2006-06-30 | 2009-08-15 | Saab Ab | Abfeueranordnung zum abschiessen von gegenmassnahmemitteln |
DE102007018452A1 (de) * | 2007-04-17 | 2008-10-23 | Bayer Cropscience Ag | Verfahren zur verbesserten Nutzung des Produktionspotentials transgener Pflanzen |
US7950222B2 (en) * | 2007-07-27 | 2011-05-31 | Cummins, Inc. | System and method for cleaning combustion soot from exhaust gas treatment sensors |
EP2042496A1 (de) | 2007-09-18 | 2009-04-01 | Bayer CropScience AG | Verfahren zur Herstellung von 4-Aminobut-2-enoliden |
EP2230236A1 (de) * | 2009-03-16 | 2010-09-22 | Bayer CropScience AG | Neues Verfahren zur Herstellung von Enaminocarbonyl-Verbindungen |
EP2230237A1 (de) * | 2009-03-16 | 2010-09-22 | Bayer CropScience AG | Neues Verfahren zur Herstellung von Enaminocarbonyl-Verbindungen |
US8566593B2 (en) | 2009-07-06 | 2013-10-22 | Intel Corporation | Method and apparatus of deriving security key(s) |
-
2010
- 2010-10-20 WO PCT/EP2010/065807 patent/WO2011051151A1/de active Application Filing
- 2010-10-20 JP JP2012534688A patent/JP2013508339A/ja active Pending
- 2010-10-20 KR KR1020127013332A patent/KR20120102060A/ko not_active Application Discontinuation
- 2010-10-20 CN CN2010800484512A patent/CN102741244A/zh active Pending
- 2010-10-20 MX MX2012004796A patent/MX2012004796A/es not_active Application Discontinuation
- 2010-10-20 EP EP10766065A patent/EP2493881A1/de not_active Withdrawn
- 2010-10-20 BR BR112012009808A patent/BR112012009808A2/pt not_active Application Discontinuation
- 2010-10-22 US US12/910,201 patent/US8324392B2/en not_active Expired - Fee Related
-
2012
- 2012-04-03 IL IL219013A patent/IL219013A0/en unknown
- 2012-10-31 US US13/665,001 patent/US8476448B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
MX2012004796A (es) | 2012-06-08 |
US8476448B2 (en) | 2013-07-02 |
CN102741244A (zh) | 2012-10-17 |
EP2493881A1 (de) | 2012-09-05 |
KR20120102060A (ko) | 2012-09-17 |
IL219013A0 (en) | 2012-06-28 |
US20130059731A1 (en) | 2013-03-07 |
US20110130288A1 (en) | 2011-06-02 |
JP2013508339A (ja) | 2013-03-07 |
US8324392B2 (en) | 2012-12-04 |
WO2011051151A1 (de) | 2011-05-05 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B11E | Dismissal acc. art. 34 of ipl - requirements for examination incomplete | ||
B11T | Dismissal of application maintained [chapter 11.20 patent gazette] |