CN101801948B - 4-氨基丁-2-烯羟酸内酯的制备方法 - Google Patents
4-氨基丁-2-烯羟酸内酯的制备方法 Download PDFInfo
- Publication number
- CN101801948B CN101801948B CN200880107465XA CN200880107465A CN101801948B CN 101801948 B CN101801948 B CN 101801948B CN 200880107465X A CN200880107465X A CN 200880107465XA CN 200880107465 A CN200880107465 A CN 200880107465A CN 101801948 B CN101801948 B CN 101801948B
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- CN
- China
- Prior art keywords
- alkyl
- general formula
- compound
- group
- chlorine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Links
- 0 *C(C(C(OC1)=O)=C1N=O)=O Chemical compound *C(C(C(OC1)=O)=C1N=O)=O 0.000 description 3
- NXSHHTJWIOPOBF-UHFFFAOYSA-N CCOC(C(C(OC1)=O)=C1O)=O Chemical compound CCOC(C(C(OC1)=O)=C1O)=O NXSHHTJWIOPOBF-UHFFFAOYSA-N 0.000 description 2
- JCGNDDUYTRNOFT-UHFFFAOYSA-N O=C(C1)COC1=O Chemical compound O=C(C1)COC1=O JCGNDDUYTRNOFT-UHFFFAOYSA-N 0.000 description 1
- XNGNCFNYBYDSQH-UHFFFAOYSA-N OC(C(C(OC1)=O)=C1O)=O Chemical compound OC(C(C(OC1)=O)=C1O)=O XNGNCFNYBYDSQH-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07116639A EP2042496A1 (de) | 2007-09-18 | 2007-09-18 | Verfahren zur Herstellung von 4-Aminobut-2-enoliden |
| EP07116639.1 | 2007-09-18 | ||
| PCT/EP2008/007270 WO2009036899A1 (de) | 2007-09-18 | 2008-09-05 | Verfahren zur herstellung von 4-aminobut-2-enoliden |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN2012102326181A Division CN102775305A (zh) | 2007-09-18 | 2008-09-05 | 4-氨基丁-2-烯羟酸内酯的制备方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN101801948A CN101801948A (zh) | 2010-08-11 |
| CN101801948B true CN101801948B (zh) | 2013-10-30 |
Family
ID=39167552
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN200880107465XA Active CN101801948B (zh) | 2007-09-18 | 2008-09-05 | 4-氨基丁-2-烯羟酸内酯的制备方法 |
| CN2012102326181A Pending CN102775305A (zh) | 2007-09-18 | 2008-09-05 | 4-氨基丁-2-烯羟酸内酯的制备方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN2012102326181A Pending CN102775305A (zh) | 2007-09-18 | 2008-09-05 | 4-氨基丁-2-烯羟酸内酯的制备方法 |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US8273904B2 (enExample) |
| EP (2) | EP2042496A1 (enExample) |
| JP (1) | JP5611043B2 (enExample) |
| KR (1) | KR101516606B1 (enExample) |
| CN (2) | CN101801948B (enExample) |
| BR (1) | BRPI0816911B1 (enExample) |
| DK (1) | DK2193128T3 (enExample) |
| ES (1) | ES2612058T3 (enExample) |
| IL (1) | IL203761A (enExample) |
| MX (1) | MX2010001963A (enExample) |
| TW (1) | TWI432419B (enExample) |
| WO (1) | WO2009036899A1 (enExample) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2230237A1 (de) | 2009-03-16 | 2010-09-22 | Bayer CropScience AG | Neues Verfahren zur Herstellung von Enaminocarbonyl-Verbindungen |
| EP2230236A1 (de) | 2009-03-16 | 2010-09-22 | Bayer CropScience AG | Neues Verfahren zur Herstellung von Enaminocarbonyl-Verbindungen |
| MX2012001675A (es) * | 2009-08-11 | 2012-03-06 | Bayer Cropscience Ag | Procedimiento para preparar 2,4-dioxotetrahidrofuran-3-carboxilato s. |
| TW201111370A (en) * | 2009-08-18 | 2011-04-01 | Bayer Cropscience Ag | Novel process for the preparation of 4-aminobut-2-enolides |
| CN102741244A (zh) | 2009-10-26 | 2012-10-17 | 拜耳作物科学公司 | 4-[[(6-氯吡啶-3-基)甲基](2,2-二氟乙基)氨基]呋喃-2(5h)-酮的新固体形式 |
| WO2011051242A1 (de) | 2009-10-27 | 2011-05-05 | Bayer Technology Services Gmbh | Co-kristall von 4- { [ (6-chlorpyrid-3-yl) methyl] (2,2-difluorethyl) amino} furan-2 (5h) -on mit salizylsäure und dessen verwendung als pestizid |
| US20120270904A1 (en) * | 2009-10-27 | 2012-10-25 | Bayer Technology Services Gmbh | Co-crystal of 4-furan-2(5h)-one with oxalic acid and use thereof as pesticide |
| US20120283294A1 (en) | 2009-10-27 | 2012-11-08 | Bayer Technology Services Gmbh | Co-crystal of 4-furan-2(5h)-one with benzoic acid and use thereof as pesticide |
| DK2516421T3 (en) * | 2009-12-23 | 2016-11-28 | Bayer Ip Gmbh | New process for the preparation of 4-aminobut-2-enoliden starting from 4-alkoxyfuran-2 (5H) -one or 4-arylalkoxyfuran-2- (5H) -one |
| US20130331417A1 (en) * | 2010-12-09 | 2013-12-12 | Bayer Intellectual Property Gmbh | Insecticidal mixtures with improved properties |
| EP2648515A1 (en) * | 2010-12-09 | 2013-10-16 | Bayer Intellectual Property GmbH | Pesticidal mixtures with improved properties |
| JP5970002B2 (ja) * | 2011-03-03 | 2016-08-17 | バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH | 4−ヒドロキシ−2−オキソ−2,5−ジヒドロフラン−3−カルボン酸化合物のナトリウム塩またはカリウム塩の製造方法 |
| KR101977919B1 (ko) * | 2012-08-01 | 2019-05-13 | 바이엘 크롭사이언스 악티엔게젤샤프트 | 특정 4-하이드록시-2-옥소-2,5-디하이드로푸란-3-카복실산 에스테르의 알칼리 금속 염의 다단 제조방법 |
| CN105503708B (zh) * | 2016-01-26 | 2018-05-29 | 南开大学 | 一类含二氟乙基的杂环化合物及其制备方法和用途 |
| EP4295683A1 (en) | 2022-06-21 | 2023-12-27 | Bayer Aktiengesellschaft | Agrochemical formulations comprising crystalline form a of 4-[(6-chloro-3-pyridylmethyl)(2,2-difluoroethyl)amino]furan-2(5h)-one |
| KR20250020435A (ko) | 2022-06-06 | 2025-02-11 | 바이엘 악티엔게젤샤프트 | 4-[(6-클로로-3-피리딜메틸)(2,2-디플루오로에틸)아미노]푸란-2(5h)-온의결정질 형태 a를 포함하는 농약 제제 |
| WO2025114238A1 (en) | 2023-12-01 | 2025-06-05 | Bayer Aktiengesellschaft | Solid agrochemical formulations comprising crystalline form a of 4-[(6-chloro-3-pyridylmethyl)(2,2- difluoroethyl)amino]furan-2(5h)-one |
| CN122476959A (zh) | 2023-12-05 | 2026-07-28 | 拜耳公司 | 包含氟吡呋喃酮的液体农用化学制剂 |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0539588A1 (en) * | 1990-07-05 | 1993-05-05 | Nippon Soda Co., Ltd. | Amine derivative |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH503722A (de) | 1969-05-28 | 1971-02-28 | Lonza Ag | Verfahren zur Herstellung von Tetronsäure |
| DE3311003A1 (de) | 1983-03-25 | 1984-09-27 | Bayer Ag, 5090 Leverkusen | Chromon- und thiochromonsubstituierte 1,4-dihydropyridinlactone, mehrere verfahren zu ihrer herstellung und ihre verwendung in arzneimitteln |
| CH658056A5 (de) | 1984-02-09 | 1986-10-15 | Lonza Ag | Verfahren zur herstellung von tetronsaeure. |
| US5010176A (en) | 1988-11-10 | 1991-04-23 | Eli Lilly And Company | Antibody-drug conjugates |
| JPH054966A (ja) * | 1990-07-05 | 1993-01-14 | Nippon Soda Co Ltd | アミン誘導体、その製法及び殺虫剤 |
| DE102006015470A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
| DE102006015467A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
| DE102006015468A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
| CN1974532B (zh) * | 2006-12-13 | 2010-12-29 | 井冈山学院 | 羧酸二异丙基二乙基酯的制备方法及其应用 |
-
2007
- 2007-09-18 EP EP07116639A patent/EP2042496A1/de not_active Ceased
-
2008
- 2008-09-05 JP JP2010525229A patent/JP5611043B2/ja active Active
- 2008-09-05 CN CN200880107465XA patent/CN101801948B/zh active Active
- 2008-09-05 WO PCT/EP2008/007270 patent/WO2009036899A1/de not_active Ceased
- 2008-09-05 KR KR1020107007178A patent/KR101516606B1/ko active Active
- 2008-09-05 EP EP08801865.0A patent/EP2193128B1/de active Active
- 2008-09-05 MX MX2010001963A patent/MX2010001963A/es active IP Right Grant
- 2008-09-05 US US12/677,769 patent/US8273904B2/en active Active
- 2008-09-05 BR BRPI0816911-0A patent/BRPI0816911B1/pt active IP Right Grant
- 2008-09-05 CN CN2012102326181A patent/CN102775305A/zh active Pending
- 2008-09-05 DK DK08801865.0T patent/DK2193128T3/en active
- 2008-09-05 ES ES08801865.0T patent/ES2612058T3/es active Active
- 2008-09-17 TW TW097135546A patent/TWI432419B/zh active
-
2010
- 2010-02-07 IL IL203761A patent/IL203761A/en active IP Right Grant
-
2012
- 2012-08-22 US US13/591,431 patent/US9550745B2/en active Active
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0539588A1 (en) * | 1990-07-05 | 1993-05-05 | Nippon Soda Co., Ltd. | Amine derivative |
Non-Patent Citations (3)
| Title |
|---|
| Alexander C. Campbell, et al..Synthesis of (E)- and (Z)-Pulvinones.《J. CHEM. SOC. PERKIN TRANS. I》.RSC,1985,(第9-10期),第1567-1576页. * |
| T. P. C. Mulholland, et al..A Synthesis of Tetronic Acid [Furan-2(3H),4(5H)-dione] and Three Analogues.《J. CHEM. SOC. PERKIN TRANS. I》.RSC,1972,第1卷第1225-1231页. * |
| T.P.C.Mulholland et al..A Synthesis of Tetronic Acid [Furan-2(3H) |
Also Published As
| Publication number | Publication date |
|---|---|
| JP5611043B2 (ja) | 2014-10-22 |
| US9550745B2 (en) | 2017-01-24 |
| BRPI0816911A8 (pt) | 2015-10-27 |
| US20100190990A1 (en) | 2010-07-29 |
| KR101516606B1 (ko) | 2015-04-30 |
| MX2010001963A (es) | 2010-03-10 |
| EP2042496A1 (de) | 2009-04-01 |
| IL203761A (en) | 2015-09-24 |
| TW200920741A (en) | 2009-05-16 |
| EP2193128B1 (de) | 2016-10-26 |
| US8273904B2 (en) | 2012-09-25 |
| BRPI0816911A2 (pt) | 2015-03-17 |
| EP2193128A1 (de) | 2010-06-09 |
| CN102775305A (zh) | 2012-11-14 |
| ES2612058T3 (es) | 2017-05-11 |
| BRPI0816911B1 (pt) | 2022-04-12 |
| CN101801948A (zh) | 2010-08-11 |
| KR20100061826A (ko) | 2010-06-09 |
| US20120323023A1 (en) | 2012-12-20 |
| WO2009036899A1 (de) | 2009-03-26 |
| JP2011500513A (ja) | 2011-01-06 |
| TWI432419B (zh) | 2014-04-01 |
| DK2193128T3 (en) | 2017-01-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| C06 | Publication | ||
| PB01 | Publication | ||
| C10 | Entry into substantive examination | ||
| SE01 | Entry into force of request for substantive examination | ||
| C14 | Grant of patent or utility model | ||
| GR01 | Patent grant | ||
| ASS | Succession or assignment of patent right |
Owner name: BAYER INTELLECTUAL PROPERTY GMBH Free format text: FORMER OWNER: BAYER LANDWIRTSCHAFTLICHE KULTURPFLANZEN SCIENCE AG Effective date: 20150529 |
|
| C41 | Transfer of patent application or patent right or utility model | ||
| TR01 | Transfer of patent right |
Effective date of registration: 20150529 Address after: German Monheim Patentee after: BAYER INTELLECTUAL PROPERTY GmbH Address before: German Monheim Patentee before: BAYER CROPSCIENCE AG |
|
| CP03 | Change of name, title or address |
Address after: 50 Alfred Nobel Street, Monheim, Rhine, Germany 40789 Patentee after: BAYER INTELLECTUAL PROPERTY GmbH Address before: Germany Patentee before: BAYER INTELLECTUAL PROPERTY GmbH |
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| CP03 | Change of name, title or address | ||
| TR01 | Transfer of patent right |
Effective date of registration: 20240112 Address after: 50 Alfred Nobel Street, Monheim, Rhine, Germany 40789 Patentee after: BAYER CROPSCIENCE AG Address before: 50 Alfred Nobel Street, Monheim, Rhine, Germany 40789 Patentee before: BAYER INTELLECTUAL PROPERTY GmbH |
|
| TR01 | Transfer of patent right |