JP2010539244A5 - - Google Patents
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- Publication number
- JP2010539244A5 JP2010539244A5 JP2010525985A JP2010525985A JP2010539244A5 JP 2010539244 A5 JP2010539244 A5 JP 2010539244A5 JP 2010525985 A JP2010525985 A JP 2010525985A JP 2010525985 A JP2010525985 A JP 2010525985A JP 2010539244 A5 JP2010539244 A5 JP 2010539244A5
- Authority
- JP
- Japan
- Prior art keywords
- pain
- compound
- compound according
- acute
- composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 0 C*N(C1CC=CCCCC(C)C1)S(C)(=O)=O Chemical compound C*N(C1CC=CCCCC(C)C1)S(C)(=O)=O 0.000 description 17
- JUJWROOIHBZHMG-UHFFFAOYSA-N c1ccncc1 Chemical compound c1ccncc1 JUJWROOIHBZHMG-UHFFFAOYSA-N 0.000 description 3
- LPAGFVYQRIESJQ-UHFFFAOYSA-N C1c2ccccc2NC1 Chemical compound C1c2ccccc2NC1 LPAGFVYQRIESJQ-UHFFFAOYSA-N 0.000 description 2
- XMSNMAGPGAYJHP-UHFFFAOYSA-N CSCC1c2ccccc2NCC1 Chemical compound CSCC1c2ccccc2NCC1 XMSNMAGPGAYJHP-UHFFFAOYSA-N 0.000 description 2
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US99442307P | 2007-09-19 | 2007-09-19 | |
| PCT/US2008/076928 WO2009039328A1 (en) | 2007-09-19 | 2008-09-19 | Pyridyl sulfonamides as modulators of ion channels |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010539244A JP2010539244A (ja) | 2010-12-16 |
| JP2010539244A5 true JP2010539244A5 (https=) | 2012-11-29 |
Family
ID=40352214
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010525985A Withdrawn JP2010539244A (ja) | 2007-09-19 | 2008-09-19 | イオンチャネルのモジュレーターとしてのピリジルスルホンアミド |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7994174B2 (https=) |
| EP (1) | EP2201008A1 (https=) |
| JP (1) | JP2010539244A (https=) |
| CN (1) | CN101842372A (https=) |
| AU (1) | AU2008302205A1 (https=) |
| CA (1) | CA2699892A1 (https=) |
| MX (1) | MX2010003009A (https=) |
| NZ (1) | NZ584009A (https=) |
| WO (1) | WO2009039328A1 (https=) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7615563B2 (en) * | 2003-08-08 | 2009-11-10 | Gonzalez Iii Jesus E | Compositions useful as inhibitors of voltage-gated sodium channels |
| KR20080015102A (ko) * | 2005-05-10 | 2008-02-18 | 버텍스 파마슈티칼스 인코포레이티드 | 이온 채널 조절인자로서의 바이사이클릭 유도체 |
| ATE527251T1 (de) * | 2005-05-16 | 2011-10-15 | Vertex Pharma | Bicyclische derivate als modulatoren von ionenkanälen |
| MX2008003337A (es) * | 2005-09-09 | 2008-09-26 | Vertex Pharma | Derivados biciclicos como modulares de canales ionicos regulados por voltaje. |
| EP1948597A1 (en) * | 2005-10-21 | 2008-07-30 | Vertex Pharmaceuticals Incorporated | Derivatives for modulation of ion channels |
| NZ593074A (en) | 2005-12-21 | 2012-04-27 | Vertex Pharma | sulfonamide-pyrrolidone derivatives as Modulators of Ion Channels |
| DK2142529T3 (da) * | 2007-04-27 | 2014-02-10 | Purdue Pharma Lp | Trpv1-antagonister og anvendelser deraf |
| AU2008256937A1 (en) | 2007-05-25 | 2008-12-04 | Vertex Pharmaceuticals Incorporated | Ion channel modulators and methods of use |
| EP2231655B1 (en) | 2007-11-13 | 2011-08-31 | Vertex Pharmaceuticals Incorporated | 4(-3-(-2-(phenyl)morpholino)-2-oxopyrrolidin-1-yl)-n-(thiazol-2-yl)benzenesulfonamide derivatives and related compounds as modulators of ion channels for the treatment of pain |
| CN101910166A (zh) * | 2007-11-13 | 2010-12-08 | 沃泰克斯药物股份有限公司 | 用作钠离子通道调节剂的杂环衍生物 |
| RU2011103451A (ru) * | 2008-07-01 | 2012-08-10 | Вертекс Фармасьютикалз Инкорпорейтед (Us) | Гетероциклические производные в качестве модуляторов ионных каналов |
| EP2480531B1 (en) | 2009-09-21 | 2014-11-05 | ChemoCentryx, Inc. | Pyrrolidinone carboxamide derivatives as chemerin-r (chemr23) modulators |
| HRP20170507T1 (hr) | 2011-06-22 | 2017-06-02 | Purdue Pharma Lp | Trpv1 antagonisti uključujući dihidroksi supstituente i njihove uporabe |
| ES2602140T3 (es) | 2011-06-27 | 2017-02-17 | Newron Pharmaceuticals S.P.A. | Derivados de arilalquilaminocarboxamida fluorados |
| US10510973B2 (en) * | 2014-12-17 | 2019-12-17 | Universal Display Corporation | Color-stable organic light emitting diode stack |
| WO2020113094A1 (en) | 2018-11-30 | 2020-06-04 | Nuvation Bio Inc. | Pyrrole and pyrazole compounds and methods of use thereof |
| US12588382B2 (en) | 2019-07-29 | 2026-03-24 | Universal Display Corporation | Color stable multicolor OLED device structures |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7615356B2 (en) | 2000-07-10 | 2009-11-10 | Vertex Pharmaceuticals (San Diego) Llc | Ion channel assay methods |
| WO2004103980A1 (en) | 2003-05-21 | 2004-12-02 | Biovitrum Ab | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type i |
| US7615563B2 (en) * | 2003-08-08 | 2009-11-10 | Gonzalez Iii Jesus E | Compositions useful as inhibitors of voltage-gated sodium channels |
| US8202861B2 (en) * | 2003-08-08 | 2012-06-19 | Vertex Pharmaceuticals Incorporated | Compositions useful as inhibitors of voltage-gated sodium channels |
| JP2007261945A (ja) | 2004-04-07 | 2007-10-11 | Taisho Pharmaceut Co Ltd | チアゾール誘導体 |
| KR20080015102A (ko) * | 2005-05-10 | 2008-02-18 | 버텍스 파마슈티칼스 인코포레이티드 | 이온 채널 조절인자로서의 바이사이클릭 유도체 |
| ATE527251T1 (de) * | 2005-05-16 | 2011-10-15 | Vertex Pharma | Bicyclische derivate als modulatoren von ionenkanälen |
| GT200600196A (es) * | 2005-05-23 | 2007-01-15 | Compuestos n-formil de hidroxilamina | |
| MX2007015726A (es) * | 2005-06-09 | 2008-03-04 | Vertex Pharma | Derivados de indano como moduladores de canales ionicos. |
| MX2008003337A (es) * | 2005-09-09 | 2008-09-26 | Vertex Pharma | Derivados biciclicos como modulares de canales ionicos regulados por voltaje. |
| RU2008118350A (ru) * | 2005-10-12 | 2009-11-20 | Вертекс Фармасьютикалз Инкорпорейтед (Us) | Бифенильные производные в качестве модуляторов потенциалзависимых ионных каналов |
| EP1948597A1 (en) * | 2005-10-21 | 2008-07-30 | Vertex Pharmaceuticals Incorporated | Derivatives for modulation of ion channels |
| NZ593074A (en) * | 2005-12-21 | 2012-04-27 | Vertex Pharma | sulfonamide-pyrrolidone derivatives as Modulators of Ion Channels |
| CN101910166A (zh) * | 2007-11-13 | 2010-12-08 | 沃泰克斯药物股份有限公司 | 用作钠离子通道调节剂的杂环衍生物 |
| EP2231655B1 (en) * | 2007-11-13 | 2011-08-31 | Vertex Pharmaceuticals Incorporated | 4(-3-(-2-(phenyl)morpholino)-2-oxopyrrolidin-1-yl)-n-(thiazol-2-yl)benzenesulfonamide derivatives and related compounds as modulators of ion channels for the treatment of pain |
| RU2011103451A (ru) * | 2008-07-01 | 2012-08-10 | Вертекс Фармасьютикалз Инкорпорейтед (Us) | Гетероциклические производные в качестве модуляторов ионных каналов |
-
2008
- 2008-09-17 US US12/212,063 patent/US7994174B2/en not_active Expired - Fee Related
- 2008-09-19 EP EP08831349A patent/EP2201008A1/en not_active Withdrawn
- 2008-09-19 MX MX2010003009A patent/MX2010003009A/es active IP Right Grant
- 2008-09-19 CN CN200880113677A patent/CN101842372A/zh active Pending
- 2008-09-19 AU AU2008302205A patent/AU2008302205A1/en not_active Abandoned
- 2008-09-19 WO PCT/US2008/076928 patent/WO2009039328A1/en not_active Ceased
- 2008-09-19 JP JP2010525985A patent/JP2010539244A/ja not_active Withdrawn
- 2008-09-19 NZ NZ584009A patent/NZ584009A/en not_active IP Right Cessation
- 2008-09-19 CA CA2699892A patent/CA2699892A1/en not_active Abandoned
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