JP2010529193A - 置換ピラゾール化合物 - Google Patents
置換ピラゾール化合物 Download PDFInfo
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- JP2010529193A JP2010529193A JP2010512173A JP2010512173A JP2010529193A JP 2010529193 A JP2010529193 A JP 2010529193A JP 2010512173 A JP2010512173 A JP 2010512173A JP 2010512173 A JP2010512173 A JP 2010512173A JP 2010529193 A JP2010529193 A JP 2010529193A
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
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| JP2016523976A (ja) * | 2013-07-11 | 2016-08-12 | アジオス ファーマシューティカルズ， インコーポレイテッド | 癌の処置のためのｉｄｈ２突然変異体阻害剤としての２，４−または４，６−ジアミノピリミジン化合物 |
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| JP2004509113A (ja) * | 2000-09-15 | 2004-03-25 | バーテックス ファーマシューティカルズ インコーポレイテッド | プロテインキナーゼインヒビターとして有用なピラゾール化合物 |
| JP2007510626A (ja) * | 2003-10-17 | 2007-04-26 | アストラゼネカ アクチボラグ | 癌の治療に使用の４−（ピラゾール−３−イルアミノ）ピリミジン誘導体 |
| WO2006074057A2 (en) * | 2004-12-30 | 2006-07-13 | Exelixis, Inc. | Pyrimidine derivatives as kinase modulators and method of use |
| WO2007041358A2 (en) * | 2005-09-30 | 2007-04-12 | Miikana Therapeutics, Inc. | Substituted pyrazole compounds |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2016523976A (ja) * | 2013-07-11 | 2016-08-12 | アジオス ファーマシューティカルズ， インコーポレイテッド | 癌の処置のためのｉｄｈ２突然変異体阻害剤としての２，４−または４，６−ジアミノピリミジン化合物 |
Also Published As
| Publication number | Publication date |
|---|---|
| CA2683152A1 (en) | 2008-12-18 |
| US20090029992A1 (en) | 2009-01-29 |
| EP2166849A1 (en) | 2010-03-31 |
| WO2008154026A1 (en) | 2008-12-18 |
| EP2166849A4 (en) | 2010-09-15 |
| AU2008262291A1 (en) | 2008-12-18 |
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