JP2010520307A5 - - Google Patents

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Publication number
JP2010520307A5
JP2010520307A5 JP2009552883A JP2009552883A JP2010520307A5 JP 2010520307 A5 JP2010520307 A5 JP 2010520307A5 JP 2009552883 A JP2009552883 A JP 2009552883A JP 2009552883 A JP2009552883 A JP 2009552883A JP 2010520307 A5 JP2010520307 A5 JP 2010520307A5
Authority
JP
Japan
Prior art keywords
ylidenemethyl
thiazolidine
benzonitrile
dioxo
phenoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2009552883A
Other languages
English (en)
Japanese (ja)
Other versions
JP2010520307A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2008/056018 external-priority patent/WO2008109731A2/en
Publication of JP2010520307A publication Critical patent/JP2010520307A/ja
Publication of JP2010520307A5 publication Critical patent/JP2010520307A5/ja
Pending legal-status Critical Current

Links

JP2009552883A 2007-03-07 2008-03-06 エストロゲン関連受容体−アルファモジュレーターとしての置換フェノキシn−アルキル置換チアゾリジンジオン Pending JP2010520307A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US89345807P 2007-03-07 2007-03-07
PCT/US2008/056018 WO2008109731A2 (en) 2007-03-07 2008-03-06 Substituted phenoxy n-alkylated thiazoledinedione as estrogen related receptor-alpha modulators

Publications (2)

Publication Number Publication Date
JP2010520307A JP2010520307A (ja) 2010-06-10
JP2010520307A5 true JP2010520307A5 (cg-RX-API-DMAC7.html) 2011-03-24

Family

ID=39720674

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009552883A Pending JP2010520307A (ja) 2007-03-07 2008-03-06 エストロゲン関連受容体−アルファモジュレーターとしての置換フェノキシn−アルキル置換チアゾリジンジオン

Country Status (26)

Country Link
US (2) US8119669B2 (cg-RX-API-DMAC7.html)
EP (1) EP2132188B1 (cg-RX-API-DMAC7.html)
JP (1) JP2010520307A (cg-RX-API-DMAC7.html)
KR (1) KR20090118103A (cg-RX-API-DMAC7.html)
CN (1) CN101679326B (cg-RX-API-DMAC7.html)
AR (1) AR065656A1 (cg-RX-API-DMAC7.html)
AT (1) ATE537157T1 (cg-RX-API-DMAC7.html)
AU (1) AU2008222749A1 (cg-RX-API-DMAC7.html)
BR (1) BRPI0808662B8 (cg-RX-API-DMAC7.html)
CA (1) CA2679965A1 (cg-RX-API-DMAC7.html)
CL (1) CL2008000669A1 (cg-RX-API-DMAC7.html)
CY (1) CY1112778T1 (cg-RX-API-DMAC7.html)
DK (1) DK2132188T3 (cg-RX-API-DMAC7.html)
EA (1) EA200970838A1 (cg-RX-API-DMAC7.html)
ES (1) ES2377165T3 (cg-RX-API-DMAC7.html)
HR (1) HRP20120160T1 (cg-RX-API-DMAC7.html)
IL (1) IL200758A0 (cg-RX-API-DMAC7.html)
MX (1) MX2009009519A (cg-RX-API-DMAC7.html)
NZ (1) NZ579418A (cg-RX-API-DMAC7.html)
PL (1) PL2132188T3 (cg-RX-API-DMAC7.html)
PT (1) PT2132188E (cg-RX-API-DMAC7.html)
RS (1) RS52247B (cg-RX-API-DMAC7.html)
SI (1) SI2132188T1 (cg-RX-API-DMAC7.html)
TW (1) TW200902507A (cg-RX-API-DMAC7.html)
WO (1) WO2008109731A2 (cg-RX-API-DMAC7.html)
ZA (1) ZA200906953B (cg-RX-API-DMAC7.html)

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EP2220083B1 (en) 2007-11-14 2017-07-19 Janssen Pharmaceuticals, Inc. Imidazo[1,2-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
WO2009105621A1 (en) * 2008-02-22 2009-08-27 The Ohio State University Research Foundation Androgen receptot-ablative agents
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AU2009304293B2 (en) 2008-10-16 2012-04-26 Addex Pharma S.A. Indole and benzomorpholine derivatives as modulators of metabotropic glutamate receptors
JP5690277B2 (ja) 2008-11-28 2015-03-25 ジャンセン ファーマシューティカルズ, インコーポレイテッド. 代謝型グルタミン酸受容体の調節因子としてのインドールおよびベンゾオキサジン誘導体
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US8937060B2 (en) 2009-05-12 2015-01-20 Janssen Pharmaceuticals, Inc. 1,2,4-triazolo [4,3-A] pyridine derivatives and their use for the treatment of prevention of neurological and psychiatric disorders
KR20120035158A (ko) 2009-05-12 2012-04-13 얀센 파마슈티칼즈, 인코포레이티드 1,2,4?트리아졸로[4,3?a]피리딘 유도체 및 mGluR2 수용체의 양성 알로스테릭 조절자로서의 그의 용도
JP2011057644A (ja) * 2009-09-14 2011-03-24 Sumitomo Chemical Co Ltd 3型17β−ヒドロキシステロイドデヒドロゲナーゼを阻害するための化合物の使用およびそのための医薬組成物
JP2011057643A (ja) * 2009-09-14 2011-03-24 Sumitomo Chemical Co Ltd 3型17β−ヒドロキシステロイドデヒドロゲナーゼを阻害するための化合物の使用およびそのための医薬組成物
TW201144303A (en) 2010-02-17 2011-12-16 Janssen Pharmaceutica Nv Aminothiazolones as estrogen related receptor-α modulators
CA2814996C (en) 2010-11-08 2019-10-01 Janssen Pharmaceuticals, Inc. 1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
CN103298809B (zh) 2010-11-08 2016-08-31 杨森制药公司 1,2,4-三唑并[4,3-a]吡啶衍生物及其作为MGLUR2受体的正变构调节剂的用途
EP2643320B1 (en) 2010-11-08 2015-03-04 Janssen Pharmaceuticals, Inc. 1,2,4-TRIAZOLO[4,3-a]PYRIDINE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS
WO2012153775A1 (ja) * 2011-05-10 2012-11-15 国立大学法人神戸大学 Ras機能阻害作用を有するチオキソチアゾリジン誘導体
WO2013018929A1 (en) 2011-08-04 2013-02-07 Takeda Pharmaceutical Company Limited Nitrogen-containing heterocyclic compound
CN102949364A (zh) * 2011-08-30 2013-03-06 天津药物研究院 一种含有效成分盐酸维拉佐酮的缓释片
JP5865995B2 (ja) 2012-03-26 2016-02-17 日本ケミファ株式会社 骨・軟部に発生する巨細胞性腫瘍または軟骨肉腫の予防または治療剤
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JO3368B1 (ar) 2013-06-04 2019-03-13 Janssen Pharmaceutica Nv مركبات 6، 7- ثاني هيدرو بيرازولو [5،1-a] بيرازين- 4 (5 يد)- اون واستخدامها بصفة منظمات تفارغية سلبية لمستقبلات ميجلور 2
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JO3367B1 (ar) 2013-09-06 2019-03-13 Janssen Pharmaceutica Nv مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2
KR20160055932A (ko) 2013-09-25 2016-05-18 닛뽕 케미파 가부시키가이샤 골·연부에 발생하는 거세포성 종양, 연골육종 또는 골육종의 예방, 치료 또는 전이 예방을 위한 약제, 동맥색전술용 국소 주입제 및 인공골
HRP20191646T1 (hr) 2014-01-21 2019-12-13 Janssen Pharmaceutica Nv Kombinacije koje sadržavaju pozitivne alosteričke modulatore ili ortosteričke agoniste metabotropnog glutamatergičnog receptora podtip 2 i njihova uporaba
CN109999033B (zh) 2014-01-21 2022-12-23 詹森药业有限公司 包括代谢型谷氨酸能受体亚型2的正别构调节物或正位激动剂的组合及其用途
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