JP2010505848A - 眼内圧を低下させるための種交差性ａ３アデノシン受容体アンタゴニストの効果的送達 - Google Patents
眼内圧を低下させるための種交差性ａ３アデノシン受容体アンタゴニストの効果的送達 Download PDFInfo
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- JP2010505848A JP2010505848A JP2009531464A JP2009531464A JP2010505848A JP 2010505848 A JP2010505848 A JP 2010505848A JP 2009531464 A JP2009531464 A JP 2009531464A JP 2009531464 A JP2009531464 A JP 2009531464A JP 2010505848 A JP2010505848 A JP 2010505848A
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- mrs
- intraocular pressure
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- antagonist
- adenosine
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US85017506P | 2006-10-06 | 2006-10-06 | |
| PCT/US2007/021409 WO2008045330A2 (en) | 2006-10-06 | 2007-10-05 | Effective delivery of cross-species a3 adenosine-receptor antagonists to reduce intraocular pressure |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010505848A true JP2010505848A (ja) | 2010-02-25 |
| JP2010505848A5 JP2010505848A5 (https=) | 2010-11-25 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009531464A Pending JP2010505848A (ja) | 2006-10-06 | 2007-10-05 | 眼内圧を低下させるための種交差性ａ３アデノシン受容体アンタゴニストの効果的送達 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20090258836A1 (https=) |
| EP (1) | EP2076267A4 (https=) |
| JP (1) | JP2010505848A (https=) |
| AU (1) | AU2007307157A1 (https=) |
| BR (1) | BRPI0715318A2 (https=) |
| CA (1) | CA2665616A1 (https=) |
| MX (1) | MX2009003750A (https=) |
| WO (1) | WO2008045330A2 (https=) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2020511437A (ja) * | 2017-03-21 | 2020-04-16 | フューチャー メディスン カンパニー リミテッドＦｕｔｕｒｅ Ｍｅｄｉｃｉｎｅ Ｃｏ．， Ｌｔｄ． | アデノシン誘導体を含む緑内障の予防及び治療用薬学的組成物 |
| JP2021504494A (ja) * | 2017-11-29 | 2021-02-15 | フューチャー・メディシン・カンパニー・リミテッドＦｕｔｕｒｅ Ｍｅｄｉｃｉｎｅ Ｃｏ．， Ｌｔｄ． | アデノシン誘導体を含む網膜疾患または視神経疾患の予防及び治療用薬学的組成物 |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG182285A1 (en) | 2010-01-11 | 2012-08-30 | Inotek Pharmaceuticals Corp | Combination, kit and method of reducing intraocular pressure |
| EA201290958A1 (ru) * | 2010-03-26 | 2013-04-30 | Инотек Фармасьютикалз Корпорейшн | Способ снижения внутриглазного давления у людей с применением n6-циклопентиладенозина (cpa), производных cpa или их пролекарств |
| BR112014018413A8 (pt) | 2012-01-26 | 2017-07-11 | Inotek Pharmaceuticals Corp | Polimorfos anidros de nitrato de metila [(2r,3s,4r,5r)-5-(6-(ciclopentilamino)-9h-purin-9-il)-3,4-diidroxitetraidrofuran-2-il)] e processos de preparação do mesmo |
| CA2903114A1 (en) | 2013-03-15 | 2014-09-25 | Inotek Pharmaceuticals Corporation | Ophthalmic formulations |
| ES2578363B1 (es) | 2015-01-22 | 2017-01-31 | Palobiofarma, S.L. | Moduladores de los receptores A3 de adenosina |
| HK1254892A1 (zh) | 2016-01-14 | 2019-08-02 | 韩德株式会社 | 拮抗a3腺苷受体的化合物、其制备方法、及其医学用途 |
| ES2676535B1 (es) | 2017-01-20 | 2019-04-29 | Palobiofarma Sl | Moduladores de los receptores a3 de adenosina |
| CN109666053A (zh) * | 2017-10-16 | 2019-04-23 | 张家口华健致远生物科技有限公司 | 一种a3腺苷受体激动剂及其用途 |
| US11395597B2 (en) * | 2018-06-26 | 2022-07-26 | General Electric Company | System and method for evaluating blood flow in a vessel |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2000516910A (ja) * | 1996-01-29 | 2000-12-19 | アメリカ合衆国 | ジヒドロピリジン―、ピリジン―、ベンゾピラン―オン―およびトリアゾロキナゾリン誘導体、それらの製造およびそれらのアデノシン受容体アンタゴニストとしての用途 |
| JP2003522729A (ja) * | 1998-07-16 | 2003-07-29 | ザ トラスティーズ オヴ ザ ユニヴァーシティー オヴ ペンシルバニア | 眼内圧の低下方法 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL133680A0 (en) * | 1999-09-10 | 2001-04-30 | Can Fite Technologies Ltd | Pharmaceutical compositions comprising an adenosine receptor agonist or antagonist |
-
2007
- 2007-10-05 JP JP2009531464A patent/JP2010505848A/ja active Pending
- 2007-10-05 WO PCT/US2007/021409 patent/WO2008045330A2/en not_active Ceased
- 2007-10-05 AU AU2007307157A patent/AU2007307157A1/en not_active Abandoned
- 2007-10-05 BR BRPI0715318-0A patent/BRPI0715318A2/pt not_active IP Right Cessation
- 2007-10-05 EP EP07852549.0A patent/EP2076267A4/en not_active Withdrawn
- 2007-10-05 CA CA002665616A patent/CA2665616A1/en not_active Abandoned
- 2007-10-05 MX MX2009003750A patent/MX2009003750A/es active IP Right Grant
-
2009
- 2009-04-06 US US12/419,062 patent/US20090258836A1/en not_active Abandoned
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2000516910A (ja) * | 1996-01-29 | 2000-12-19 | アメリカ合衆国 | ジヒドロピリジン―、ピリジン―、ベンゾピラン―オン―およびトリアゾロキナゾリン誘導体、それらの製造およびそれらのアデノシン受容体アンタゴニストとしての用途 |
| JP2003522729A (ja) * | 1998-07-16 | 2003-07-29 | ザ トラスティーズ オヴ ザ ユニヴァーシティー オヴ ペンシルバニア | 眼内圧の低下方法 |
Non-Patent Citations (3)
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| JPN6012048547; Ｉｎｖｅｓｔ Ｏｐｈｔｈａｌｍｏｌ Ｖｉｓ Ｓｃｉ Ｖｏｌ．４２, 2001, ｐｐ．１８４１-６ * |
| JPN6013010323; Ｃｕｒｒ Ｅｙｅ Ｒｅｓ Ｖｏｌ．３０, 2005, ｐｐ．７４７-５４ * |
| JPN6013010325; Ｂｉｏｏｒｇ Ｍｅｄ Ｃｈｅｍ Ｌｅｔｔ Ｖｏｌ．１６, 2005, ｐｐ．５９６-６０１ * |
Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2020511437A (ja) * | 2017-03-21 | 2020-04-16 | フューチャー メディスン カンパニー リミテッドＦｕｔｕｒｅ Ｍｅｄｉｃｉｎｅ Ｃｏ．， Ｌｔｄ． | アデノシン誘導体を含む緑内障の予防及び治療用薬学的組成物 |
| US11185556B2 (en) | 2017-03-21 | 2021-11-30 | Future Medicine Co., Ltd. | Pharmaceutical composition for preventing and treating glaucoma, containing adenosine derivative |
| US12083140B2 (en) | 2017-03-21 | 2024-09-10 | Future Medicine Co., Ltd. | Pharmaceutical composition for preventing and treating glaucoma, containing adenosine derivative |
| JP2021504494A (ja) * | 2017-11-29 | 2021-02-15 | フューチャー・メディシン・カンパニー・リミテッドＦｕｔｕｒｅ Ｍｅｄｉｃｉｎｅ Ｃｏ．， Ｌｔｄ． | アデノシン誘導体を含む網膜疾患または視神経疾患の予防及び治療用薬学的組成物 |
| JP7160384B2 (ja) | 2017-11-29 | 2022-10-25 | フューチャー・メディシン・カンパニー・リミテッド | アデノシン誘導体を含む網膜疾患または視神経疾患の予防及び治療用薬学的組成物 |
| JP2023011577A (ja) * | 2017-11-29 | 2023-01-24 | フューチャー・メディシン・カンパニー・リミテッド | アデノシン誘導体を含む網膜疾患または視神経疾患の予防及び治療用薬学的組成物 |
| JP7577347B2 (ja) | 2017-11-29 | 2024-11-05 | フューチャー・メディシン・カンパニー・リミテッド | アデノシン誘導体を含む網膜疾患または視神経疾患の予防及び治療用薬学的組成物 |
Also Published As
| Publication number | Publication date |
|---|---|
| AU2007307157A1 (en) | 2008-04-17 |
| EP2076267A4 (en) | 2013-07-31 |
| BRPI0715318A2 (pt) | 2013-07-16 |
| EP2076267A2 (en) | 2009-07-08 |
| CA2665616A1 (en) | 2008-04-17 |
| WO2008045330A3 (en) | 2008-06-26 |
| WO2008045330A2 (en) | 2008-04-17 |
| MX2009003750A (es) | 2009-06-18 |
| US20090258836A1 (en) | 2009-10-15 |
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