JP2010132677A5 - - Google Patents
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- Publication number
- JP2010132677A5 JP2010132677A5 JP2010016076A JP2010016076A JP2010132677A5 JP 2010132677 A5 JP2010132677 A5 JP 2010132677A5 JP 2010016076 A JP2010016076 A JP 2010016076A JP 2010016076 A JP2010016076 A JP 2010016076A JP 2010132677 A5 JP2010132677 A5 JP 2010132677A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- oxo
- fluoro
- formula
- pdg
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IBPCT/IB2006/054189 | 2006-11-10 | ||
| IB2006054189 | 2006-11-10 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009535864A Division JP4484965B2 (ja) | 2006-11-10 | 2007-11-09 | ５−ヒドロキシメチル−オキサゾリジン−２−オン誘導体 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2010132677A JP2010132677A (ja) | 2010-06-17 |
| JP2010132677A5 true JP2010132677A5 (cg-RX-API-DMAC7.html) | 2010-12-24 |
| JP5490553B2 JP5490553B2 (ja) | 2014-05-14 |
Family
ID=39170372
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009535864A Expired - Fee Related JP4484965B2 (ja) | 2006-11-10 | 2007-11-09 | ５−ヒドロキシメチル−オキサゾリジン−２−オン誘導体 |
| JP2010016076A Expired - Fee Related JP5490553B2 (ja) | 2006-11-10 | 2010-01-27 | ５−ヒドロキシメチル−オキサゾリジン−２−オン誘導体 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009535864A Expired - Fee Related JP4484965B2 (ja) | 2006-11-10 | 2007-11-09 | ５−ヒドロキシメチル−オキサゾリジン−２−オン誘導体 |
Country Status (27)
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003031443A1 (en) | 2001-10-04 | 2003-04-17 | Morphochem Aktiengesellschaft für kombinatorische Chemie | Dual actions antibiotics comprising a oxazoldinone and a quinolone or naphthyridinone moiety |
| US20070155714A1 (en) | 2003-04-30 | 2007-07-05 | Morphochem Aktiengesellschaft Fur Kombinatorische Chemie | Use of oxazolidinone-quinoline hybrid antibiotics for the treatment of anthrax and other infections |
| DE10340485B4 (de) | 2003-09-03 | 2015-05-13 | Morphochem AG Aktiengesellschaft für kombinatorische Chemie | Verfahren zur Herstellung von Oxazolidinon-Chinolon Hybriden |
| US8158797B2 (en) | 2003-12-18 | 2012-04-17 | Morphochem Aktiengesellschaft Fur Kombinatorische Chemie | Oxazolidinone-quinolone hybrid antibiotics |
| BRPI0417193B8 (pt) | 2003-12-18 | 2021-05-25 | Morphochem Ag Fuer Komb Chemie | antibióticos híbridos de oxazolidinona-quinolona, seus sais monossódicos, dissódicos ou trissódicos e seus pró-fármacos, composições farmacêuticas, e seu uso |
| US8124623B2 (en) | 2006-11-10 | 2012-02-28 | Actelion Pharmaceuticals Ltd. | 5-hydroxymethyl-oxazolidin-2-one-derivatives and their uses as antibacterials |
| AU2009245351B2 (en) * | 2008-05-09 | 2015-01-22 | Actelion Pharmaceuticals Ltd | 5-hydroxymethyl-oxazolidin-2-one derivatives for treating bacterial intestinal diseases |
| MX344529B (es) * | 2011-11-08 | 2016-12-19 | Actelion Pharmaceuticals Ltd | Derivados antibioticos de 2 - oxo -oxazolidin - 3, 5 -diilo. |
| CA2912728C (en) | 2013-05-28 | 2021-04-13 | Morphochem Aktiengesellschaft Fur Kombinatorische Chemie | Combination therapy comprising oxazolidinone-quinolones for use in treating bacterial infections |
| NZ713945A (en) | 2013-05-28 | 2020-05-29 | Morphochem Aktiengesellschaft Fuer Komb Chemie | Oxazolidinone-quinolone hybrid antibacterials for the parenteral treatment or prophylaxis of bacterial diseases |
| WO2016079757A2 (en) * | 2014-11-19 | 2016-05-26 | Symed Labs Limited | Novel processes for preparing 5-hydroxymethyl-oxazolidin-2-one derivatives |
| WO2017146246A1 (ja) * | 2016-02-26 | 2017-08-31 | 大塚製薬株式会社 | ピペリジン誘導体 |
| US10087171B2 (en) | 2016-12-19 | 2018-10-02 | Actelion Pharmaceuticals Ltd | Crystalline forms of cadazolid |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SU1156597A3 (ru) * | 1982-04-28 | 1985-05-15 | Е.И.Дюпон Де Немур Энд Компани (Фирма) | Способ получени производных 3-( @ -алкилсульфонилфенил)оксазолидинона или их фармацевтически приемлемых кислотно-аддитивных солей |
| US4461773A (en) * | 1982-09-15 | 1984-07-24 | E. I. Dupont De Nemours And Company | P-Oxooxazolidinylbenzene compounds as antibacterial agents |
| US6413981B1 (en) * | 1999-08-12 | 2002-07-02 | Ortho-Mcneil Pharamceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
| US6608081B2 (en) * | 1999-08-12 | 2003-08-19 | Ortho-Mcneil Pharmaceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
| CA2424402A1 (en) * | 2000-12-21 | 2002-08-01 | Pharmacia & Upjohn Company | Antimicrobial quinolone derivatives and use of the same to treat bacterial infections |
| AU2002256995A1 (en) * | 2001-02-07 | 2002-08-28 | Ortho-Mcneil Pharmaceutical, Inc. | Pyridoarylphenyl oxazolidinone antibacterials, and related compositions and methods |
| WO2003031443A1 (en) * | 2001-10-04 | 2003-04-17 | Morphochem Aktiengesellschaft für kombinatorische Chemie | Dual actions antibiotics comprising a oxazoldinone and a quinolone or naphthyridinone moiety |
| US20070155714A1 (en) * | 2003-04-30 | 2007-07-05 | Morphochem Aktiengesellschaft Fur Kombinatorische Chemie | Use of oxazolidinone-quinoline hybrid antibiotics for the treatment of anthrax and other infections |
| CN100544719C (zh) * | 2003-04-30 | 2009-09-30 | 莫弗凯姆联合化学股份公司 | 噁唑烷酮-喹啉杂化物抗生素用于制备治疗炭疽和其它感染的药物中的用途 |
| KR100854211B1 (ko) * | 2003-12-18 | 2008-08-26 | 동아제약주식회사 | 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물 |
| BRPI0417193B8 (pt) * | 2003-12-18 | 2021-05-25 | Morphochem Ag Fuer Komb Chemie | antibióticos híbridos de oxazolidinona-quinolona, seus sais monossódicos, dissódicos ou trissódicos e seus pró-fármacos, composições farmacêuticas, e seu uso |
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2007
- 2007-11-09 JP JP2009535864A patent/JP4484965B2/ja not_active Expired - Fee Related
- 2007-11-09 NZ NZ577538A patent/NZ577538A/en not_active IP Right Cessation
- 2007-11-09 PT PT07827038T patent/PT2086968E/pt unknown
- 2007-11-09 CN CN2007800418985A patent/CN101535305B/zh not_active Expired - Fee Related
- 2007-11-09 AT AT07827038T patent/ATE544764T1/de active
- 2007-11-09 CL CL200703232A patent/CL2007003232A1/es unknown
- 2007-11-09 DK DK07827038.6T patent/DK2086968T3/da active
- 2007-11-09 PL PL07827038T patent/PL2086968T3/pl unknown
- 2007-11-09 TW TW096142564A patent/TWI374138B/zh not_active IP Right Cessation
- 2007-11-09 MX MX2009004764A patent/MX2009004764A/es active IP Right Grant
- 2007-11-09 CA CA2668280A patent/CA2668280C/en active Active
- 2007-11-09 AU AU2007318901A patent/AU2007318901B2/en not_active Ceased
- 2007-11-09 HR HRP20120385TT patent/HRP20120385T1/hr unknown
- 2007-11-09 BR BRPI0718862A patent/BRPI0718862B8/pt not_active IP Right Cessation
- 2007-11-09 EP EP07827038A patent/EP2086968B1/en active Active
- 2007-11-09 WO PCT/IB2007/054557 patent/WO2008056335A1/en not_active Ceased
- 2007-11-09 ES ES07827038T patent/ES2380388T3/es active Active
- 2007-11-09 RU RU2009121812/04A patent/RU2453546C2/ru active
- 2007-11-09 SI SI200730902T patent/SI2086968T1/sl unknown
- 2007-11-09 MY MYPI20091893A patent/MY148847A/en unknown
- 2007-11-09 KR KR1020097010924A patent/KR101118402B1/ko not_active Expired - Fee Related
- 2007-11-12 AR ARP070105031A patent/AR063788A1/es active IP Right Grant
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2009
- 2009-05-07 IL IL198645A patent/IL198645A/en active IP Right Grant
- 2009-06-01 MA MA31939A patent/MA30960B1/fr unknown
- 2009-06-09 NO NO20092209A patent/NO344727B1/no unknown
- 2009-06-09 ZA ZA200904028A patent/ZA200904028B/xx unknown
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2010
- 2010-01-27 JP JP2010016076A patent/JP5490553B2/ja not_active Expired - Fee Related
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2012
- 2012-04-24 CY CY20121100383T patent/CY1112696T1/el unknown